The first of two tables displays the raw information used to construct POSEIDON. The second table corresponds to the processed data, in which only the usable samples were kept (the pre-processing steps are thoroughly described in the scientific paper.
This first table lists the literature-mined information used to generate the dataset for POSEIDON, comprising information on 2.371 peptide samples. However, please note that not all these peptides can be used in the same manner. This table informs on:
The values can be sorted by clicking on the arrows near the column names. The global search box on the top of the table can be used to query the entire table. Additionally, the search boxes on the footer of the table can be used to query the individual columns.
Peptide | Cell line | Cargo | PubmedID | Uptake | Units | Conc. | Time | Temp. | Method | Type | Sequence |
---|---|---|---|---|---|---|---|---|---|---|---|
Peptide | Cell line | Cargo | PubmedID | Uptake | Units | Conc. | Time | Temp. | Method | Type | Sequence |
Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 650 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRRR |
Tat (49-56) | Jurkat cells | Fluorescein | 11087855 | 31.25 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRR |
Tat (49-55) | Jurkat cells | Fluorescein | 11087855 | 10 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQR |
Tat (50-57) | Jurkat cells | Fluorescein | 11087855 | 22.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | KKRRQRRR |
Tat (51-57) | Jurkat cells | Fluorescein | 11087855 | 20 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | KRRQRRR |
D-Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 1800 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rkkrrqrrr |
Retro - Tat (57-49) | Jurkat cells | Fluorescein | 11087855 | 2450 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRQRRKKR |
D-Tat (57-49) | Jurkat cells | Fluorescein | 11087855 | 3600 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrqrrkkr |
Ala49 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 16.25 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | AKKRRQRRR |
Ala50 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 32.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RAKRRQRRR |
Ala51 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 37.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKARRQRRR |
Ala52 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 20 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKARQRRR |
Ala53 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 30 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRAQRRR |
Ala54 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 132.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRARRR |
Ala55 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 32.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQARR |
Ala56 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 35 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRAR |
Ala57 substitution mutant of Tat (49-57) | Jurkat cells | Fluorescein | 11087855 | 12.5 | Mean Fluorescence intensity | 12.5 uM | 10 min | 23ºC | Flow cytometry | Cellular uptake | RKKRRQRRA |
R5 | Jurkat cells | Fluorescein | 11087855 | 100 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRR |
R6 | Jurkat cells | Fluorescein | 11087855 | 500 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRR |
R7 | Jurkat cells | Fluorescein | 11087855 | 1225 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRR |
R8 | Jurkat cells | Fluorescein | 11087855 | 1700 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
R9 | Jurkat cells | Fluorescein | 11087855 | 2650 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
D-R5 | Jurkat cells | Fluorescein | 11087855 | 150 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrr |
D-R6 | Jurkat cells | Fluorescein | 11087855 | 950 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrr |
D-R7 | Jurkat cells | Fluorescein | 11087855 | 3100 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrr |
D-R8 | Jurkat cells | Fluorescein | 11087855 | 4400 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrrr |
D-R9 | Jurkat cells | Fluorescein | 11087855 | 5125 | Mean Fluorescence intensity | 12.5 uM | 15 min | 23ºC | Flow cytometry | Cellular uptake | rrrrrrrrr |
I | Aortic endothelial cells | Fluorescein | 10323198 | 228 ± 54 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAALKLA |
KLA1 | Aortic endothelial cells | nan | 10323198 | 161 ± 21 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKAWKAALKLA |
KLA2 | Aortic endothelial cells | nan | 10323198 | 15 ± 6 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKAALKAWKAAAKLA |
KLA3 | Aortic endothelial cells | nan | 10323198 | <10 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKAAAKAWKAAAKAA |
KLA11 | Aortic endothelial cells | nan | 10323198 | 47 ± 7 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KITLKLAIKAWKLALKAA |
KLA5 | Aortic endothelial cells | nan | 10323198 | 68 ± 2 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KIAAKSIAKIWKSILKIA |
KLA12 | Aortic endothelial cells | nan | 10323198 | 149 ± 20 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAKALAKLWKALAKAA |
KLA13 | Aortic endothelial cells | nan | 10323198 | 15 ± 4 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKWAKLALKAA |
KLA14 | Aortic endothelial cells | nan | 10323198 | 29 ± 14 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLLAKAAKKWLLLALKAA |
KLA9 | Aortic endothelial cells | nan | 10323198 | 44 ± 10 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLLAKAALKWLLKALKAA |
KLA10 | Aortic endothelial cells | nan | 10323198 | 218 ± 31 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALKKLLAKWLAAAKALL |
KLA15 | Aortic endothelial cells | nan | 10323198 | 226 ± 19 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLAAALLKKWKKLAAALL |
KLA8 | Aortic endothelial cells | Fluorescein | 10323198 | 341 ± 58 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAALLKKWAKLLAALK |
CPP-II | Aortic endothelial cells | Fluorescein | 10323198 | 371 ± 56 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KALAALLKKLAKLLAALK |
CPP-III | Aortic endothelial cells | Fluorescein | 10323198 | 218 ± 23 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAALK |
CPP-IV | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKALKAALKLA |
CPP-V | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALKAA |
CPP-VI | Aortic endothelial cells | Fluorescein | 10323198 | <30 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLGLKLGLKGLKGGLKLG |
CPP-VII | Aortic endothelial cells | Fluorescein | 10323198 | 42 ± 12.4 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALKLALKALQAALQLA |
CPP-VIII | Aortic endothelial cells | Fluorescein | 10323198 | 461 ± 44 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | KLALQLALQALQAALQLA |
CPP-IX | Aortic endothelial cells | Fluorescein | 10323198 | 5670 ± 3971 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | QLALQLALQALQAALQLA |
CPP-X | Aortic endothelial cells | Fluorescein | 10323198 | 135 ± 14.6 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | ELALELALEALEAALELA |
CPP-XI | Aortic endothelial cells | Fluorescein | 10323198 | 539 ± 80 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | LKTLATALTKLAKTLTTL |
CPP-XIII | Aortic endothelial cells | Fluorescein | 10323198 | 141 ± 54 | pmol internalized peptide / mg protein | 1.8 uM | 30 min | 37ºC | HPCL-analysis | Internalization | LKTLTETLKELTKTLTEL |
pAntpHD (43-58) | Cortical striatal cells | Biotin | 8663410 | 0.24 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQIKIWFQNRRMKWKK |
pAntpHD (58-43) | Cortical striatal cells | Biotin | 8663410 | 0.26 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | KKWKMRRNQFWIKIQR |
D form of pAntpHD (43-58) | Cortical striatal cells | Biotin | 8663410 | 0.45 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | rqikiwfqnrrmkwkk |
pAntpHD (Pro50) | Cortical striatal cells | Biotin | 8663410 | 0.88 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQIKIWFPNRRMKWKK |
pAntpHD (3Pro) | Cortical striatal cells | Biotin | 8663410 | 0.18 | OD (optical density values) | 44 uM | 2h | 4ºC | ELISA | Internalization | RQPKIWFPNRRKPWKK |
pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 100.0 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKK |
pAntp (43-57) | HaCaT cells | Biotin | 10784032 | 57 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWK |
pAntp (43-56) | HaCaT cells | Biotin | 10784032 | 47.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKW |
pAntp (43-55) | HaCaT cells | Biotin | 10784032 | 28 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMK |
pAntp (43-54) | HaCaT cells | Biotin | 10784032 | 19.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRM |
pAntp (43-53) | HaCaT cells | Biotin | 10784032 | 25 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRR |
pAntp (43-52) | HaCaT cells | Biotin | 10784032 | 15 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNR |
pAntp (43-51) | HaCaT cells | Biotin | 10784032 | 18 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQN |
pAntp (43-50) | HaCaT cells | Biotin | 10784032 | 13 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQ |
pAntp (43-48) | HaCaT cells | Biotin | 10784032 | 20 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIW |
pAntp (44-58) | HaCaT cells | Biotin | 10784032 | 87 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | QIKIWFQNRRMKWKK |
pAntp (45-58) | HaCaT cells | Biotin | 10784032 | 94 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | IKIWFQNRRMKWKK |
pAntp (46-58) | HaCaT cells | Biotin | 10784032 | 67 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | KIWFQNRRMKWKK |
pAntp (47-58) | HaCaT cells | Biotin | 10784032 | 48 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | IWFQNRRMKWKK |
pAntp (48-58) | HaCaT cells | Biotin | 10784032 | 52 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | WFQNRRMKWKK |
pAntp (49-58) | HaCaT cells | Biotin | 10784032 | 64 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | FQNRRMKWKK |
pAntp (50-58) | HaCaT cells | Biotin | 10784032 | 60 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | QNRRMKWKK |
pAntp (51-58) | HaCaT cells | Biotin | 10784032 | 60 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | NRRMKWKK |
pAntp (52-58) | HaCaT cells | Biotin | 10784032 | 50 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RRMKWKK |
pAntp (53-58) | HaCaT cells | Biotin | 10784032 | 22 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RMKWKK |
Ala43 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 89 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | AQIKIWFQNRRMKWKK |
Ala44 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 67 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RAIKIWFQNRRMKWKK |
Ala45 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 82 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQAKIWFQNRRMKWKK |
Ala46 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 52 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIAIWFQNRRMKWKK |
Ala47 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 56 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKAWFQNRRMKWKK |
Ala48 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 68 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIAFQNRRMKWKK |
Ala49 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 89.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWAQNRRMKWKK |
Ala50 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 90 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFANRRMKWKK |
Ala51 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 61 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQARRMKWKK |
Ala52 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 42 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNARMKWKK |
Ala53 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 31 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRAMKWKK |
Ala54 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 87.5 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRAKWKK |
Ala55 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 26 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMAWKK |
Ala56 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 41 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKAKK |
Ala57 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 21 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWAK |
Ala58 substitution mutant of pAntp (43-58) | HaCaT cells | Biotin | 10784032 | 23 | % Absorbance relative to peptide 1 (405 nm) | 40 uM | 60 min | nan | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKA |
Crot (27-39) | NIH-3T3 cells | FITC | 21319732 | 3176 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCCKK |
Crot (27-39) derevative 1 | NIH-3T3 cells | FITC | 21319732 | 3344 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKCCKK |
Crot (27-39) derevative 2 | NIH-3T3 cells | FITC | 21319732 | 1909 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKCCKK |
CyLoP-1 | NIH-3T3 cells | FITC | 21319732 | 4050 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCCKK |
Crot (27-39) derevative 3 | NIH-3T3 cells | FITC | 21319732 | 1511 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKCCKK |
Crot (27-39) derevative 4 | NIH-3T3 cells | FITC | 21319732 | 1516 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCKK |
Crot (27-39) derevative 5 | NIH-3T3 cells | FITC | 21319732 | 1202 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKKK |
Crot (27-39) derevative 6 | NIH-3T3 cells | FITC | 21319732 | 100 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDRWRWKKK |
Crot (27-39) derevative 7 | NIH-3T3 cells | FITC | 21319732 | 1043 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KDCRWRWKCCKK |
Crot (27-39) derevative 8 | NIH-3T3 cells | FITC | 21319732 | 1583 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCRWRWKCCKK |
Crot (27-39) derevative 9 | NIH-3T3 cells | FITC | 21319732 | 1226 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRWRWKCCKK |
Crot (27-39) derevative 10 | NIH-3T3 cells | FITC | 21319732 | 1937 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKXCKK |
Crot (27-39) derevative 11 | NIH-3T3 cells | FITC | 21319732 | 1741 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKXCKK |
Crot (27-39) derevative 12 | NIH-3T3 cells | FITC | 21319732 | 943 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKCXKK |
Crot (27-39) derevative 13 | NIH-3T3 cells | FITC | 21319732 | 2044 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKXCKK |
Crot (27-39) derevative 14 | NIH-3T3 cells | FITC | 21319732 | 1347 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCXKK |
Crot (27-39) derevative 15 | NIH-3T3 cells | FITC | 21319732 | 1211 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKXCKK |
Crot (27-39) derevative 16 | NIH-3T3 cells | FITC | 21319732 | 1256 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKXXKK |
Crot (27-39) derevative 17 | NIH-3T3 cells | FITC | 21319732 | 872 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | DCRWRWKXXKK |
Crot (27-39) derevative 18 | NIH-3T3 cells | FITC | 21319732 | 1390 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKXXKK |
Crot (27-39) derevative 19 | NIH-3T3 cells | FITC | 21319732 | 405 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RWRWKXXKK |
Crot (27-39) derevative 20 | NIH-3T3 cells | FITC | 21319732 | 2172 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCSKK |
Crot (27-39) derevative 21 | NIH-3T3 cells | FITC | 21319732 | 1867 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKCCKK |
Crot (27-39) derevative 22 | NIH-3T3 cells | FITC | 21319732 | 572 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKCSKK |
Crot (27-39) derevative 23 | NIH-3T3 cells | FITC | 21319732 | 475 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKSCKK |
Crot (27-39) derevative 24 | NIH-3T3 cells | FITC | 21319732 | 415 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKSSKK |
Crot (27-39) derevative 25 | NIH-3T3 cells | FITC | 21319732 | 193 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | SRWRWKSSKK |
Crot (27-39) derevative 26 | NIH-3T3 cells | FITC | 21319732 | 2656 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRFRWKCCKK |
Crot (27-39) derevative 27 | NIH-3T3 cells | FITC | 21319732 | 2476 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRFKCCKK |
Crot (27-39) derevative 28 | NIH-3T3 cells | FITC | 21319732 | 2569 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRFRFKCCKK |
Crot (27-39) derevative 29 | NIH-3T3 cells | FITC | 21319732 | 2109 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | crwrwkcckk |
Crot (27-39) derevative 30 | NIH-3T3 cells | FITC | 21319732 | 1713 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCCKWRWRCK |
Crot (27-39) derevative 31 | NIH-3T3 cells | FITC | 21319732 | 1449 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | kcckwrwrck |
Crot (27-39) derevative 32 | NIH-3T3 cells | FITC | 21319732 | 1529 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CrWRWKCCKK |
Crot (27-39) derevative 33 | NIH-3T3 cells | FITC | 21319732 | 1229 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRwRWKCCKK |
Crot (27-39) derevative 34 | NIH-3T3 cells | FITC | 21319732 | 1304 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWrWKCCKK |
Crot (27-39) derevative 35 | NIH-3T3 cells | FITC | 21319732 | 1412 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRwKCCKK |
Crot (27-39) derevative 36 | NIH-3T3 cells | FITC | 21319732 | 1488 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CrwrwKCCKK |
Crot (27-39) derevative 37 | NIH-3T3 cells | FITC | 21319732 | 2376 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCGCKK |
Crot (27-39) derevative 38 | NIH-3T3 cells | FITC | 21319732 | 3056 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KCGCRWRWKCGCKK |
Crot (27-39) derevative 39 | NIH-3T3 cells | FITC | 21319732 | 1922 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | CRWRWKCG |
Crot (27-39) derevative 40 | NIH-3T3 cells | FITC | 21319732 | 1943 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKCCKK |
Crot (27-39) derevative 41 | NIH-3T3 cells | FITC | 21319732 | 734 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKXCKK |
Crot (27-39) derevative 42 | NIH-3T3 cells | FITC | 21319732 | 162 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKXXKK |
Crot (27-39) derevative 43 | NIH-3T3 cells | FITC | 21319732 | 2816 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRWRWKCXKK |
Crot (27-39) derevative 44 | NIH-3T3 cells | FITC | 21319732 | 1542 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | MDCRWRWKCXKK |
Crot (27-39) derevative 45 | NIH-3T3 cells | FITC | 21319732 | 2335 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKCSKK |
Crot (27-39) derevative 46 | NIH-3T3 cells | FITC | 21319732 | 1188 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKSCKK |
Crot (27-39) derevative 47 | NIH-3T3 cells | FITC | 21319732 | 987 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKCCKK |
Crot (27-39) derevative 48 | NIH-3T3 cells | FITC | 21319732 | 615 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRWKSSKK |
Crot (27-39) derevative 49 | NIH-3T3 cells | FITC | 21319732 | 496 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKSSKK |
Crot (27-39) derevative 50 | NIH-3T3 cells | FITC | 21319732 | 856 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKSCKK |
Crot (27-39) derevative 51 | NIH-3T3 cells | FITC | 21319732 | 1244 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDSRWRWKCSKK |
Crot (27-39) derevative 52 | NIH-3T3 cells | FITC | 21319732 | 1272 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRWRPKCCKK |
Crot (27-39) derevative 53 | NIH-3T3 cells | FITC | 21319732 | 347 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKCCKK |
Crot (27-39) derevative 54 | NIH-3T3 cells | FITC | 21319732 | 251 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKCCKK |
Crot (27-39) derevative 55 | NIH-3T3 cells | FITC | 21319732 | 222 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKXCKK |
Crot (27-39) derevative 56 | NIH-3T3 cells | FITC | 21319732 | 257 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDXRPRPKCXKK |
Crot (27-39) derevative 57 | NIH-3T3 cells | FITC | 21319732 | 294 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKXCKK |
Crot (27-39) derevative 58 | NIH-3T3 cells | FITC | 21319732 | 353 | Mean Fluorescence intensity | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KMDCRPRPKCXKK |
Penetratin (pAntp) | NIH-3T3 cells | FITC | 21319732 | 27.5 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | RQIKIWFQNRRMKWKK |
Tat (49-57) | NIH-3T3 cells | FITC | 21319732 | 55.0 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rkkrrqrrr |
Tat (57-49) | NIH-3T3 cells | FITC | 21319732 | 46.25 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rrrqrrkkr |
R8 | NIH-3T3 cells | FITC | 21319732 | 47.5 | % Intracellular fluorescence of CyLoP-1 | 2.5 uM | 18h | 37ºC | Fluorescence spectroscopy | Cellular uptake | rrrrrrrr |
DPV3 | HeLa cells | PO, IgG | 15859953 | 176 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | RKKRRRESRKKRRRES |
DPV3 | HCT116 cells | PO, IgG | 15859953 | 168 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | RKKRRRESRKKRRRES |
DPV3 | K562 cells | PO, IgG | 15859953 | 36 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | RKKRRRESRKKRRRES |
DPV1047 | HeLa cells | PO, IgG | 15859953 | 24 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | VKRGLKLRHVRPRVTRMDV |
DPV1047 | HCT116 cells | PO, IgG | 15859953 | 20 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | VKRGLKLRHVRPRVTRMDV |
DPV1047 | K562 cells | PO, IgG | 15859953 | 180 | pg PO/ 1000 cells | 1 mg/mL | 4h | 37ºC | Confocal laser scanning system (clss) | Internalization | VKRGLKLRHVRPRVTRMDV |
Bip1 | DAMI cells | Fluorescein | 21359136 | 97± 4.3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPMLK |
Bip2 | DAMI cells | Fluorescein | 21359136 | 61±1.7 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPTLK |
Bip2 | HeLa cells | Fluorescein | 21359136 | 1280 | Mean Fluorescence intensity | 1600 uM | 3h | nan | FACS | Cell-Penetration | VPTLK |
Bip3 | DAMI cells | Fluorescein | 21359136 | 79 ± 1.5 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPALR |
Bip4 | DAMI cells | Fluorescein | 21359136 | 90 ± 3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VSALK |
Bip5 | DAMI cells | Fluorescein | 21359136 | 65 ± 3.7 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | PMLKE |
Bip6 | DAMI cells | Fluorescein | 21359136 | 71 ± 2.2 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPALK |
Bip9 | DAMI cells | Fluorescein | 21359136 | 100 ± 2.3 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | KLPVM |
Bip10 | DAMI cells | Fluorescein | 21359136 | 47 ± 1.4 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | IPMIK |
Bip16 | DAMI cells | Fluorescein | 21359136 | 70 ± 4 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPTLQ |
Bip19 | DAMI cells | Fluorescein | 21359136 | 80±1.9 | Cellular uptake (%) | 200 uM | 3h | 37ºC | FACS | Cell-Penetration | VPTLE |
Inv1 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 47.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | VNADIKATTVFGGKYVSLTTP |
Inv2 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 104.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | GKYVSLTTPKNPTKRRITPKDV |
Inv3 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 607.5 / 2400 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTEINT |
Inv4 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 104.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | RSVTTEINTLFQTLTSIAEKVDP |
Inv5 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 626.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | AEKVDPVKLNLTLSAAAEALTGLGDK |
Inv6 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 155 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | GLGDKFGESIVNANTVLDDLNSRMPQSRHDIQQL |
Inv7 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 57 / 75 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | GDVYADAAPDLFDFLDSSVTTARTINA |
Inv8 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 47.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | ARTINAQQAELDSALLAAAGFGNTTADVFDRG |
Inv9 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 76 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | ADVFDRGGPYLQRGVADLVPTATLLDTYSP |
Inv10 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 33.25 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | LDTYSPELFCTIRNFYDADRPDRGAAA |
Inv11 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 123.5 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTEINT |
Inv3.3 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 50 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPDDVIDVRSVTTEINT |
Inv3.4 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 1200 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKKVIDVRSVTTEINT |
Inv3.5 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 2650 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVRSVTTKINT |
Inv3.6 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 50 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDV |
Inv3.7 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 75 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKRRITPKDVIDVESVTTEINT |
Inv3.8 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 150 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TARRITPKDVIDVRSVTTEINT |
Inv3.9 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 100 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | TKAARITPKDVIDVRSVTTEINT |
Inv3.10 | HeLa cells | (FITC)-labeled latex microspheres | 16620748 | 1925 | Fluorescence intensity | 0.05 umol | nan | 37ºC | Flow cytometry | Uptake | HHHHHHTKRRITPKDVIDVRSVTTEINT |
No.14 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSPTTRRYG |
No.14-1 | CHO cells | Fluorescein | 19956900 | 650 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRYG |
No.14-2 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSATTRRYG |
No.14-7 | CHO cells | Fluorescein | 19956900 | 850 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | KLWMRWYSPWTRRYG |
No.14-8 | CHO cells | Fluorescein | 19956900 | 650 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPWTRRYG |
No.14-9 | CHO cells | Fluorescein | 19956900 | 530 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPWTRRWG |
No.14-11 | CHO cells | Fluorescein | 19956900 | 220 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | ALWMRWYSPTTRRYG |
No.14-12 | CHO cells | Fluorescein | 19956900 | 800 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RAWMRWYSPTTRRYG |
No.14-13 | CHO cells | Fluorescein | 19956900 | 750 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLAMRWYSPTTRRYG |
No.14-14 | CHO cells | Fluorescein | 19956900 | 750 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWARWYSPTTRRYG |
No.14-15 | CHO cells | Fluorescein | 19956900 | 90 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMAWYSPTTRRYG |
No.14-16 | CHO cells | Fluorescein | 19956900 | 50 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRAYSPTTRRYG |
No.14-17 | CHO cells | Fluorescein | 19956900 | 790 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWASPTTRRYG |
No.14-18 | CHO cells | Fluorescein | 19956900 | 800 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYAPTTRRYG |
No.14-20 | CHO cells | Fluorescein | 19956900 | 880 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPATRRYG |
No.14-21 | CHO cells | Fluorescein | 19956900 | 810 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTARRYG |
No.14-22 | CHO cells | Fluorescein | 19956900 | 370 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTARYG |
No.14-3R | CHO cells | Fluorescein | 19956900 | 150 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRAYG |
No.14-23 | CHO cells | Fluorescein | 19956900 | 840 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRAG |
No.14-35 | CHO cells | Fluorescein | 19956900 | 860 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLWMRWYSPTTRRYA |
No.14-24 | CHO cells | Fluorescein | 19956900 | 440 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLLMRLYSPTTRRYG |
No.14-25 | CHO cells | Fluorescein | 19956900 | 830 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLFMRFYSPTTRRYG |
No.14-26 | CHO cells | Fluorescein | 19956900 | 860 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLIMRIYSPTTRRYG |
No.14-29 | CHO cells | Fluorescein | 19956900 | 590 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLVMRVYSPTTRRYG |
No.14-30 | CHO cells | Fluorescein | 19956900 | 890 | Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Translocation | RLYMRYYSPTTRRYG |
pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 1350 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHSK |
pVEC mutant 1 | Human bowes melanoma cells | Fluorescein | 16808894 | 300 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | ALIILRRRIRKQAHAHSK |
pVEC mutant 2 | Human bowes melanoma cells | Fluorescein | 16808894 | 500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LAIILRRRIRKQAHAHSK |
pVEC mutant 3 | Human bowes melanoma cells | Fluorescein | 16808894 | 375 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLAILRRRIRKQAHAHSK |
pVEC mutant 4 | Human bowes melanoma cells | Fluorescein | 16808894 | 700 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIALRRRIRKQAHAHSK |
pVEC mutant 5 | Human bowes melanoma cells | Fluorescein | 16808894 | 450 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIIARRRIRKQAHAHSK |
pVEC mutant 6 | Human bowes melanoma cells | Fluorescein | 16808894 | 2500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILARRIRKQAHAHSK |
pVEC mutant 7 | Human bowes melanoma cells | Fluorescein | 16808894 | 1125 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRARIRKQAHAHSK |
pVEC mutant 8 | Human bowes melanoma cells | Fluorescein | 16808894 | 2175 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRAIRKQAHAHSK |
pVEC mutant 9 | Human bowes melanoma cells | Fluorescein | 16808894 | 800 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRARKQAHAHSK |
pVEC mutant 10 | Human bowes melanoma cells | Fluorescein | 16808894 | 1500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIARKQAHAHSK |
pVEC mutant 11 | Human bowes melanoma cells | Fluorescein | 16808894 | 1800 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRAQAHAHSK |
pVEC mutant 12 | Human bowes melanoma cells | Fluorescein | 16808894 | 1500 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKAAHAHSK |
pVEC mutant 13 | Human bowes melanoma cells | Fluorescein | 16808894 | 1850 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQaHAHSK |
pVEC mutant 14 | Human bowes melanoma cells | Fluorescein | 16808894 | 550 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAAAHSK |
pVEC mutant 15 | Human bowes melanoma cells | Fluorescein | 16808894 | 1125 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHaHSK |
pVEC mutant 16 | Human bowes melanoma cells | Fluorescein | 16808894 | 1550 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAASK |
pVEC mutant 17 | Human bowes melanoma cells | Fluorescein | 16808894 | 2150 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHAK |
pVEC mutant 18 | Human bowes melanoma cells | Fluorescein | 16808894 | 2100 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | LLIILRRRIRKQAHAHSA |
Retro-pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 400 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KSHAHAQKRIRRRLIILL |
D form of pVEC | Human bowes melanoma cells | Fluorescein | 16808894 | 1150 | pmol/mg protein Cellular uptake | 10 uM | 1h | 37ºC | Fluorescence spectroscopy | Uptake | lliilrrrirkqahahsk |
Bac1-7 | RAW264.7 cells | Fluorescein | 12450378 | 90 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRP |
Bac-1-15 | RAW264.7 cells | Fluorescein | 12450378 | 200 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRP |
Bac1-24 | RAW264.7 cells | Fluorescein | 12450378 | 35 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRPRPLPFPRPG |
Bac1-17 | RAW264.7 cells | Fluorescein | 12450378 | 130 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RRIRPRPPRLPRPRPRP |
Bac5-24 | RAW264.7 cells | Fluorescein | 12450378 | 60 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPPRLPRPRPRPLPFPRPG |
Bac7-24 | RAW264.7 cells | Fluorescein | 12450378 | 90 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PPRLPRPRPRPLPFPRPG |
Bac9-24 | RAW264.7 cells | Fluorescein | 12450378 | 100 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | RLPRPRPRPLPFPRPG |
Bac13-24 | RAW264.7 cells | Fluorescein | 12450378 | 80 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPRPLPFPRPG |
Bac15-24 | RAW264.7 cells | Fluorescein | 12450378 | 555 | Intracellular Fluorescence | 5 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | PRPLPFPRPG |
ARF(1-22) | MCF7 cells | Fluorescein | 17984975 | 1300 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | MVRRFLVTLRIRRACGPPRVRV |
ARF(1-22) scr | MCF7 cells | Fluorescein | 17984975 | 1000 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | FVTRGCPRRLVARLIRVMVPRR |
ARF(2-14) | MCF7 cells | Fluorescein | 17984975 | 750 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | VRRFLVTLRIRRA |
ARF(2-14) scr | MCF7 cells | Fluorescein | 17984975 | 150 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | RVRILARFLRTRV |
ARF(19-31) | MCF7 cells | Fluorescein | 17984975 | 1050 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | RVRVFVVHIPRLT |
ARF(19-31) scr | MCF7 cells | Fluorescein | 17984975 | 250 | pmol/mg protein Cellular uptake | 5 umol/L | 1h | nan | Fluorescence spectroscopy | Uptake | VIRVHFRLPVRTV |
Cyt C 71-101 | U373 MG cells | nan | 20659686 | 100 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | GTKMIFVGIKKKEERADLIAYLKKA |
Cyt C 86-101 | U373 MG cells | nan | 20659686 | 4 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KKKEERADLIAYLKKA |
Cyt 79-92 | U373 MG cells | nan | 20659686 | 8 | Fluorescence (fold/basal) | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KMIFVGIKKKEERA |
Cyt 79-88 | U373 MG cells | nan | 20659686 | 4.5 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KMIFVGIKKK |
Cyt 4-13 | U373 MG cells | nan | 20659686 | 7 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | EKGKKIFIMK |
Cyt 5-13 | U373 MG cells | nan | 20659686 | 41 | Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | KGKKIFIMK |
hLF peptide | HeLa cells | Fluorescein | 19858187 | 40 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
M1 | HeLa cells | Fluorescein | 19858187 | 33.75 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSC |
M2 | HeLa cells | Fluorescein | 19858187 | 7.5 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSSIKR |
M3 | HeLa cells | Fluorescein | 19858187 | 6.25 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | KCFQWQRNMRKVR |
M4 | HeLa cells | Fluorescein | 19858187 | 4.375 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | FQWQRNMRKVRGPPVS |
M5 | HeLa cells | Fluorescein | 19858187 | 7.5 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | QWQRNMRKVRGPPVSCIKR |
M6 | HeLa cells | Fluorescein | 19858187 | 3.75 | Fluorescence intensity | 10 uM | 30 min | nan | Flow cytometry | Uptake | QWQRNMRKVR |
MPG Mutant | HS-68 | Fluorescein | 12771197 | 70 | Fluorescence intensity (%) | Charge ratio = 5:1 (MPG/DNA) | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
MPG Mutant | Cos-7 cells | Fluorescein | 12771197 | 5 | Fluorescence intensity (%) | Charge ratio = 10:1 | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
MPG Mutant | HeLa cells | Fluorescein | 12771197 | 10 | Fluorescence intensity (%) | Charge ratio = 10:1 | 30 min | 37ºC | Fluorescent Microscopy | Transfection | GALFLGFLGAAGSTMGAWSQPKSKRKV |
Sweet Arrow Protein (SAP) (E) | HeLa cells | Fluorescein | 21365733 | 11.15 | Fluorescence intensity | 50 uM | 3h | 37ºC | Flow cytometry | Cellular internalization | VELPPPVELPPPVELPPP |
Sweet Arrow Protein (SAP) (E) | A549 cells | Fluorescein | 21365733 | 5 | Fluorescence intensity | 50 uM | 3h | 37ºC | Flow cytometry | Cellular internalization | VELPPPVELPPPVELPPP |
Glu-Oct-6 | DU-145 | FITC | 21029412 | 600 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAAGRKRKKRT |
Glu | DU-145 | FITC | 21029412 | 140 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEE |
Glu-Ala | DU-145 | FITC | 21029412 | 120 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAA |
Glu-Lys | DU-145 | FITC | 21029412 | 280 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | EEEAAKKK |
6-Oct | DU-145 | FITC | 21029412 | 580 | Geo Mean Fluorescence intensity | 300 uM | 4h | 37ºC | Flow cytometry | Uptake | GRKRKKRT |
Phe-Oct-6 | DU-145 | FITC | 21029412 | 100 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | FFFAAGRKRKKRT |
Asn-Oct-6 | DU-145 | FITC | 21029412 | 55 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | NNNAAGRKRKKRT |
Tyr-Oct-6 | DU-145 | FITC | 21029412 | 115 | Geo Mean Fluorescence intensity | 300 uM | 1h | 37ºC | Flow cytometry | Uptake | YYYAAGRKRKKRT |
M918 | HeLa cells | Fluorescein | 17622242 | 3400 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | nan | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
M918 | MCF7 cells | Fluorescein | 17622242 | 1700 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | nan | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
M918 | Hifko cells | Fluorescein | 17622242 | 2700 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | nan | Fluorescence spectroscopy | Internalization | MVTVLFRRLRIRRACGPPRVRV |
TP10 | HeLa cells | Fluorescein | 17622242 | 1000 | pmol/mg protein Cellular uptake | 5 umol/l | 1h | nan | Fluorescence spectroscopy | Internalization | AGYLLGKINLKALAALAKKIL |
NF-kB | MCF7 cells | Fluorescein | 12204694 | 4 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | VQRKRQKLMP |
TFIIE BETA | MCF7 cells | Fluorescein | 12204694 | 5 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | SKKKKTKV |
6-Oct | MCF7 cells | Fluorescein | 12204694 | 14 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | GRKRKKRT |
TCF1-ALPHA | MCF7 cells | Fluorescein | 12204694 | 7 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | GKKKKRKREKL |
SV40 | MCF7 cells | Fluorescein | 12204694 | 3 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | PKKKRKV |
HATF3 | MCF7 cells | Fluorescein | 12204694 | 4 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | ERKKRRRE |
C.e SDC3 | MCF7 cells | Fluorescein | 12204694 | 2.8 | Mnlog FITC | 50 uM | 4h | nan | Flow cytometry | Cellular uptake | FKKFRKF |
SynB1 | K562 cells | NBD, TAMRA | 12783857 | 7 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | RGGRLSYSRRRFSTSTGR |
D-SynB1 | K562 cells | NBD | 12783857 | 7.5 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | rggrlsysrrrfststgr |
SynB3 | K562 cells | NBD, TAMRA | 12783857 | 16 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | RRLSYSRRRF |
D-SynB3 | K562 cells | NBD | 12783857 | 17.5 | Fluorescence intensity | 6 uM | 65 min | 37ºC | Flow cytometry | Internalization | rrlsysrrrf |
SynB5 | K562 cells | NBD, TAMRA | 12783857 | 62.5 | Fluorescence intensity | 3 uM | 65 min | 37ºC | Flow cytometry | Internalization | RGGRLAYLRRRWAVLGR |
MG2d | HeLa cells | Texas Red | 12417587 | 16 | nmol/mg protein | 15 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | GIGKFLHSAKKWGKAFVGQIMNC |
BF2d | HeLa cells | Texas Red | 12417587 | 1.5 | nmol/mg protein | 15 uM | 30 min | 37ºC | Fluorescence spectroscopy | Uptake | TRSSRAGLQWPVGRVHRLLRKGGC |
PolyP 1 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPP |
PolyP 2 | HeLa cells | Fluorescein | 15054781 | 100 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPPVRLPPP |
PolyP 3 (SAP) | HeLa cells | Fluorescein | 15054781 | 575 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VRLPPPVRLPPPVRLPPP |
PolyP 4 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPP |
PolyP 5 | HeLa cells | Fluorescein | 15054781 | 10 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPPVHLPPP |
PolyP 6 | HeLa cells | Fluorescein | 15054781 | 160 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VHLPPPVHLPPPVHLPPP |
PolyP 7 | HeLa cells | Fluorescein | 15054781 | 0 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPP |
PolyP 8 | HeLa cells | Fluorescein | 15054781 | 200 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPPVKLPPP |
PolyP 9 | HeLa cells | Fluorescein | 15054781 | 230 | Fluorescence intensity | 50 uM | 3h | 37ºC | Fluorescent Microscopy | Cellular uptake | VKLPPPVKLPPPVKLPPP |
hClock-(35-47) | ECV304 cells | FITC | 15346201 | 74 | Mean Fluorescence intensity | 4 uM | 1h | 37ºC | Fluorescent Microscopy | Internalization | KRVSRNKSEKKRR |
Penetratin {pAntp-(43-58)} | CHO-K1 cells | Rho | 15937518 | 21.25 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKK |
Penetratin {pAntp-(43-58)} | HeLa cells | Rho | 15937518 | 3.13 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKK |
Penetratin {pAntp-(43-58)} | A549 cells | Rho | 15937518 | 2.29 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKK |
pAntpƒ-PKI | CHO-K1 cells | Rho | 15937518 | 21.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
pAntpƒ-PKI | HeLa cells | Rho | 15937518 | 8.13 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
pAntpƒ-PKI | A549 cells | Rho | 15937518 | 4.16 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
Tat | CHO-K1 cells | Rho | 15937518 | 3.54 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQ |
Tat | HeLa cells | Rho | 15937518 | 1.83 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQ |
Tat | A549 cells | Rho | 15937518 | 1.68 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQ |
Tat-PKI | CHO-K1 cells | Rho | 15937518 | 5.41 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
Tat-PKI | HeLa cells | Rho | 15937518 | 2.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
Tat-PKI | A549 cells | Rho | 15937518 | 1.84 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
Transportan | CHO-K1 cells | Rho | 15937518 | 2 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKIL |
Transportan | HeLa cells | Rho | 15937518 | 1.6 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKIL |
Transportan | A549 cells | Rho | 15937518 | 1 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKIL |
Transportan-PKI | CHO-K1 cells | Rho | 15937518 | 18 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
Transportan-PKI | HeLa cells | Rho | 15937518 | 15.6 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
Transportan-PKI | A549 cells | Rho | 15937518 | 9 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
R11 | CHO-K1 cells | Rho | 15937518 | 31.16 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRR |
R11 | HeLa cells | Rho | 15937518 | 43.93 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRR |
R11 | A549 cells | Rho | 15937518 | 12.12 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRR |
R11-PKI | CHO-K1 cells | Rho | 15937518 | 7.5 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
R11-PKI | HeLa cells | Rho | 15937518 | 6.06 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
R11-PKI | A549 cells | Rho | 15937518 | 3.63 | Fold Change in GeoMean Fluorescence of control sample | 5 uM | 30 min | nan | FACS | Uptake | RRRRRRRRRRRTYADFIASGRTGRRNAI |
R9 | HeLa cells | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
R9 | MC57 | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
R9 | Jurkat cells | Fluorescein | 21867915 | 100.0 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | RRRRRRRRR |
r9 | HeLa cells | Fluorescein | 21867915 | 53.13 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
r9 | MC57 | Fluorescein | 21867915 | 46.87 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
r9 | Jurkat cells | Fluorescein | 21867915 | 90.62 | Cellular uptake (%) | 5 uM | 45 min | 37ºC | FCS | Uptake | rrrrrrrrr |
MAP | A549 cells | Fluorescein | 21875799 | 15 | Mean Fluorescence intensity/mg protein | 2 uM | 6h | 37ºC | Fluorescence spectroscopy | Internalization | KLALKLALKALKAALKLAGC |
MAP (Aib) | A549 cells | Fluorescein | 21875799 | 160 | Mean Fluorescence intensity/mg protein | 2 uM | 6h | 37ºC | Fluorescence spectroscopy | Internalization | KLULKLULKULKAULKLUGC |
HIV-1 Rev (34-50) | CHO-K1 cells | Alexa488 | 19707187 | 6.6 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRQARRNRRRRWRERQRGC |
HIV-1 Rev (34-50) | HeLa cells | Alexa488 | 19707187 | 6.0 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRQARRNRRRRWRERQRGC |
HIV-1 Rev (34-50) | Jurkat cells | Alexa488 | 19707187 | 2.5 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRQARRNRRRRWRERQRGC |
FHV coat (35-49) | CHO-K1 cells | Alexa488 | 19707187 | 21.1 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | RRRRNRTRRNRRRVRGC |
FHV coat (35-49) | HeLa cells | Alexa488 | 19707187 | 16.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | RRRRNRTRRNRRRVRGC |
FHV coat (35-49) | Jurkat cells | Alexa488 | 19707187 | 15.9 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | RRRRNRTRRNRRRVRGC |
BMV Gag (7-25) | CHO-K1 cells | Alexa488 | 19707187 | 1.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KMTRAQRRAAARRNRWTARGC |
BMV Gag (7-25) | HeLa cells | Alexa488 | 19707187 | 1.3 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KMTRAQRRAAARRNRWTARGC |
BMV Gag (7-25) | Jurkat cells | Alexa488 | 19707187 | 1.6 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KMTRAQRRAAARRNRWTARGC |
HTLV-II Rex (4-16) | CHO-K1 cells | Alexa488 | 19707187 | 1.3 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRRQRTRRARRNRGC |
HTLV-II Rex (4-16) | HeLa cells | Alexa488 | 19707187 | 1.2 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRRQRTRRARRNRGC |
HTLV-II Rex (4-16) | Jurkat cells | Alexa488 | 19707187 | 1.8 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | TRRQRTRRARRNRGC |
Human cJun (252-279) | CHO-K1 cells | Alexa488 | 19707187 | 14.4 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | FACS | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
Human cJun (252-279) | HeLa cells | Alexa488 | 19707187 | 12.4 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | FACS | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
Human cJun (252-279) | Jurkat cells | Alexa488 | 19707187 | 10.5 | Relative Cellular uptake | 5 umol/L | 30 min | 37ºC | FACS | Uptake | RIKAERKRMRNRIAASKSRKRKLERIARGC |
Human cFos (139-164) | CHO-K1 cells | Alexa488 | 19707187 | 0.9 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
Human cFos (139-164) | HeLa cells | Alexa488 | 19707187 | 0.8 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
Human cFos (139-164) | Jurkat cells | Alexa488 | 19707187 | 1.0 | Relative Cellular uptake | 5 umol/L | 30 min. | 37ºC | FACS | Uptake | KRRIRRERNKMAAAKSRNRRRELTDTGC |
cTat | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 1.68 | % Amount transported into basolateral fluid | nan | 2h | 37ºC | Gamma-well counter | Absorption | crkkrrqrrr |
cr9 | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 2.46 | % Amount transported into basolateral fluid | nan | 2h | 37ºC | Gamma-well counter | Absorption | crrrrrrrrr |
ck9 | Rat alveolar epithelial cell monolayers (RAECM) | Insulin | 19228019 | 0.38 | % Amount transported into basolateral fluid | nan | 2h | 37ºC | Gamma-well counter | Absorption | ckkkkkkkkk |
(RW)4 | SK-OV-3 cells | Doxorubicin | 23301519 | 31 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
cyclic [W(RW)4] | SK-OV-3 cells | Doxorubicin | 23301519 | 81 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WRWKKKKA |
NF51 | CHO cells | Plasmid DNA, SCO, siRNA | 23357356 | 1,00E+10 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | HEK293 cells | Plasmid DNA, SCO, siRNA | 23357356 | 1,00E+06 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | U2OS cells | Plasmid DNA, SCO, siRNA | 23357356 | 5.45E8 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | U87 cells | Plasmid DNA, SCO, siRNA | 23357356 | 7.78E7 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | MEF cells | Plasmid DNA, SCO, siRNA | 23357356 | 1.81E6 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | Jurkat cells | Plasmid DNA, SCO, siRNA | 23357356 | 3.63E4 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF51 | A20 cells | Plasmid DNA, SCO, siRNA | 23357356 | 7.27E2 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGOINLKALAALAKKIL |
NF53 | CHO cells | Plasmid DNA, SCO, siRNA | 23357356 | 1.17E2 | RFU/mg | 1.5 uM | 4h | nan | Fluorescent Microscopy | Transfection | AGYLLGKINLKALAALAKKIL |
PA 2 | PPC-1 | Rho | 23349939 | 6 | pmol/ug total protein | nan | nan | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
PA 2 | M21 | Rho | 23349939 | 7.1 | pmol/ug total protein | nan | nan | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
PA 3 | PPC-1 | Rho | 23349939 | 5 | pmol/ug total protein | nan | nan | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
PA 4 | PPC-1 | DSP-PEG2000, Rho | 23349939 | 4 | pmol/ug total protein | nan | nan | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
PA 5 | PPC-1 | DSP-PEG2000, Rho | 23349939 | 3 | pmol/ug total protein | nan | nan | 37ºC | Fluorescence spectroscopy | Association | RPARPAR |
FP-lipo | Human keratinocyte (HaCaT) cell | Liposome, folic acid | 23515421 | 54 | Fluorescence intensity | 500 uM as lipid concentration | 4h | 37ºC | Fluorescence spectroscopy | Uptake | KETWWETWWTEWSQPKKKRKVC |
FP-lipo | HeLa cells | Liposome, folic acid | 23515421 | 157 | Fluorescence intensity | 500 uM as lipid concentration | 4h | 37ºC | Fluorescence spectroscopy | Uptake | KETWWETWWTEWSQPKKKRKVC |
R5 | A549 cells | pDNA | 23534410 | 1,00E+04 | RFU/mg | 10 N/P (CaCl2 100 mM) | 52h | nan | Fluorescent Microscopy | Transfection | RRRRR |
R7 | A549 cells | pDNA | 23534410 | 1,00E+07 | RFU/mg | 10 N/P (CaCl2 100 mM) | 52h | nan | Fluorescent Microscopy | Transfection | RRRRRRR |
6xHis-TAT-SOD | HeLa cells | Cu,Zn-superoxide dismutase | 23289802 | 90 | Cellular uptake (%) | nan | 1h | 37ºC | FACS | Uptake | YGRKKRRQRRR |
Ypep-GFP | Human prostate adenocarcinoma cells (PC-3) | eGFP, Phage | 23521800 | 147 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQ |
Ypep-GFP | Human prostate carcinoma cells (LNCaP) | eGFP, Phage | 23521800 | 37 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQ |
Ypep-GFP | human embryonic lung fibroblasts (MRC-9) | eGFP, Phage | 23521800 | 105 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQ |
Ypep-GFP | human spleen fibroblasts (Hs 697.Sp) | eGFP, Phage | 23521800 | 26 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQ |
Ypep-GFP | HEK293T cells | eGFP, Phage | 23521800 | 18 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQ |
Ypep-GFP-Ypep | Human prostate adenocarcinoma cells (PC-3) | eGFP, Phage | 23521800 | 1350 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQYTFGLKTSFNVQ |
Ypep-GFP-Ypep | Human prostate carcinoma cells (LNCaP) | eGFP, Phage | 23521800 | 450 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQYTFGLKTSFNVQ |
Ypep-GFP-Ypep | human embryonic lung fibroblasts (MRC-9) | eGFP, Phage | 23521800 | 375 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQYTFGLKTSFNVQ |
Ypep-GFP-Ypep | human spleen fibroblasts (Hs 697.Sp) | eGFP, Phage | 23521800 | 100 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQYTFGLKTSFNVQ |
Ypep-GFP-Ypep | HEK293T cells | eGFP, Phage | 23521800 | 50 | Mean Fluorescence intensity | 5uM | 3h | 37ºC | Flow cytometry | Internalization | YTFGLKTSFNVQYTFGLKTSFNVQ |
CRGDK | human metastatic breast cancer cell line MDA-MB- 231 | Doxorubicin, DSPE- PEG2000 | 23634882 | 19000 | Mean Fluorescence intensity | 10 ug/mL Dox | 30 min | 37ºC | Flow cytometry | Uptake | CRGDK |
Peptide 599 | Human tongue squamous cell carcinoma (SCC) CAL 27 | siRNA | 24019920 | 45 | pmol siRNA / mg protein | 100:1 molar excess of siRNAs | 2.5 h | nan | Fluorescent Microscopy | Transfection | GLFEAIEGFIENGWEGMIDGWYGGGGrrrrrrrrrK |
CH2 R4 H2 C | S-180 sarcoma cells | siRNA | 23911914 | 700 | Mean Fluorescence intensity/cell | N/P ratio 20 | 4h | nan | Flow cytometry | Transfection | CHHRRRRHHC |
IL-13p | U87 cells | Cou-6, DiR | 24120853 | 75 | Fluorescence intensity | 100 ug/mL IL-13p | 1h | nan | Flow cytometry | Uptake | TAMRAVDKLLLHLKKLFREGQFNRNFESIIICRDRT |
IL-13p | HUVEC cells | Cou-6, DiR | 24120853 | 67.5 | Fluorescence intensity | 100 ug/mL IL-13p | 1h | nan | Flow cytometry | Uptake | TAMRAVDKLLLHLKKLFREGQFNRNFESIIICRDRT |
STR-R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 260 | Mean Fluorescence intensity | 100 nM siRNA | 3h | nan | Flow cytometry | Transfection | RRRRRRRR |
STR-H8R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 160 | Mean Fluorescence intensity | 100 nM siRNA | 3h | nan | Flow cytometry | Transfection | HHHHHHHHRRRRRRRR |
STR-H8R15 | CHO-K1 cells | GAPDH siRNA | 25193363 | 195 | Mean Fluorescence intensity | 100 nM siRNA | 3h | nan | Flow cytometry | Transfection | HHHHHHHHRRRRRRRRRRRRRRR |
STR-H12R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 187 | Mean Fluorescence intensity | 100 nM siRNA | 3h | nan | Flow cytometry | Transfection | HHHHHHHHHHHHRRRRRRRRRRRRRRR |
STR-H16R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 220 | Mean Fluorescence intensity | 100 nM siRNA | 3h | nan | Flow cytometry | Transfection | HHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
STR-H20R8 | CHO-K1 cells | GAPDH siRNA | 25193363 | 211 | Mean Fluorescence intensity | 100 nM | 3h | nan | Flow cytometry | Transfection | HHHHHHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
1b | HeLa cells | Carboxyfluorescein | 25188671 | 0.18 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLLRLL |
2b | HeLa cells | Carboxyfluorescein | 25188671 | 0.23 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLLRLX |
3b | HeLa cells | Carboxyfluorescein | 25188671 | 0.23 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLLRLXRLX |
4b | HeLa cells | Carboxyfluorescein | 25188671 | 0.85 | Cellular uptake | 100 nM | 2h | 37ºC | Fluorescence spectroscopy | Uptake | RLXRLXRLX |
Penetratin | nan | Insulin | 24973720 | 13 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | nan | nan | Absorption | RQIKIWFQNRRMKWKK |
Penetratin | nan | Insulin | 24973720 | 55 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | nan | nan | Absorption | RQIKIWFQNRRMKWKK |
RALA peptide | ZR-75-1 human breast cancer | pDNA | 24995949 | 57.0 | % Transfection | N/P ratio 10 | 48h | nan | Flow cytometry | Transfection | WEARLARALARALARHLARALARA |
RALA peptide | PC3 cells | pDNA | 24995949 | 27.0 | % Transfection | N/P ratio 10 | 48h | nan | Flow cytometry | Transfection | WEARLARALARALARHLARALARA |
C24-LMWP | A549 cells | PLGA-NPs | 25003794 | 492 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | nan | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
C24-LMWP | MCF7 cells | PLGA-NPs | 25003794 | 93.2 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | nan | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
hLF WT | HeLa cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF WT | Jurkat cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF WT | Ovcar-3 cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF WT | Caco-2 cells | Fluorescein | 24270856 | 100 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF W5A | HeLa cells | Fluorescein | 24270856 | 52.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF Q6A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF M9A | HeLa cells | Fluorescein | 24270856 | 55 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF P15A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF V12R | HeLa cells | Fluorescein | 24270856 | 75 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7A | HeLa cells | Fluorescein | 24270856 | 70 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R13A | HeLa cells | Fluorescein | 24270856 | 72.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7A/V12R | HeLa cells | Fluorescein | 24270856 | 70 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R13A/P15R | HeLa cells | Fluorescein | 24270856 | 57.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF +4R | HeLa cells | Fluorescein | 24270856 | 240 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF +4R | Jurkat cells | Fluorescein | 24270856 | 95 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF +4R | Ovcar-3 cells | Fluorescein | 24270856 | 90 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF +4R | Caco-2 cells | Fluorescein | 24270856 | 132.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF lin+4R | HeLa cells | Fluorescein | 24270856 | 137.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF lin+4R | Jurkat cells | Fluorescein | 24270856 | 200 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF lin+4R | Ovcar-3 cells | Fluorescein | 24270856 | 165 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF lin+4R | Caco-2 cells | Fluorescein | 24270856 | 460 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7 | HeLa cells | Fluorescein | 24270856 | 57.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7 | Jurkat cells | Fluorescein | 24270856 | 87.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7 | Ovcar-3 cells | Fluorescein | 24270856 | 55 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF R7 | Caco-2 cells | Fluorescein | 24270856 | 85 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF K7 | HeLa cells | Fluorescein | 24270856 | 50 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF K7 | Jurkat cells | Fluorescein | 24270856 | 75 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF K7 | Ovcar-3 cells | Fluorescein | 24270856 | 60 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF K7 | Caco-2 cells | Fluorescein | 24270856 | 87.5 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | KCFQWQRNMRKVRGPPVSCIKR |
hLF Hcy | HeLa cells | Fluorescein | 24270856 | 85 | Median Normalized Fluorescence | 5 uM | 30 min | 37ºC | Flow cytometry | Uptake | K-Hey-FQWQRNMRKVRGPPVS-Hey-IKR |
Pep1 | HeLa cells | Plasmid DNA | 24462902 | 150 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRR |
Pep1 | A549 cells | Plasmid DNA | 24462902 | 20 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRR |
Pep2 | HeLa cells | Plasmid DNA | 24462902 | 200 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRRSPRR |
Pep2 | A549 cells | Plasmid DNA | 24462902 | 30 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRRSPRR |
Pep3 | HeLa cells | Plasmid DNA | 24462902 | 700 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRRKKKKSPRRKKKKSPRR |
Pep3 | A549 cells | Plasmid DNA | 24462902 | 38 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDSPRRKKKKSPRRKKKKSPRR |
Pep3(Mutant) | HeLa cells | Plasmid DNA | 24462902 | 750 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDGPRRKKKKGPRRKKKKGPRR |
Pep3(Mutant) | A549 cells | Plasmid DNA | 24462902 | 37.5 | Mean Fluorescence intensity/cell | N/P ratio 20 | nan | nan | Flow cytometry | Transfection | GRGDGPRRKKKKGPRRKKKKGPRR |
PF21 | HEK293 cells | Plasmid DNA | 24463071 | 1,00E+04 | Fold increase | 760 nM | 24h | nan | Fluorescence spectroscopy | Transfection | WLKLLKKWLKLWKKLLKLW |
PF22 | HEK293 cells | Plasmid DNA | 24463071 | 4,00E+04 | Fold increase | 760 nM | 24h | nan | Fluorescence spectroscopy | Transfection | FLKLLKKFLKLFKKLLKLF |
PF28 | HEK293 cells | Plasmid DNA | 24463071 | 1,00E+05 | Fold increase | 760 nM | 24h | nan | Fluorescence spectroscopy | Transfection | WLKLWKKWLKLW |
FAM-1 | HeLa cells | Carboxyfluorescein | 24661993 | 1500 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BRRXRRXRRX |
ent FAM-1 | HeLa cells | Carboxyfluorescein | 24661993 | 1940 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BrrXrrXrrX |
FAM-2 | HeLa cells | Carboxyfluorescein | 24661993 | 845 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BRrXRrXRrX |
FAM-3 | HeLa cells | Carboxyfluorescein | 24661993 | 625 | pmol/mg protein Cellular uptake | 3 uM | 2 h | 37°C | Fluorescence spectroscopy | Uptake | BXRXRXXRXRXXRXRX |
RIPL | LNCaP | FITC | 24704199 | 78.3 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
RIPL | SK-OV-3 cells | FITC | 24704199 | 16.6 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
RIPL | MCF7 cells | FITC | 24704199 | 31.6 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
RIPL | DU-145 | FITC | 24704199 | 10 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
RIPL | PC3 cells | FITC | 24704199 | 23.3 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
RIPL | HaCaT cells | FITC | 24704199 | 4.16 | Mean Fluorescence intensity | 1 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLRRRRRRRRC |
R8 | LNCaP | FITC | 24704199 | 12.4 | Mean Fluorescence intensity | 3 uM | 2h | 37ºC | Flow cytometry | Uptake | RRRRRRRRC |
IPL | LNCaP | FITC | 24704199 | 9 | Mean Fluorescence intensity | 3 uM | 2h | 37ºC | Flow cytometry | Uptake | IPLVVPLC |
EGFP-TAT | Mouse macrophage-like cell line J774 A.1 | eGFP | 24746937 | 79.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | YGRKKRRQRRR |
EGFP-VP_22 | Mouse macrophage-like cell line J774 A.3 | eGFP | 24746937 | 58.1 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | DAATARGRGRSAASRPTERPRAPARSASRPRRPVD |
EGFP-LMWP | Mouse macrophage-like cell line J774 A.5 | eGFP | 24746937 | 98.8 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | GSVSRRRRRRGGRRRR |
EGFP-hcT(9-32) | Mouse macrophage-like cell line J774 A.6 | eGFP | 24746937 | 35.6 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | LGTYTQDFNKFHTFPQTAIGVGAP |
EGFP-R12 | Mouse macrophage-like cell line J774 A.10 | eGFP | 24746937 | 75.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Internalization | RRRRRRRRRRRR |
Hph-1 | HeLa cells | Hph1Hph1dsRBD/FAM-labeled siRNA complex | 24768403 | 99.0 | % Positive cells | 100 uM siRNA | 1h | nan | Flow cytometry | Uptake | YARVRRRGPRR |
Mgpe-9 | A549 cells | Plasmid DNA | 24816284 | 2,00E+06 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | MCF7 cells | Plasmid DNA | 24816284 | 8,00E+08 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | HeLa cells | Plasmid DNA | 24816284 | 2,00E+04 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | HEK | Plasmid DNA | 24816284 | 8,00E+07 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | T47D | Plasmid DNA | 24816284 | 1,00E+06 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | B16 cells | Plasmid DNA | 24816284 | 4,00E+07 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | MDA-MB-231 cells | Plasmid DNA | 24816284 | 8,00E+06 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | B35 | Plasmid DNA | 24816284 | 5,00E+07 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | U87 cells | Plasmid DNA | 24816284 | 4,00E+07 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | CHO-K1 cells | Plasmid DNA | 24816284 | 5900 | Mean Fluorescence intensity | Charge ratio = 0.5 / Charge ratio 5 | 4h | 37ºC | Flow cytometry | Cellular uptake | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | H1299 | Plasmid DNA | 24816284 | 1,00E+08 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | Jurkat cells | Plasmid DNA | 24816284 | 2,00E+04 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-9 | RAW264.7 cells | Plasmid DNA | 24816284 | 7,00E+05 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CRRLRHLRHHYRRRWHRFRC |
Mgpe-10 | A549 cells | Plasmid DNA | 24816284 | 4,00E+04 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | MCF7 cells | Plasmid DNA | 24816284 | 6,00E+06 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | HeLa cells | Plasmid DNA | 24816284 | 2,00E+02 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | HEK | Plasmid DNA | 24816284 | 5,00E+06 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | T47D | Plasmid DNA | 24816284 | 1,00E+04 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | B16 cells | Plasmid DNA | 24816284 | 2,00E+05 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | MDA-MB-231 cells | Plasmid DNA | 24816284 | 5,00E+02 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | B35 | Plasmid DNA | 24816284 | 4,00E+03 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | U87 cells | Plasmid DNA | 24816284 | 4,00E+05 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | CHO-K1 cells | Plasmid DNA | 24816284 | 400 | Mean Fluorescence intensity | Charge ratio = 0.5 / Charge ratio 5 | 4h | 37ºC | Flow cytometry | Cellular uptake | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | H1299 | Plasmid DNA | 24816284 | 4,00E+05 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | Jurkat cells | Plasmid DNA | 24816284 | 2,00E+02 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
Mgpe-10 | RAW264.7 cells | Plasmid DNA | 24816284 | 2,00E+04 | RFU/mg | Charge ratio 5 | 1h | nan | Fluorescent Microscopy | Transfection | CLLYWFRRRHRHHRRRHRRC |
cF?R4-PCP | HeLa cells | PCP, miniPEG-DE(pCAP)LI-NH2 | 24896852 | 3510 | Mean Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Uptake | FRRRRQ |
R9-PCP | HeLa cells | PCP, miniPEG-DE(pCAP)LI-NH2 | 24896852 | 960 | Mean Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Uptake | RRRRRRRRR |
Tat-PCP | HeLa cells | PCP, miniPEG-DE(pCAP)LI-NH2 | 24896852 | 290 | Mean Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Uptake | RKKRRQRRR |
Antp-PCP | HeLa cells | PCP, miniPEG-DE(pCAP)LI-NH2 | 24896852 | 400 | Mean Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
Xentry peptides 1 | HepG2 cells | FITC, TAMRA | 24811205 | 1850 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLR |
Xentry peptides 2 | HepG2 cells | FITC, TAMRA | 24811205 | 250 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LLR |
Xentry peptides 3 | HepG2 cells | FITC, TAMRA | 24811205 | 750 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LLLR |
Xentry peptides 4 | HepG2 cells | FITC, TAMRA | 24811205 | 575 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LLLLR |
Xentry peptides 5 | HepG2 cells | FITC, TAMRA | 24811205 | 300 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LLLRR |
Xentry peptides 6 | HepG2 cells | FITC, TAMRA | 24811205 | 1200 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | IIIR |
Xentry peptides 7 | HepG2 cells | FITC, TAMRA | 24811205 | 1150 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | VVVR |
Xentry peptides 8 | HepG2 cells | FITC, TAMRA | 24811205 | 950 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLK |
Xentry peptides 9 | HepG2 cells | FITC, TAMRA | 24811205 | 1525 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLH |
Xentry peptides 10 | HepG2 cells | FITC, TAMRA | 24811205 | 1675 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLE |
Xentry peptides 11 | HepG2 cells | FITC, TAMRA | 24811205 | 1137 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLN |
Xentry peptides 12 | HepG2 cells | FITC, TAMRA | 24811205 | 1550 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | LCLQ |
Xentry peptides 13 | HepG2 cells | FITC, TAMRA | 24811205 | 3150 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | lclr |
Xentry peptides 14 | HepG2 cells | FITC, TAMRA | 24811205 | 1675 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | lcl |
Xentry peptides 15 | HepG2 cells | FITC, TAMRA | 24811205 | 750 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | icir |
Xentry peptides 16 | HepG2 cells | FITC, TAMRA | 24811205 | 500 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | vcvr |
Xentry peptides 17 | HepG2 cells | FITC, TAMRA | 24811205 | 1150 | Fluorescence intensity | 10 uM | 3h | 37ºC | Fluorescence spectroscopy | Uptake | vlclr |
ACPP | A549 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 85 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
ACPP | MDA-MB-231 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 86 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
ACPP | Human bronchial epithelial (HBE) cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 9.6 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
ACPP | HepG2 cells | ACPP-HPMA Copolymer-Coated Adenovirus Conjugates | 25000246 | 96 | Relative fluorescence | 10^4 particles | 1h | 37ºC | Fluoroskan plate reader | Uptake | EEEEEEEEPLGLAGRRRRRRRRN |
F(SG)4R8 | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 147.3 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
F(SG)4R8 | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 150.0 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
G(SG)4R8 | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 105.2 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
G(SG)4R8 | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 100.0 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
F(SG)4Pen | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 221.0 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
F(SG)4Pen | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 118.75 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
G(SG)4Pen | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 105.2 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
G(SG)4Pen | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 100.0 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
F(SG)4TP10 | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 884.2 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
F(SG)4TP10 | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 462.5 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
G(SG)4TP10 | HeLa cells | Alexa488, bovine serum albumin, QDs | 25108152 | 105.2 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
G(SG)4TP10 | KG1a cells | Alexa488, bovine serum albumin, QDs | 25108152 | 100.0 | Relative fluorescence (%) | 2 uM | 1h | 37ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
LMWP | Pluripotent mouse mesenchymal progenitor cell line (C3H10T1/2) | TAZ | 24648725 | 98.9 | % Positive cells | 100 nM | 20 min | 37ºC | Flow cytometry | Internalization | VSRRRRRRGGRRRR |
R7 | nan | ESRRB recombinant protein | 24693491 | 53.3 | Relative fluorescence | 2 ug/ml | 24h | nan | Immunocytochemistry | Transduction | RRRRRRR |
Pip6a | Murine H2k mdx myoblasts | phosphorodiamidate morpholino oligomers (PMO) | 24366877 | 12812 | RFU/mg | 1 uM | 4h | nan | Fluorescence spectroscopy | Internalization | RXRRBRRXRYQFLIRXRBRXRB |
Pip6a | C2C12 cells | phosphorodiamidate morpholino oligomers (PMO) | 24366877 | 7916 | RFU/mg | 1 uM | 4h | nan | Fluorescence spectroscopy | Internalization | RXRRBRRXRYQFLIRXRBRXRB |
R9 | CHO-K1 cells | Biotin-gly4 | 25112713 | 8.0 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRRRRRRRR |
R9 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 2.5 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRRRRRRRR |
TAT(47-57) | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | YGRKKRRQRRR |
TAT(47-57) | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.725 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | YGRKKRRQRRR |
R6L3 | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.3 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRLLRRLRR |
R6L3 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRLLRRLRR |
Penetratin | CHO-K1 cells | Biotin-gly4 | 25112713 | 0.3 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RQIKIWFQNRRMKWKK |
Penetratin | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 0.2 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RQIKIWFQNRRMKWKK |
R6W3 | CHO-K1 cells | Biotin-gly4 | 25112713 | 9 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRWWRRWRR |
R6W3 | xylose transferase- or GAG-deficient CHO-pgsA745 cells (GAGneg) | Biotin-gly4 | 25112713 | 5.0 | Internalized peptide (uM) | 10 uM | 70 min | 37ºC | MALDI-TOF | Internalization | RRWWRRWRR |
MCa UF1-9-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 4.7e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | GD(Abu)LPHLKLC |
Tat-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 9.0e+4 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | YGRKKRRQRRRC |
Pen-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 1.3e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | RQIKIWFQNRRMKWKKC |
PolyR-C-Cy5 | Undifferentiated malignant glioma rat (F98) cell line | Cy5 | 24276021 | 1.4e+5 | Fluorescence intensity | 10 uM | 2h | 37ºC | Flow cytometry | Penetration | RRRRRRRRRC |
Alexa488-Melan-A-TAT | Dendritic cells | Alexa488, ovalbumin | 24372650 | 9500 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVRKKRRQRRR |
Alexa488-Melan-A-TAT | HUVEC cells | Alexa488, ovalbumin | 24372650 | 4500 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVRKKRRQRRR |
Alexa488-Melan-A-TAT | Jurkat cells | Alexa488, ovalbumin | 24372650 | 4500 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVRKKRRQRRR |
Alexa488-Melan-A-polyLys (control peptide) | Dendritic cells | Alexa488, ovalbumin | 24372650 | 4800 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVKKKKKQKKK |
Alexa488-Melan-A-polyLys (control peptide) | HUVEC cells | Alexa488, ovalbumin | 24372650 | 3000 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVKKKKKQKKK |
Alexa488-Melan-A-polyLys (control peptide) | Jurkat cells | Alexa488, ovalbumin | 24372650 | 3000 | Mean Fluorescence intensity | 3 ug/ml | 60 min | 37ºC | Flow cytometry | Uptake | CELAGIGILTVKKKKKQKKK |
CF-BP16 | MCF7 cells | Carboxyfluorescein | 24480922 | 1431 ± 307 | Mean Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Uptake | KKLFKKILKKL |
CF-BP16 | mouse embryonic fibroblast 3T3 | Carboxyfluorescein | 24480922 | 1829 ± 335 | Mean Fluorescence intensity | 50 uM | 1h | 37ºC | Flow cytometry | Uptake | KKLFKKILKKL |
BP328 | MCF7 cells | Carboxyfluorescein | 24480922 | 1789 ± 221 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | CREKA-KKLFKKILKKL |
BP328 | mouse embryonic fibroblast 3T3 | Carboxyfluorescein | 24480922 | 1300 ± 221 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | CREKA-KKLFKKILKKL |
BP326 | MCF7 cells | Carboxyfluorescein, CLB | 24480922 | 4272 ± 453 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | KKLFKKILKKL |
BP330 | MCF7 cells | Carboxyfluorescein, CLB | 24480922 | 3966 ± 217 | Mean Fluorescence intensity | 25 uM | 3h | 37ºC | Flow cytometry | Uptake | CREKA-KKLFKKILKKL |
Penetratin | Wong-Kilbourne-derived human conjunctival epithelial cells (NHC) | Carboxyfluorescein | 24521351 | 13000 | Mean Fluorescence intensity | 57 umol/L | 1h | 37ºC | Flow cytometry | Uptake | RQIKIWFQNRRMKWKKK |
Arg5-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 2.0 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRR |
Arg8-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 10 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
TAT-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 10 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRR |
RTAT-ELPBC | HeLa cells | BH3 peptide drug and ELPBC | 24611762 | 4.0 | Cell Fluorescence | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | YGRGGRRGRRR |
IA0 (Bicyclic) (integral arginine peptides) | HeLa cells | FITC | 24697151 | 0 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGSGSGCGSGSGSCG |
IA2 | HeLa cells | FITC | 24697151 | 1.25 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGRGSGCGSGRGSCG |
IA4a | HeLa cells | FITC | 24697151 | 3.75 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACRGSGRGCGRGSGRCG |
IA4b | HeLa cells | FITC | 24697151 | 10 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACSGRGRGCGRGRGSCG |
IA6b | HeLa cells | FITC | 24697151 | 20 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACGRGRGRCRGRGRGCG |
IA8b | HeLa cells | FITC | 24697151 | 45 | Normalized Median Fluorescence | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | ACRRSRRGCGRRSRRCG |
GST-(HE)8EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 240 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
GST-(HE)10EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 190 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
GST-(HE)12EFG5YG(RG)6 | HeLa cells | GST | 24697211 | 80 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRGRGRGRGRGRG |
GST-(HE)8EFG5YGR6G6 | HeLa cells | GST | 24697211 | 370 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
GST-(HE)10EFG5YGR6G6 | HeLa cells | GST | 24697211 | 335 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
GST-(HE)12EFG5YGR6G6 | HeLa cells | GST | 24697211 | 100 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRRRRRRGGGGGG |
GST-(HE)12EFG5-TAT | HeLa cells | GST | 24697211 | 327 | ng molecule / mg cell protein | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Uptake | HEHEHEHEHEHEHEHEHEHEHEHEEFGGGGGYGRKKRRQRRR |
LK-1 | HeLa cells | FITC | 25056130 | 67 | % Positive cells | 100 nM | 12h | nan | FACS | Uptake | LKKLLKLLKKLLKLAG |
LK-2 | HeLa cells | FITC | 25056130 | 70 | % Positive cells | 100 nM | 12h | nan | FACS | Uptake | LKKLCKLLKKLCKLAG |
VG-21 | HEp-2 | FITC | 25154664 | 35.3 | % Positive cells | 1 nM | 48h | nan | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
VG-21 | HeLa cells | FITC | 25154664 | 43.8 | % Positive cells | 1 nM | 48h | nan | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
VG-21 | Vero | FITC | 25154664 | 32.4 | % Positive cells | 1 nM | 48h | nan | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
VG-21 | Cos-7 cells | FITC | 25154664 | 26.6 | % Positive cells | 1 nM | 48h | nan | Flow cytometry | Uptake | VTPHHVLVDEYTGEWVDSQFK |
[R4W4]Cyclic | SK-OV-3 cells | Fluorescein | 25157458 | 3650 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry, CLSM | Uptake | RRRRWWWW |
PF3 | HeLa cells | pGL3, siRNA, SCO | 25135660 | 1 | Relative Cellular uptake | 0.5 uM | 30 min | 37ºC | FACS | Uptake | AGYLLGKINLKALAALAKKIL |
NF1 | HeLa cells | pGL3, siRNA, SCO | 25135660 | 0.97 | Relative Cellular uptake | 0.5 uM | 30 min | 37ºC | FACS | Uptake | AGYLLGKTNLKALAALAKKIL |
NF51 | HeLa cells | pGL3, siRNA, SCO | 25135660 | 0.77 | Relative Cellular uptake | 0.5 uM | 30 min | 37ºC | FACS | Uptake | AGYLLGOINLKALAALAKKIL |
PNIPAM-FL-TAT Peptide | A549 cells | poly(N-isopropylacrylamide) (PNIPAM) microgel particles | 25170605 | 1500 | Relative fluorescence | 200 ug/ml | 24h | nan | Flow cytometry | Uptake | YGRKKRRQRRR |
Trehalose-KRKRWHW-Heparin | Mammalian cells | Trehalose | 24583082 | 20 | mM Intracellular concentration | 8 mM Trehalose | 1h | 37ºC | Flow cytometry | Interalization | KRKRWHW |
SP-TatCherry | A549 cells | mCherry | 24928321 | 2800 | Mean Fluorescence intensity | 13 uM | 24h | nan | Fluorescence spectroscopy | Transduction | YGRKKRRQRRR |
SP-Tatm3xCherry | A549 cells | mCherry | 24928321 | 3900 | Mean Fluorescence intensity | 13 uM | 24h | nan | Fluorescence spectroscopy | Transduction | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
SP-Tatm3xCherry | CHO-K1 cells | mCherry | 24928321 | 15900 | Mean Fluorescence intensity | 13 uM | 24h | nan | Fluorescence spectroscopy | Transduction | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
Penetratin | None | Insulin | 24973720 | 15 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | nan | nan | Absorption | RQIKIWFQNRRMKWKK |
Penetratin | None | Insulin | 24973720 | 55 | Plasma insulin concentration (uU/mL) | 5 mM | 30 min | nan | nan | Absorption | RQIKIWFQNRRMKWKK |
MCoTI-II | HeLa cells | Alexa488 | 24985034 | 1.0 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
MCoTI-M1 | HeLa cells | Alexa488 | 24985034 | 0.95 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGWCGSGSD |
MCoTI-M2 | HeLa cells | Alexa488 | 24985034 | 1.08 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSD |
MCoTI-M3 | HeLa cells | Alexa488 | 24985034 | 0.52 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGWCGSGSD |
MCoTI-M4 | HeLa cells | Alexa488 | 24985034 | 1.65 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSR |
MCoTI-M5 | HeLa cells | Alexa488 | 24985034 | 1.73 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPRILRRCRRDSDCPGACICRGNGYCGSGSK |
MCoTI-M6 | HeLa cells | Alexa488 | 24985034 | 1.95 | Normalized Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
SFTI-1 | HeLa cells | Alexa488 | 24985034 | 1.00 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICFPD |
D-SFTI-1 | HeLa cells | Alexa488 | 24985034 | 1.17 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | grctksippicfpd |
SFTI-M1 | HeLa cells | Alexa488 | 24985034 | 1.04 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GACTKSIPPICFPD |
SFTI-M2 | HeLa cells | Alexa488 | 24985034 | 0.86 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICFPA |
SFTI-M3 | HeLa cells | Alexa488 | 24985034 | 1.13 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICWPD |
SFTI-M4 | HeLa cells | Alexa488 | 24985034 | 1.00 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTKSIPPICWPK |
SFTI-M5 | HeLa cells | Alexa488 | 24985034 | 1.26 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRCTRSIPPKCWPD |
SFTI-M6 | HeLa cells | Alexa488 | 24985034 | 1.13 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRXTKSIPPIXFPD |
SFTI-M7 | HeLa cells | Alexa488 | 24985034 | 0.82 | Normalized Mean Fluorescence intensity | 16 uM | 1h | 37ºC | Flow cytometry | Uptake | GRXTKSIPPIXFPD |
TAT | HeLa cells | Alexa488 | 24985034 | 3.0 / 6.0 | Mean Fluorescence intensity | 8 uM MCoTI-II / 16 uM SFTI-1 | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRRPPQG |
C24-LMWP | A549 cells | LMWP/PLGA nanoparticles, Doxorubicin | 25003794 | 872 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | nan | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
C24-LMWP | MCF7 cells | LMWP/PLGA nanoparticles, Doxorubicin | 25003794 | 153 | Median Fluorescence intensity | Equal to a DOX dose of 10 ug/mL | 4h | nan | Flow cytometry | Uptake | VSRRRRRRGGRRRR |
VIP-TAT | Neuro2a cells | FITC | 25086267 | 1.81 ± 0.34 | % Brain uptake efficiency (% of total peptide i. p. injection of VIP-TAT) | 100 nmol/kg | nan | nan | Fluorescence spectroscopy | Uptake | HSDAVFTDNYTALRKQMAVKKYLNSILNYGRKKRRQRRR |
Cys(BSH)-Arg11-NH2 | U87 cells | BSH | 24452095 | 391.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | nan | Immunocytochemistry | Uptake | RRRRRRRRRRR |
Cys(BSH)-Lys[Cys(BSH)-]Arg11-NH2 | U87 cells | BSH | 24452095 | 391.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | nan | Immunocytochemistry | Uptake | RRRRRRRRRRR |
[Cys(BSH)]4-(Lys)3-Arg11-NH2 | U87 cells | BSH | 24452095 | 588.8 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | nan | Immunocytochemistry | Uptake | RRRRRRRRRRR |
Cys(BSH)-TAT | U87 cells | BSH | 24452095 | 150 | ng^10B/10^6 cells | 10 uM BSH-11R (Boron concentration) | 12h | nan | Immunocytochemistry | Uptake | GRKKRRQRRR |
Cys(BSH)-R11 | U87 cells | BSH | 24452095 | 219.4 | ng^10B/10^6 cells Boron concentration | 10 uM BSH-11R | 2h | nan | Immunocytochemistry | Uptake | RRRRRRRRRRR |
Peptide I | CHO-K1 cells | Carboxyfluorescein | 25096299 | 64 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | FACS | Uptake | RXRRXRRXRRXR |
Peptide II | CHO-K1 cells | Carboxyfluorescein | 25096299 | 71 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | FACS | Uptake | RXRRXRRXRRXR |
Peptide III | CHO-K1 cells | Carboxyfluorescein | 25096299 | 85 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | FACS | Uptake | RXRRXRRXRRXR |
Peptide IV | CHO-K1 cells | Carboxyfluorescein | 25096299 | 75 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | FACS | Uptake | RXRRXRRXRRXR |
Peptide V | CHO-K1 cells | Carboxyfluorescein | 25096299 | 31 | Mean Fluorescence intensity | 10 uM | 4h | 37ºC | FACS | Uptake | RXRRXRRXRRXR |
IRQ | Caco-2 cells | FITC-sCT, SLN | 24968819 | 2.17 | FITC-sCT ug/mg protein | 50 ug/ml | 1h | 37ºC | Fluorescent Microscopy | Uptake | IRQRRRR |
IRQ | goblet like HT29-MTX cells | FITC-sCT, SLN | 24968819 | 2.17 | FITC-sCT ug/mg protein | 50 ug/ml | 1h | 37ºC | Fluorescent Microscopy | Uptake | IRQRRRR |
CSK | Caco-2 cells | FITC-sCT, SLN | 24968819 | 3.6 | FITC-sCT ug/mg protein | 50 ug/ml | 1h | 37ºC | Fluorescent Microscopy | Uptake | CSKSSDYQC |
CSK | goblet like HT29-MTX cells | FITC-sCT, SLN | 24968819 | 3.6 | FITC-sCT ug/mg protein | 50 ug/ml | 1h | 37ºC | Fluorescent Microscopy | Uptake | CSKSSDYQC |
Tat | HUVEC cells | Ultrasound contrast agent (UCA), FITC | 24985759 | 18.74 ± 0.47 | % Average transfection efficiency | nan | 24h | 37ºC | Flow cytometry | Transfection | CGYGRKKRRQRRRGC |
MAP | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 6000 | Fluorescence intensity | 1 uM | 30 min | nan | Flow cytometry | Uptake | KLALKLALKALKAALKLA |
pAntp | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 3300 | Fluorescence intensity | 1 uM | 30 min | nan | Flow cytometry | Uptake | RQIKIWFQNRRMKWKK |
Arg9 | Rat basophilic leukemia RBL-2H3 cells | Fluorescein | 25016968 | 7500 | Fluorescence intensity | 1 uM | 30 min | nan | Flow cytometry | Uptake | RRRRRRRRR |
R8-RGD-lipo | C6 cells | CFPE-labeled liposomes, RGD | 24651033 | 225 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR-c(RGDfK) |
R8-RGD-lipo | bEnd.3 cells | CFPE-labeled liposomes, RGD | 24651033 | 225 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR-c(RGDfK) |
R8-RGD-lipo | HeLa cells | CFPE-labeled liposomes, RGD | 24651033 | 10.5 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR-c(RGDfK) |
R8-lipo | C6 cells | CFPE-labeled liposomes | 24651033 | 100 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
R8-lipo | bEnd.3 cells | CFPE-labeled liposomes | 24651033 | 120 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
R8-lipo | HeLa cells | CFPE-labeled liposomes | 24651033 | 11 | Mean Fluorescence intensity | 1.5 ug/mL lipossomes | 4h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
TAT-BID | PC3 cells | BID | 25326334 | 70.0 | Cellular uptake (%) | 40 ug/ml | 120 min | nan | Western blot | nan | YGRKKRRQRRR |
TAT-BID | LNCaP | BID | 25326334 | 100.0 | Cellular uptake (%) | 30 ug/ml | 120 min | nan | Western blot | nan | YGRKKRRQRRR |
TAT-BID | A549 cells | BID | 25326334 | 60.0 | Cellular uptake (%) | 40 ug/ml | 120 min | nan | Western blot | nan | YGRKKRRQRRR |
TAT-BID | HeLa cells | BID | 25326334 | 20.0 | Cellular uptake (%) | 40 ug/ml | 120 min | nan | Western blot | nan | YGRKKRRQRRR |
TAT-lyophiliosomes | HeLa cells | Lyophiliosomes and FITC labelled | 25369131 | 86±3 | % Positive cells | 25 µg/ml | 1h | nan | FACS | Internalization | YGRKKRRQRRR |
TAT-lyophiliosomes | Ovcar-3 cells | Lyophiliosomes and FITC labelled | 25369131 | 97±3 | % Positive cells | 25 µg/ml | 1h | nan | FACS | Internalization | YGRKKRRQRRR |
TAT-lyophiliosomes | Caco-2 cells | Lyophiliosomes and FITC labelled | 25369131 | 87±3 | % Positive cells | 25 µg/ml | 1h | nan | FACS | Internalization | YGRKKRRQRRR |
TAT-lyophiliosomes | SK-OV-3 cells | Lyophiliosomes and FITC labelled | 25369131 | 95±10 | % Positive cells | 25 µg/ml | 1h | nan | FACS | Internalization | YGRKKRRQRRR |
KST | K562 cells | Avidin-FITC | 25387797 | 26 | Fluorescence intensity | 5 uM | 18h | 37ºC | Flow cytometry | Uptake | KSTGKANKITITNDKGRLSK |
PTX-TAT-LP | Murine B16F1 melanoma tumor cells | PTX with liposome,GSH | 25449709 | 12.6 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Uptake | CAYGRKKRRQRRR |
PTX-C-TAT-LP | Murine B16F1 melanoma tumor cells | PTX with liposome,GSH | 25449709 | 7 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Uptake | CAYGRKKRRQRRR |
PTX-N-TAT-LP | Murine B16F1 melanoma tumor cells | PTX with liposome,GSH | 25449709 | 2.25 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Uptake | CYGRKKRRQRRR |
Tat2-Nat | primary culture of human corneal epithelial cells | Natamycin, FITC | 25467959 | 34 000 | FITC Mean Intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | RKKRRQRRRRKKRRQRRR |
MTat2-Nat | primary culture of human corneal epithelial cells | Natamycin, FITC | 25467959 | 11 000 | FITC Mean Intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | AKKRRQRRRAKKRRQRRR |
TP-biot1 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 400 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
TP-biot1 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 220 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
TP-biot13 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 80 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
TP-biot13 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 90 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | GWTLNSAGYLLGKINLKALAALAKKIL |
TP10-biot1 | HT29 cells | Streptavidin conjugated with FITC | 25511292 | 50 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
TP10-biot1 | HCT116 cells | Streptavidin conjugated with FITC | 25511292 | 150 | Fluorescence intensity | 4 uM CPP | 2h | 25ºC | Flow cytometry | Uptake | AGYLLGKINLKALAALAKKIL |
Tpl | Plant cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 116 | RFU | 20 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWCFRVCYRGICYRRCRGK |
Tpl | HeLa cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 150 | RFU | 30 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWCFRVCYRGICYRRCRGK |
MTpl-1 | Plant cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 114 | RFU | 20 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWSFRVSYRGISYRRSRGK |
MTpl-1 | HeLa cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 145 | RFU | 30 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWSFRVSYRGISYRRSRGK |
MTpl-2 | Plant cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 152 | RFU | 20 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWFRVYRGIYRRRGK |
MTpl-2 | HeLa cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 485 | RFU | 30 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWFRVYRGIYRRRGK |
MTpl-3 | Plant cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 34 | RFU | 20 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWCFAVCYAGICYAACAGK |
MTpl-3 | HeLa cells | beta-glucuronidase enzyme, beta-galactosidase | 25514997 | 35 | RFU | 30 uM | 1h | nan | Fluorescence spectroscopy | Uptake | KWCFAVCYAGICYAACAGK |
cTAT-GFP | HeLa cells | eGFP | 25521313 | 80.0 | Cellular uptake (%) | 150 uM | 60 min | 37ºC | CLSM | Uptake | rRrGrKkRr |
TAT-GFP | HeLa cells | eGFP | 25521313 | 1.0 | Cellular uptake (%) | 150 uM | 60 min | 37ºC | CLSM | Uptake | rRrGrKkRr |
V1 | Jurkat cells | FITC labelled peptide | 25524829 | 931 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRGRRG |
V2 | Jurkat cells | FITC labelled peptide | 25524829 | 2750 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRRRRR |
V2R | Jurkat cells | FITC labelled peptide | 25524829 | 0 | Mean Fluorescence intensity | 10 uM | 10 min | 37ºC | Flow cytometry | Uptake | RRRRRR |
RVG-9LR | Neuro2a cells | siRNA | 25544044 | 1527±121 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | 24h | nan | Flow cytometry | Transfection | RRRRRRRRR |
RVG-9LR | Jurkat cells | siRNA | 25544044 | 20.97±0.99 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | nan | nan | Flow cytometry | Transfection | RRRRRRRRR |
RVG-9DR | Neuro2a cells | siRNA | 25544044 | 627±124 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | 24h | nan | Flow cytometry | Transfection | rrrrrrrrr |
RVG-9DR | Jurkat cells | siRNA | 25544044 | 18.60±0.82 | Mean Fluorescence intensity | Final Concentration between 1/5 uM | nan | nan | Flow cytometry | Transfection | rrrrrrrrr |
R8-GALA-liposome-IgG | HeLa cells | Liposome, IgG | 25546552 | 36.6 | Geo Mean Fluorescence intensity | nan | 30 min | nan | Flow cytometry | Uptake | RRRRRRRR |
R8-GALA-liposome | HeLa cells | Liposome | 25546552 | 68 | Geo Mean Fluorescence intensity | nan | 1 h | nan | Flow cytometry | Uptake | RRRRRRRR |
R8-liposome | HeLa cells | Liposome | 25546552 | 94 | Geo Mean Fluorescence intensity | nan | 1h | nan | Flow cytometry | Uptake | RRRRRRRR |
5-FAM-H3R8 | MCF7 cells | Carboxyfluorescein | 25547808 | 24.67 | Geo Mean Fluorescence intensity | 1 uM | 4h | nan | Flow cytometry | Uptake | HHHRRRRRRRR |
MTS-(5-FAM)- H3R8 | MCF7 cells | Carboxyfluorescein, MTS | 25547808 | 171.18 | Geo Mean Fluorescence intensity | 1 uM | 4h | nan | Flow cytometry | Uptake | HHHRRRRRRRR |
DSPE-PEG-2K-TAT | Bovine chondriocytes | Rhodamine labelled miscelleS, Liposome | 23186944 | 10 | Mean Fluorescence intensity | 0.5 mg/ml | 1h | 37ºC | nan | nan | YGRKKRRQRRR-C |
DNA-IL-PEI | HEK293 cells | DNA, PEI | 23999223 | 1.56 | umol of ONPG/mg of protein | PEI N/P 5, IL N/P 5 | 48h | nan | Fluorescent Microscopy | Transfection | HILPWKWPWWPWRR |
DNA-IL-PEI | NIH-3T3 cells | DNA, PEI | 23999223 | 0.87 | umol of ONPG/mg of protein | PEI N/P 5, IL N/P 5 | 48h | nan | Fluorescent Microscopy | Transfection | HILPWKWPWWPWRR |
CS-Lin-Pen | HEK293 cells | FITC labeled CS-Lin | 24083483 | 85 | % Transfection | nan | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
CS-Lin-Pen | CHO cells | FITC labeled CS-Lin | 24083483 | 60 | % Transfection | nan | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
CS-Lin-Pen | Human cervical adenocarcinoma | FITC labeled CS-Lin | 24083483 | 55 | % Transfection | nan | 4h | 37ºC | Flow cytometry | Transfection | RQIKIWFQNRRMKWKKGG |
Bac-ELP-H1 | D54 cells | Rhodamine labeled ELP | 23372821 | 50 | ug CPP-ELP / g tissue (C6) | nan | 4h | nan | Fluorescent Microscopy | Uptake | MRRIRPRPPRLPRPRPRPLPFPRPGGCYPG |
SynB1-ELP-H1 | D54 cells | Rhodamine labeled ELP | 23372821 | 92 | ug CPP-ELP / g tissue (C6) | nan | 4h | nan | Fluorescent Microscopy | Uptake | RGGRLSYSRRRFSTSTGRA |
I-TYR-L-Mca | F98 glioma cell culture | Radiolabelled Iodine (125I) | 24667409 | 20 | Intracellular concenctration (uM) | 10000 nM | 2h | 37ºC | Gamma-well counter | Uptake | YGDCLPHLKLCKENKDCCSKKCKRRGTNIEKRCR |
PC-CC9/miRNA | Panc-1 | miRNA | 23298779 | 78.08 | Cellular uptake (%) | 0.15 uM | 2h | nan | Flow cytometry | Uptake | CRGDKGPDC |
PC-CC9/miRNA | 293T cells | miRNA | 23298779 | 51.07 | Cellular uptake (%) | 0.15 uM | 2h | nan | Flow cytometry | Uptake | CRGDKGPDC |
Tm3+-DOTA-CAT | SN56 cells | MRI probe [DOTA-caged metal ion (Tmü?)] | 23281285 | 19.0 ± 2.0 | % Positive cells | 5 uM | 30 min | 37ºC | CLSM | Uptake | GRKKRRQRRR |
TAT-EGFP | The mouse macrophage J774 A.1 cells | eGFP | 24746937 | 79.2 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Uptake | YGRKKRRQRRR |
LMWP-EGFP | The mouse macrophage J774 A.1 cells | eGFP | 24746937 | 98.8 | % Positive cells | 10 umol/L | 1h | 37ºC | Flow cytometry | Uptake | GSVSRRRRRRGGRRRR |
R8-lip | Bone marrow dendritic cells | Liposome | 24901376 | 10.7 | Fluorescence intensity | 40 uM | 2h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
fTAT | HeLa cells | TMR | 24930129 | 1300 | Normalized Mean Fluorescence intensity | 1 uM | 1h | nan | Flow cytometry | Uptake | CKYGRKKRRQRRR |
DOX-TAT-LIP | C6 cells | Liposome, Doxorubicin | 24893333 | 99.43 | Fluorescence intensity | 12.5 ug/mL Final Dox Concentration | 4h | 37ºC | Flow cytometry | Uptake | AYGRKKRRQRRR |
DOX-TAT-LIP | bEnd.3 cells | Liposome, Doxorubicin | 24893333 | 83.79 | Fluorescence intensity | 12.5 ug/mL Final Dox Concentration | 4h | 37ºC | Flow cytometry | Uptake | AYGRKKRRQRRR |
DOX-T7-TAT-LIP | C6 cells | Liposome, Doxorubicin, Transferin | 24893333 | 150 | Fluorescence intensity | 12.5 ug/mL Final Dox Concentration | 4h | 37ºC | Flow cytometry | Uptake | AYGRKKRRQRRR |
DOX-T7-TAT-LIP | bEnd.3 cells | Liposome, Doxorubicin, Transferin | 24893333 | 152.5 | Fluorescence intensity | 12.5 ug/mL Final Dox Concentration | 4h | 37ºC | Flow cytometry | Uptake | AYGRKKRRQRRR |
KW | MEF cells | Trehalose | 24583082 | 86 | % Positive cells | 100 uM | 4h | 37ºC | FACS | Uptake | KRKRWHW |
HIV-TAT | Porcine skin | Sodium diclofenac, celecoxib CLXB | 24798650 | 164 | ug Cumulative Na-DFC amount which penetrated through the skin / 42 ug Cumulative CLXB amount which penetrated through the skin | nan | 25h | 37ºC | HPCL-analysis | Penetration efficiencies | GRKKRRQRRRPPQ |
LMWP-TAZ | Cultured Human Dental Pulp Stem Cells (hDPSCs) | TAZ | 21990606 | 100.0 | % Positive cells | 500 nM | 30 min | nan | FACS | Transduction | VSRRRRRRGGRRRR |
pVEC | CHO-K1 cells | Plasmid DNA | 21996011 | 14 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLIILRRRIRKQAHAHSK |
S6KR | CHO-K1 cells | Plasmid DNA | 21996011 | 15 | Mean Fluorescence intensity / % FITC Positive cells | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLHILRRSIRKQAHAIRK |
S9R | CHO-K1 cells | Plasmid DNA | 21996011 | 58 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLRILRRSIRRARRAIRR |
S6R | CHO-K1 cells | Plasmid DNA | 21996011 | 18 | Mean Fluorescence intensity | Charge ratio = 10 | 4h | 37ºC | Flow cytometry | Uptake | LLHILRRSIRRQAHAIRR |
CPPK | HEK | FITC | 22076844 | 900 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAMPGEPRRANVMAHKLEPASLQLR NSCA |
CPPK | HeLa cells | FITC | 22076844 | 930 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAMPGEPRRANVMAHKLEPASLQLR NSCA |
CPPL | HEK | FITC | 22076844 | 1500 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAPQRDTVGGRTTPPSWGPAKAQLRNSCA |
CPPL | HeLa cells | FITC | 22076844 | 2500 | Fold change in average fluorescence | 10 nM | 3 h | 37°C | Confocal laser scanning system (clss) | Uptake | MAPQRDTVGGRTTPPSWGPAKAQLRNSCA |
Tat | ARPE-19 cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
Tat | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
Tat | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRRPPQ |
II | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
II | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
II | CHO cells | Fluorescein | 22100438 | 1.14 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRRRPPQ |
III | ARPE-19 cells | Fluorescein | 22100438 | 0.9 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
III | CHO cells | Fluorescein | 22100438 | 1.00 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
III | CHO cells | Fluorescein | 22100438 | 1.04 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRWWRPPQ |
IV | ARPE-19 cells | Fluorescein | 22100438 | 0.96 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
IV | CHO cells | Fluorescein | 22100438 | 1.14 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
IV | CHO cells | Fluorescein | 22100438 | 1.07 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRWWRRPPQ |
V | ARPE-19 cells | Fluorescein | 22100438 | 0.82 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
V | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
V | CHO cells | Fluorescein | 22100438 | 0.98 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRWWRQRWWRWWRPPQ |
VI | ARPE-19 cells | Fluorescein | 22100438 | 1.02 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
VI | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
VI | CHO cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRRRPPQ |
VII | ARPE-19 cells | Fluorescein | 22100438 | 0.92 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
VII | CHO cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
VII | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRAARPPQ |
VIII | ARPE-19 cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
VIII | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
VIII | CHO cells | Fluorescein | 22100438 | 0.83 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRAARRPPQ |
IX | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
IX | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
IX | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRAARQRAARAARPPQ |
X | ARPE-19 cells | Fluorescein | 22100438 | 0.95 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
X | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
X | CHO cells | Fluorescein | 22100438 | 0.77 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRRRPPQ |
XI | ARPE-19 cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
XI | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
XI | CHO cells | Fluorescein | 22100438 | 0.73 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRRLLRPPQ |
XII | ARPE-19 cells | Fluorescein | 22100438 | 0.89 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
XII | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
XII | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRLLRRPPQ |
XIII | ARPE-19 cells | Fluorescein | 22100438 | 1.18 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
XIII | CHO cells | Fluorescein | 22100438 | 1.34 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
XIII | CHO cells | Fluorescein | 22100438 | 0.95 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRLLRQRLLRLLRPPQ |
XIV | ARPE-19 cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
XIV | CHO cells | Fluorescein | 22100438 | 0.84 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
XIV | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQRR-Ahx-RPPQ |
XV | ARPE-19 cells | Fluorescein | 22100438 | 0.97 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
XV | CHO cells | Fluorescein | 22100438 | 0.88 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
XV | CHO cells | Fluorescein | 22100438 | 0.76 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQRRRPPQ |
XVI | ARPE-19 cells | Fluorescein | 22100438 | 1.06 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
XVI | CHO cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
XVI | CHO cells | Fluorescein | 22100438 | 0.85 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKRRQR-Ahx-RRPPQ |
XVII | ARPE-19 cells | Fluorescein | 22100438 | 0.90 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
XVII | CHO cells | Fluorescein | 22100438 | 0.74 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
XVII | CHO cells | Fluorescein | 22100438 | 0.78 | Cellular uptake | 2.1 uM | 30 min | 37°C | Flow cytometry | Uptake | CGRKKR-Ahx-RQR-Ahx-R-ahx-RPPQ |
TAM-MP | U373 MG cells | TAMRA | 22148546 | 15.82 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | INLKALAALAKKIL |
TAM-iMP | U373 MG cells | TAMRA | 22148546 | 100.0 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | inlkalaalakkil |
TAM-rMP | U373 MG cells | TAMRA | 22148546 | 9.762 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | LIKKALAALAKLNI |
TAM-riMP | U373 MG cells | TAMRA | 22148546 | 7.990 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | likkalaalaklni |
TAM-MitP | U373 MG cells | TAMRA | 22148546 | 82.21 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | INLKKLAKL(Aib)KKIL |
TAM-iMitP | U373 MG cells | TAMRA | 22148546 | 63.06 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | inlkklakl(Aib)kkil |
TAM-rMitP | U373 MG cells | TAMRA | 22148546 | 14.75 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | LIKK(Aib)LKALKKLNI |
TAM-riMitP | U373 MG cells | TAMRA | 22148546 | 23.23 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Fluorescence spectroscopy | Translocation | likk(Aib)lkalkklni |
Cyt c-ss-MAP | HEK293 cells | Cyt C protein | 22225540 | 1105.2 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KLALKLALKALKAALKLA |
Cyt c-ss-MAP | HeLa cells | Cyt C protein | 22225540 | 1575 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | KLALKLALKALKAALKLA |
Cyt c-ss-R8 | HEK293 cells | Cyt C protein | 22225540 | 100 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | RRRRRRRR |
Cyt c-ss-R8 | HeLa cells | Cyt C protein | 22225540 | 262.5 | ng molecule / mg cell protein | 10 ug/ml | 1h | 37ºC | Fluorescence spectroscopy | Uptake | RRRRRRRR |
PenArg | HEK293T cells | Plasmid DNA | 22281502 | 5.0 | Cellular uptake (%) | charge ratio = 2 | 2h | nan | Flow cytometry | Transfection | RQIRIWFQNRRMRWRR |
PenArg-Cys | HEK293T cells | Plasmid DNA | 22281502 | 38.0 | Cellular uptake (%) | charge ratio = 2 | 2h | nan | Flow cytometry | Transfection | RQIRIWFQNRRMRWRRC |
EB1 | HEK293T cells | Plasmid DNA | 22281502 | 48.0 | Cellular uptake (%) | charge ratio = 2 | 2h | nan | Flow cytometry | Transfection | LIRLWSHLIHIWFQNRRLKWKKK |
EB1-Cys | HEK293T cells | Plasmid DNA | 22281502 | 49.0 | Cellular uptake (%) | charge ratio = 2 | 2h | nan | Flow cytometry | Transfection | LIRLWSHLIHIWFQNRRLKWKKKC |
R8 | nan | Alexa600 | 22285548 | 378.0 | Relative fluorescence (%) | 3 nmol | 24h | nan | CLSM | Tumor accumulation | RRRRRRRRGC |
r8 | nan | Alexa600, Doxorubicin | 22285548 | 932.0 | Relative fluorescence (%) | 3 nmol | 24h | nan | CLSM | Tumor accumulation | rrrrrrrrGC |
r12 | nan | Alexa600 | 22285548 | 424.0 | Relative fluorescence (%) | 3 nmol | 24h | nan | CLSM | Tumor accumulation | rrrrrrrrrrrrGC |
RV24 | T98G cell | b-galactosidase and eGFP | 22326265 | 82.46 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | nan | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
RV24 | HepG2 cells | b-galactosidase and eGFP | 22326265 | 78.85 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | nan | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
RV24 | HeLa cells | b-galactosidase and eGFP | 22326265 | 74.79 | % Positive cells | Molar ratio 50 (v/w) or (w/w) eGFP | 4h | nan | Flow cytometry | Transduction | RRRRRRRRRGPGVTWTPQAWFQWV |
GST-HE-MAP | HeLa cells | GST | 22326404 | 32 | ng/ Cell monolayer | 5 ug/ml | 1h | 37ºC | Gamma-well counter | Internalization | HEHEHEHEHEHEHEHEHEHEGGGGGKLALKLALKALKAALKLA |
TMR-R3 | U251 cells | TMR | 22465335 | 54.54 | Relative fluorescence | 1 uM | 30 min | nan | Fluorescence spectroscopy | Transduction | RRR |
PasR8 (Alexa) | HeLa cells | Alexa | 22486588 | 61 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFLIPKGRRRRRRRRGC |
LILIR8 (Alexa) | HeLa cells | Alexa | 22486588 | 18.5 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | LILIGRRRRRRRRGC |
F2R8 (Alexa) | HeLa cells | Alexa | 22486588 | 22 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFGRRRRRRRGC |
F4R8 (Alexa) | HeLa cells | Alexa | 22486588 | 100 | Mean Fluorescence intensity | 1 uM | 15 min | 37ºC | Flow cytometry | Uptake | FFFFGRRRRRRRRGC |
(r-ahx-r)4_carbamate_CF (II) | CHO-K1 cells | Plasmid DNA | 22509923 | 362.5 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | rXrrXrrXrrXr |
r8_carbamate_CF15 (VI) | CHO-K1 cells | Plasmid DNA | 22509923 | 300 | Mean Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Uptake | rrrrrrrr |
Tat | Caco-2 cells | Nanoparticle | 22531849 | 3.5 | Relative Median Fluorescence | 1.0 mg/ml | 4h | nan | FACS | Uptake | GCGGGYGRKKRRQRRR |
TAT-NBD | MDA-MB-231 cells | TMTP1 | 22580115 | 15 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | YGRKKRRQRRRGTALDWSWLQTE |
TAT-NBD | MCF7 cells | TMTP1 | 22580115 | 13 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | YGRKKRRQRRRGTALDWSWLQTE |
TMTP1-TAT-NBD | MDA-MB-231 cells | TMTP1 | 22580115 | 28.75 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | CGNVVRQGC-G-YGRK-KRRQRRR-G-TALDWSWLQTE |
TMTP1-TAT-NBD | MCF7 cells | TMTP1 | 22580115 | 2.25 | Mean Fluorescence intensity | 1 umol | 30 min | 37ºC | Fluorescent Microscopy | Association | CGNVVRQGC-G-YGRK-KRRQRRR-G-TALDWSWLQTE |
SR9 | A549 cells | Plasmid DNA | 22669044 | 3.9 | Fold of transfection efficiency | N/P ratio = 3 | 10 min | 37ºC | Flow cytometry | Transfection | SRRRRRRRRR |
PR9 | A549 cells | Plasmid DNA | 22669044 | 5.6 | Fold of transfection efficiency | N/P ratio = 3 | 10 min | 37ºC | Flow cytometry | Transfection | FFLIPKGRRRRRRRRR |
CADY-1 | HeLa cells | Doxorubicin | 22688249 | 63 | % Positive cells | 10 uM | 1h | nan | HPCL-analysis | Penetration efficiencies | GLWWKAWWKAWWKSLWWRKRKRKA |
RWR | CHO-K1 cells | Carboxyfluorescein | 22712882 | 750 | Mean Fluorescence intensity | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRWWWWRRRR |
RW MIX | CHO-K1 cells | Carboxyfluorescein | 22712882 | 1400 | Mean Fluorescence intensity | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RWRRWRRWRRWR |
1 (TAT) | NHDF | FITC | 22805558 | 1.89 | Relative fluorescence | 10 uM | 3h | nan | FACS | Uptake | YGRKKRPQRRR |
CPP2 | HeLa cells | FITC | 22805558 | 4 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | Lovo | FITC | 22805558 | 39 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | A549 cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | MCF7 cells | FITC | 22805558 | 1 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | HepG2 cells | FITC | 22805558 | 5 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | U2OS cells | FITC | 22805558 | 6 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | K562 cells | FITC | 22805558 | 2 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP2 | NHDF | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | DSLKSYWYLQKFSWR |
CPP44 | HeLa cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | Lovo | FITC | 22805558 | 2 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | A549 cells | FITC | 22805558 | 1 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | MCF7 cells | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | HepG2 cells | FITC | 22805558 | 40 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | U2OS cells | FITC | 22805558 | 3 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | K562 cells | FITC | 22805558 | 70 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
CPP44 | NHDF | FITC | 22805558 | 0 | Relative fluorescence | 10 uM | 3h | nan | Fluorescent Microscopy | Penetration efficiencies | KRPTMRFRYTWNPMK |
Polyguanidine comparators 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 56.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRRRRRR |
Polyguanidine comparators 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 36 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg-Nbtg |
NLys(1/3) variants 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 11.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe |
NLys(1/3) variants 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 92.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe-NLys-Nspe-Nspe |
NLys(1/3) variants 3 | MCF7 cells | Carboxyfluorescein | 22828784 | 23.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Npm-Npm-NLys-Npm-Npm-NLys-Npm-Npm-NLys-Npm-Npm |
NLys(1/3) variants 4 | MCF7 cells | Carboxyfluorescein | 22828784 | 7.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-Nssb-Nssb-NLys-Nssb-Nssb-NLys-Nssb-Nssb-NLys-Nssb-Nssb |
NLys(2/3) variants 1 | MCF7 cells | Carboxyfluorescein | 22828784 | 12 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-Nspe-NLys-NLys-Nspe-NLys-NLys-Nspe-NLys-NLys-Nspe |
NLys(2/3) variants 2 | MCF7 cells | Carboxyfluorescein | 22828784 | 20 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLys-Nspe-Nspe-Nspe-Nspe |
NLys(2/3) variants 3 | MCF7 cells | Carboxyfluorescein | 22828784 | 3.2 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLys-NLeu-NLeu-NLeu-NLeu-Nleu |
Guanidylated variants | MCF7 cells | Carboxyfluorescein | 22828784 | 98.4 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe |
Guanidylated variants | MCF7 cells | Carboxyfluorescein | 22828784 | 92.8 | Mean Fluorescence intensity | 8 uM | 1h | 37ºC | Flow cytometry | Uptake | Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe-Nbtg-Nspe-Nspe |
penetratin | MDCK-MDR cells | PEG-PLA | 22841849 | 20 | Nanoparticle uptake/cell | 100 ug/ml | 60 min | 37ºC | HCS analysis | Uptake | RQIKIWFQNRRMKWKK |
low molecular weight protamine (LMWP) | Caco-2 cells | Insulin-PEG-LMWP | 23863452 | 0.205 | Insulin concentration | 0.5 uM | 8 hour | nan | Fluorescence spectroscopy | Absorption | VSRRRRRRGGRRRR |
Peptide 1 | U87 cells | FITC | 25562654 | 95 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | NTCTWLKYHS |
Peptide 2 | U87 cells | FITC | 25562654 | 10 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | CASGQQGLLKLC |
Peptide 3 | U87 cells | FITC | 25562654 | 25 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YNNFAYSVFL |
Peptide 4 | U87 cells | FITC | 25562654 | 16 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | ECYPKKGQDP |
Peptide 5 | U87 cells | FITC | 25562654 | 15 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | RHVYHVLLSQ |
Peptide 6 | U87 cells | FITC | 25562654 | 15 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | HATKSQNINF |
Peptide 7 | U87 cells | FITC | 25562654 | 10 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YRDRFAFQPH |
Peptide 8 | U87 cells | FITC | 25562654 | 19 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | IWRYSLASQQ |
Peptide 9 | U87 cells | FITC | 25562654 | 19 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | YQKQAKIMCS |
Peptide 10 | U87 cells | FITC | 25562654 | 20 | Fluorescence intensity | 10 uM | 2h | 37ºC | CLSM | Uptake | VQLRRRWC |
Peptide 1-C3G | U87 cells | FITC | 25562654 | 0.75 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | NTGTWLKYHS |
Peptide 1-N? | U87 cells | FITC | 25562654 | 1.2 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TCTWLKYHS |
Peptide 1-S? | U87 cells | FITC | 25562654 | 1.15 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | NTCTWLKYH |
Peptide 1-NS? | U87 cells | FITC | 25562654 | 2 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TCTWLKYH |
Peptide 1-NTS? | U87 cells | FITC | 25562654 | 1.3 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | CTWLKYH |
Peptide 1-NTCS? | U87 cells | FITC | 25562654 | 0.5 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | TWLKYH |
Peptide 1-NTHS? | U87 cells | FITC | 25562654 | 0.8 | Relative penetration efficiency | 10 uM | 2h | 37ºC | CLSM | Uptake | CTWLKY |
TV-XIIa | A549 cells | Fluorescein, oligonucleotides | 25468041 | 15 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NII-Aib-PLL-Aib-PIC-NH2 |
P-I | A549 cells | Fluorescein, oligonucleotides | 25468041 | 0 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NII-Aib-PLLAPIC-NH2 |
P-II | A549 cells | Fluorescein, oligonucleotides | 25468041 | 5 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-ANII-Aib-PLL-Aib-PIC-NH2 |
P-III | A549 cells | Fluorescein, oligonucleotides | 25468041 | 2.5 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NIIAPLL-Aib-PIC-NH2 |
P-IV | A549 cells | Fluorescein, oligonucleotides | 25468041 | 320 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NII-Aib-Aib-LL-Aib-Aib-IC-NH2 |
P-V | A549 cells | Fluorescein, oligonucleotides | 25468041 | 20 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NII-Aib-PLL-Aib-Aib-IC-NH2 |
P-VI | A549 cells | Fluorescein, oligonucleotides | 25468041 | 18 | Mean Fluorescence intensity/mg protein | 10 uM | 2h | 37ºC | Fluorometer | Uptake | CH3CO-Aib-NII-Aib-Aib-LL-Aib-PIC-NH2 |
P1 | HeLa cells | FITC | 25459448 | 112.5 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | KKKKKKNKKLQQRGD |
P2 | HeLa cells | FITC | 25459448 | 20.8 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RGDGPRRRPRKRRGR |
P3 | HeLa cells | FITC | 25459448 | 166 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRRQKRIVVRRRLIR |
P4 | HeLa cells | FITC | 25459448 | 100 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRVWRRYRRQRWCRR |
P5 | HeLa cells | FITC | 25459448 | 75 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRARRPRRLRPAPGR |
P6 | HeLa cells | FITC | 25459448 | 208.3 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | LLRARWRRRRSRRFR |
P7 | HeLa cells | FITC | 25459448 | 83.3 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RGPRRQPRRHRRPRR |
P8 | HeLa cells | FITC | 25459448 | 950 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
Tat | HeLa cells | FITC | 25459448 | 100 | Mean Fluorescence (% of positive control TAT as 100 %) | 10 uM | 1h | 37ºC | Flow cytometry | Uptake | GRKKRRQRRRPPQ |
PolyR | nan | Carboxyfluorescein | 25894337 | 70 ± 5 | % Average area uptake | 100 uM | nan | nan | Immunohistochemistry | Penetration | RRRRRRRRR |
Antp | nan | Carboxyfluorescein | 25894337 | 0.0 | % Average area uptake | 100 uM | nan | nan | Immunohistochemistry | Penetration | RQIKIWFQNRRMKWKK |
Tat(49-57) | nan | Carboxyfluorescein | 25894337 | 27 ±13 | % Average area uptake | 100 uM | nan | nan | Immunohistochemistry | Penetration | RKKRRQRRR |
Trans | nan | Carboxyfluorescein | 25894337 | 70 ± 4 | % Average area uptake | 100 uM | nan | nan | Immunohistochemistry | Penetration | GWTLNSAGYLLGKINLKALAALAKKIL |
CendRP | nan | Carboxyfluorescein | 25894337 | 0.0 | % Average area uptake | 100 uM | nan | nan | Immunohistochemistry | Penetration | RPARPAR |
R6 | HeLa cells | FITC | 25654426 | 24 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | BRRRRRR |
R7 | HeLa cells | FITC | 25654426 | 44 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | BRRRRRRR |
R8 | HeLa cells | FITC | 25654426 | 72 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | BRRRRRRRR |
R9 | HeLa cells | FITC | 25654426 | 100 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | Ahx-RRRRRRRRR |
Cyc-R4 | HeLa cells | FITC | 25654426 | 12 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRE |
Cyc-R6 | HeLa cells | FITC | 25654426 | 26 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRE |
Cyc-R7 | HeLa cells | FITC | 25654426 | 42 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRE |
Cyc-R8 | HeLa cells | FITC | 25654426 | 124 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRRE |
Cyc-R9 | HeLa cells | FITC | 25654426 | 148 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRRRE |
Cyc-r7 | HeLa cells | FITC | 25654426 | 42 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRE |
Cyc-r8 | HeLa cells | FITC | 25654426 | 64 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRRE |
Cyc-r9 | HeLa cells | FITC | 25654426 | 70 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRRRE |
Cyc-(L,D)-R6 | HeLa cells | FITC | 25654426 | 38 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRE |
Cyc-(L,D)-R7 | HeLa cells | FITC | 25654426 | 44 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRE |
Cyc-(L,D)-R8 | HeLa cells | FITC | 25654426 | 76 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XKRRRRRRRRE |
Bicyc-0-R6 | HeLa cells | FITC | 25654426 | 17 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XERRRKKRRRE |
Bicyc-1-R6 | HeLa cells | FITC | 25654426 | 20 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XERRRKKRRRE |
Bicyc-2-R6 | HeLa cells | FITC | 25654426 | 33 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XERRRKKRRRE |
Bicyc-3-R6 | HeLa cells | FITC | 25654426 | 30 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XERRRKKRRRE |
Cyc-R3-R4 | HeLa cells | FITC | 25654426 | 66 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XRRRRKRRRE |
Cyc-R4-R3 | HeLa cells | FITC | 25654426 | 95 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XRRRKRRRRE |
Cyc-R5-R2 | HeLa cells | FITC | 25654426 | 75 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XRRKRRRRRE |
Cyc-R6-R1 | HeLa cells | FITC | 25654426 | 72 | Relative Mean Fluorescence intensity (%) | 5 mM | nan | nan | Flow cytometry | Uptake | XRKRRRRRRE |
RW9 | CHO-K1 cells | nan | 25445669 | 10.375 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRWWRRWRR |
RFFF9 | CHO-K1 cells | nan | 25445669 | 0.2 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRFFRRFRR |
RFFW9 | CHO-K1 cells | nan | 25445669 | 0.5 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRFFRRWRR |
RWFF9 | CHO-K1 cells | nan | 25445669 | 0.625 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRWFRRFRR |
RFWF9 | CHO-K1 cells | nan | 25445669 | 0.25 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRFWRRFRR |
RFWW9 | CHO-K1 cells | nan | 25445669 | 1 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRFWRRWRR |
RWWF9 | CHO-K1 cells | nan | 25445669 | 0.625 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRWWRRFRR |
RWFW9 | CHO-K1 cells | nan | 25445669 | 0.5 | pmol/uM Internalized peptide | 10 uM | 1h | 37ºC | MALDI-TOF | Uptake | Biotin-GGGGRRWFRRWRR |
nan | MDA-MB-231 cells | RNA-FAM | 34948105 | 65 000 | Fluorescence intensity | nan | 30 min | nan | Flow cytometry | Transduction | FFAARTMIWYPGAWYKRI-RNA-FAM |
TAT | HeLa cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
AKIP1 | HeLa cells | Carboxyfluorescein | 34504427 | 38.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VLERAKRRAV |
CASC3 | HeLa cells | Carboxyfluorescein | 34504427 | 54.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
CCNL2 | HeLa cells | Carboxyfluorescein | 34504427 | 2.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | NTKRRLEGAKKA |
DAPK1 | HeLa cells | Carboxyfluorescein | 34504427 | 9.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AAKFIKKRRTKSS |
ING4 | HeLa cells | Carboxyfluorescein | 34504427 | 4.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TQKEKKAARARSK |
DMAP1 | HeLa cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
VP8 | HeLa cells | Carboxyfluorescein | 34504427 | 28.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | KRKGRLRSKGKK |
NOP53 | HeLa cells | Carboxyfluorescein | 34504427 | 8.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AEADKPRRLGRLK |
AHRR | HeLa cells | Carboxyfluorescein | 34504427 | 38.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
CUL4B | HeLa cells | Carboxyfluorescein | 34504427 | 16.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TPPTSAKKRKL |
FBXO32 | HeLa cells | Carboxyfluorescein | 34504427 | 4.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VAAKKRKKDML |
TAT | PC3 cells | Carboxyfluorescein | 34504427 | 64.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
AKIP1 | PC3 cells | Carboxyfluorescein | 34504427 | 60.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VLERAKRRAV |
CASC3 | PC3 cells | Carboxyfluorescein | 34504427 | 74.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
CCNL2 | PC3 cells | Carboxyfluorescein | 34504427 | 6.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | NTKRRLEGAKKA |
DAPK1 | PC3 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AAKFIKKRRTKSS |
ING4 | PC3 cells | Carboxyfluorescein | 34504427 | 6.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TQKEKKAARARSK |
DMAP1 | PC3 cells | Carboxyfluorescein | 34504427 | 22.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
VP8 | PC3 cells | Carboxyfluorescein | 34504427 | 46.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | KRKGRLRSKGKK |
NOP53 | PC3 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AEADKPRRLGRLK |
AHRR | PC3 cells | Carboxyfluorescein | 34504427 | 54.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
CUL4B | PC3 cells | Carboxyfluorescein | 34504427 | 21.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TPPTSAKKRKL |
FBXO32 | PC3 cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VAAKKRKKDML |
TAT | U87 cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GRKKRRQRRRPPQ |
AKIP1 | U87 cells | Carboxyfluorescein | 34504427 | 40.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VLERAKRRAV |
CASC3 | U87 cells | Carboxyfluorescein | 34504427 | 49.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | PDDIKPRRIRKPRY |
CCNL2 | U87 cells | Carboxyfluorescein | 34504427 | 3.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | NTKRRLEGAKKA |
DAPK1 | U87 cells | Carboxyfluorescein | 34504427 | 24.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AAKFIKKRRTKSS |
ING4 | U87 cells | Carboxyfluorescein | 34504427 | 11.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TQKEKKAARARSK |
DMAP1 | U87 cells | Carboxyfluorescein | 34504427 | 32.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | RKRRESASSSSSVKKAKKP |
VP8 | U87 cells | Carboxyfluorescein | 34504427 | 28.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | KRKGRLRSKGKK |
NOP53 | U87 cells | Carboxyfluorescein | 34504427 | 10.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | AEADKPRRLGRLK |
AHRR | U87 cells | Carboxyfluorescein | 34504427 | 36.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | GECTYAGRKRRRPLQK |
CUL4B | U87 cells | Carboxyfluorescein | 34504427 | 18.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | TPPTSAKKRKL |
FBXO32 | U87 cells | Carboxyfluorescein | 34504427 | 3.0 | % Positive cells | 10 uM | 2h | nan | Flow cytometry | Internalization | VAAKKRKKDML |
RALA | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 61.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
HALA1 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 45.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
HALA2 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 62.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
HALA3 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 27.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
HALA4 | HeLa cells | pCMV-EGFP plasmid DNA | 34443195 | 40.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
RALA | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 41.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
HALA1 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 39.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
HALA2 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 56.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
HALA3 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 21.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
HALA4 | HEK293T cells | pCMV-EGFP plasmid DNA | 34443195 | 55.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
RALA | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 13.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALARALRACEA |
HALA1 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 10.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALARALARHLARALARALRACEA |
HALA2 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 25.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLARALAHALHACEA |
HALA3 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 4.0 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEAHLAHALAHALARHLARALARALRACEA |
HALA4 | A549 cells | pCMV-EGFP plasmid DNA | 34443195 | 8.5 | % Positive cells | N/P ratio 6 | 6h | 37ºC | Flow cytometry | Transfection | WEARLARALARALARHLAHALAHALHACEA |
PDL | SH-SY5Y cells | EGFP pDNA | 34361142 | 31.10 ± 0.5 | % Transfection | plasmid/PDL ratio 1:4 | 48h | 37ºC | Flow cytometry | Transfection | kkk |
PDL | HeLa cells | EGFP pDNA | 34361142 | 1.33 ± 0.18 | % Transfection | plasmid/PDL ratio 1:4 | 48 h | 37ºC | Flow cytometry | Transfection | kkk |
PDL | NIH-3T3 cells | EGFP pDNA | 34361142 | 0.16 ± 0.03 | % Transfection | plasmid/PDL ratio 1:4 | 48 h | 37ºC | Flow cytometry | Transfection | kkk |
TAT | H1299 | 111In-GFP-G1 | 33789931 | 6.8 | Relative Cellular uptake | 1.5 nM | 1h | 37ºC | Flow cytometry | Uptake | GRKKRRQRRRPPQGYG |
Tat(48-57) | HEK293 cells | TAMRA | 33589718 | 68333 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRR |
CTP | HEK293 cells | TAMRA | 33589718 | 43333 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GGRRARRRRRR |
TatsMTS (TMG) | HEK293 cells | TAMRA | 33589718 | 80000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRMVSAL |
Tat(49-57) | HEK293 cells | TAMRA | 33589718 | 48333 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | RKKRRQRRR |
Tat | HEK293 cells | TAMRA | 33589718 | 45833 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPPQRKC |
Tat(47-57) | HEK293 cells | TAMRA | 33589718 | 72500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YGRKKRRQRRR |
6-Oct | HEK293 cells | TAMRA | 33589718 | 73333 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKRKKRT |
K9 | HEK293 cells | TAMRA | 33589718 | 72500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | KKKKKKKKK |
D-R9 | HEK293 cells | TAMRA | 33589718 | 34166 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | RRRRRRRRR |
HIV-1 TAT peptide--Crystallins | HEK293 cells | TAMRA | 33589718 | 48333 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPQ |
CRGDK | HEK293 cells | TAMRA | 33589718 | 56666 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | CRGDK |
PAF95 | HEK293 cells | TAMRA | 33589718 | 39166 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | AAAWFW |
iRGD | HEK293 cells | TAMRA | 33589718 | 37500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | CRGDKGDPC |
Ypep-GFP-Ypep | HEK293 cells | TAMRA | 33589718 | 5000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQYTFGLKTSFNVQ |
VP1 BC loop (V) peptides | HEK293 cells | TAMRA | 33589718 | 41666 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | TVDNPASTTNKDKLFAVRK |
Peptide 1-NTCS | HEK293 cells | TAMRA | 33589718 | 55000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | TWLKYH |
Ypep-GFP | HEK293 cells | TAMRA | 33589718 | 10000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQ |
CPPP-2 | HEK293 cells | TAMRA | 33589718 | 30000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | KLPVM |
TCTPPTD | HEK293 cells | TAMRA | 33589718 | 40000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | MIIYRDLISH |
ARF(1-22) | HEK293 cells | TAMRA | 33589718 | 0 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | MVRRFLVTLRIRRACGPPRVRV |
Tat(48-57) | CHO cells | TAMRA | 33589718 | 3500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRR |
CTP | CHO cells | TAMRA | 33589718 | 2500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GGRRARRRRRR |
TatsMTS (TMG) | CHO cells | TAMRA | 33589718 | 7000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRMVSAL |
Tat(49-57) | CHO cells | TAMRA | 33589718 | 3000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | RKKRRQRRR |
Tat | CHO cells | TAMRA | 33589718 | 8000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPPQRKC |
Tat(47-57) | CHO cells | TAMRA | 33589718 | 3000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YGRKKRRQRRR |
6-Oct | CHO cells | TAMRA | 33589718 | 5000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKRKKRT |
K9 | CHO cells | TAMRA | 33589718 | 9000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | KKKKKKKKK |
D-R9 | CHO cells | TAMRA | 33589718 | 3500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | RRRRRRRRR |
HIV-1 TAT peptide--Crystallins | CHO cells | TAMRA | 33589718 | 7000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | GRKKRRQRRRPQ |
CRGDK | CHO cells | TAMRA | 33589718 | 16500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | CRGDK |
PAF95 | CHO cells | TAMRA | 33589718 | 20000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | AAAWFW |
iRGD | CHO cells | TAMRA | 33589718 | 2000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | CRGDKGDPC |
Ypep-GFP-Ypep | CHO cells | TAMRA | 33589718 | 6000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQYTFGLKTSFNVQ |
VP1 BC loop (V) peptides | CHO cells | TAMRA | 33589718 | 16000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | TVDNPASTTNKDKLFAVRK |
Peptide 1-NTCS | CHO cells | TAMRA | 33589718 | 11000 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | TWLKYH |
Ypep-GFP | CHO cells | TAMRA | 33589718 | 5500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | YTFGLKTSFNVQ |
CPPP-2 | CHO cells | TAMRA | 33589718 | 7500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | KLPVM |
TCTPPTD | CHO cells | TAMRA | 33589718 | 4500 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | MIIYRDLISH |
ARF(1-22) | CHO cells | TAMRA | 33589718 | 0 | Mean Fluorescence intensity | 5 ug | 16h | nan | Flow cytometry | Penetration efficiencies | MVRRFLVTLRIRRACGPPRVRV |
KYKGAIIGNIK | HEK293T cells | pGL3-SV40 | 31861408 | 102500 | RFU/mg | pDNA/peptide ratio 1:2500 | 4h | 37ºC | Fluorescent Microscopy | Transfection | KYKGAIIGNIK |
KYRSGAITIGY | HEK293T cells | pGL3-SV40 | 31861408 | 175000 | RFU/mg | pDNA/peptide ratio 1:2500 | 4h | 37ºC | Fluorescent Microscopy | Transfection | KYRSGAITIGY |
4Iphf-HN1 | Cal 27 | IR800 | 31450798 | 0.55 | Fluorescence intensity | 10 uM | 2h | nan | Fluorescent Microscopy | Uptake | TSPLNIHNGQKL |
f-HN1 | Cal 27 | IR800 | 31450798 | 1 | Fluorescence intensity | 10 uM | 2h | nan | Fluorescent Microscopy | Uptake | TSPLNIHNGQKL |
HNJ | Cal 27 | IR800 | 31450798 | 0.3 | Fluorescence intensity | 10 uM | 2h | nan | Fluorescent Microscopy | Uptake | NQHSKNTLLIGP |
4Iphf-HN17 | Cal 27 | IR800 | 31450798 | 4.5 | Fluorescence intensity | 10 uM | 2h | nan | Fluorescent Microscopy | Uptake | LPNSNHIKQGL |
f-HN17 | Cal 27 | IR800 | 31450798 | 1.70 | Fluorescence intensity | 10 uM | 2h | nan | Fluorescent Microscopy | Uptake | TLPNSNHIKQGL |
iPTD | HEK293T cells | Fab-F2 | 31375703 | 7750 | Mean Fluorescence intensity | 10 ug/mL | 24h | nan | Flow cytometry | Internalization | MALGPCMLLLLLLLGLRLPGVWAPPRRRRRRRRR |
CPP9 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.175E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | FRRRRQ |
CPP12 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | FRRRRQ |
aPP5.3 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MGPSQPTYPGDDAPVRDLIRFYRDLRRYLNVVTRHRY |
R8 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.725E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MRRRRRRR |
ZiF | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 0.75E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MLEPGEKPYKCPECGKSFSASAALVAHQRTHTGKKTS |
Pen | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 1.4E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MRQIKIWFQNRRMKWKK |
ZF5.3 | Saos-2 cells | Rho-labeled SNAP-tag | 30410976 | 2.125E-3 | Average Median Fluorescence intensity | 1 uM | 30 min | 37ºC | Flow cytometry | Uptake | MYSCNVCGKAFVLSRHLNRHLRVHRRAT |
TAT | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 22.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | GRKKRRQRRRPPQRKC |
84 | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 36.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | RKQKSLQTKLAENPPVPRKKRQSRPRWKQWLQK |
1746 | HEK293 cells | EDB_S11 (protein fusions) | 30135446 | 72.0 | % Green viable cells | 40 uM | 1h | 37ºC | Flow cytometry | Uptake (Endosomal escape) | PLKPKKPKTQEKKKKQPPKPKKPKTQEKKKKQPPKPKR |
PPC1 | eGFP HeLa 654 | PMO | 29721534 | 18400 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | KQPRIKRKK |
PPC2 | eGFP HeLa 654 | PMO | 29721534 | 17500 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | LKKRRKLPKKKPIRNEQ |
PPC3 | eGFP HeLa 654 | PMO | 29721534 | 23640 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | KKYRGRKRHPR |
PPC4 | eGFP HeLa 654 | PMO | 29721534 | 21370 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | APKRKKLKKRF |
PPC5 | eGFP HeLa 654 | PMO | 29721534 | 18640 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | GRKAARAPGRRKQ |
NS1 | eGFP HeLa 654 | PMO | 29721534 | 5000 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | HDLPKGG |
NS2 | eGFP HeLa 654 | PMO | 29721534 | 9320 | Mean Fluorescence intensity | 5 uM | 22h | 37ºC | Flow cytometry | Uptake | AGSHRRL |
IMT-P8 | HeLa cells | KLA | 27189051 | 285000 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
IMT-P8 | MDA-MB-231 cells | KLA | 27189051 | 161600 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
IMT-P8 | PC3 cells | KLA | 27189051 | 1037500 | Mean Fluorescence intensity | 2.5 uM | 30 min | 37ºC | Flow cytometry | Uptake | RRWRRWNRFNRRRCR |
HR9 | A549 cells | FITC | 26942714 | 94.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | CHHHHHRRRRRRRRRHHHHHC |
Lfcin | A549 cells | FITC | 26942714 | 94.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | CRRWQWRMKKLGC |
L12 | A549 cells | FITC | 26942714 | 97.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | FKCRRWQWRMKK |
L11 | A549 cells | FITC | 26942714 | 93.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | KCRRWQWRMKK |
L9 | A549 cells | FITC | 26942714 | 77.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQWRMKK |
L6 | A549 cells | FITC | 26942714 | 98.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQWR |
L5a | A549 cells | FITC | 26942714 | 95.5 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RRWQW |
L5b | A549 cells | FITC | 26942714 | 25.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RWQWR |
L4 | A549 cells | FITC | 26942714 | 9.0 | % Positive cells | 10 uM | 1h | 37ºC | Flow cytometry | Internalization | RWQW |
TAT | N2a cells | BoNTA | 35223792 | 158.75 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | GRKKRRQRRRPQ |
Pep1 | N2a cells | BoNTA | 35223792 | 117.5 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | KETWWETWWTEWSQPKKKRKV |
ZFP3 (N-Terminal) | N2a cells | BoNTA | 35223792 | 110.0 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
ZFP3 (C-Terminal) | N2a cells | BoNTA | 35223792 | 120.0 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
ZFP3 (N and C-Terminal) | N2a cells | BoNTA | 35223792 | 177.5 | Relative fluorescence (%) | 100 nM | 2h | 37ºC | Immunofluorescence analysis | Cellular uptake | EKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTGEKPYKCPECGKSFSASAALVAHQRTHTG |
SynB1 | MCF7 cells | ELP-DOXO | 35216417 | 3.2 | RFU | 2 uM dox equivalent concentration | 24h | nan | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
SynB1 | MCF7 cells | ELP-GFLG-NCDox | 35216417 | 0.8 | RFU | 2 uM dox equivalent concentration | 24h | nan | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
SynB1 | NCI/ADR | ELP-DOXO | 35216417 | 1.3 | RFU | 2 uM dox equivalent concentration | 24h | nan | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
SynB1 | NCI/ADR | ELP-GFLG-NCDox | 35216417 | 1.1 | RFU | 2 uM dox equivalent concentration | 24h | nan | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGR-VPGXGVPGXGVPGXG |
Cys-Penetratin | TR146 cell | Liposomes-salmon calcitonin (sCT) | 35210769 | 3800 | Relative Mean Fluorescence intensity | nan | 2h | 37ºC | Flow cytometry | Relative uptake | CRQIKIWFQNRRMKWKK |
PepFect 14 (PF14) | MiaPaCa-2 | Cy3-labeled AON | 35098567 | 26 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Stearyl-AGYLLGKLLOOLAAAALOOLL-NH2 |
R9 | MiaPaCa-2 | Cy3-labeled AON | 35098567 | 10 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-RRRRRRRRR-NH2 |
r9 | MiaPaCa-2 | Cy3-labeled AON | 35098567 | 2 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-rrrrrrrrr-NH2 |
hLF | MiaPaCa-2 | Cy3-labeled AON | 35098567 | 10 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-KCFQWQRNMRKVRGPPVSCIKR-NH2 |
PepFect 14 (PF14) | VCaP | Cy3-labeled AON | 35098567 | 34 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Stearyl-AGYLLGKLLOOLAAAALOOLL-NH2 |
R9 | VCaP | Cy3-labeled AON | 35098567 | 6 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-RRRRRRRRR-NH2 |
r9 | VCaP | Cy3-labeled AON | 35098567 | 3.5 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-rrrrrrrrr-NH2 |
hLF | VCaP | Cy3-labeled AON | 35098567 | 4 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-KCFQWQRNMRKVRGPPVSCIKR-NH2 |
PepFect 14 (PF14) | HeLa cells | Cy3-labeled AON | 35098567 | 36 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Stearyl-AGYLLGKLLOOLAAAALOOLL-NH2 |
R9 | HeLa cells | Cy3-labeled AON | 35098567 | 5 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-RRRRRRRRR-NH2 |
r9 | HeLa cells | Cy3-labeled AON | 35098567 | 4 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-rrrrrrrrr-NH2 |
hLF | HeLa cells | Cy3-labeled AON | 35098567 | 4 | Median Fluorescence intensity | N/P ratio 5, 0.5 uM oligonucleotide | 2h | 37ºC | Flow cytometry | Uptake | Ac-KCFQWQRNMRKVRGPPVSCIKR-NH2 |
G2R2 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.055 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRR |
G2R4 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.15 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRRRR |
G4R8 | HeLa cells | Somatropin-Hyaluronic acid | 35093459 | 0.10 | C/M ratio of somatropin (mL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGGGRRRRRRRR |
G2R2 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 1.225 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRR |
G2R4 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 1.65 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGRRRR |
G4R8 | HeLa cells | Exendin-4-Hyaluronic acid | 35093459 | 2.125 | C/M ratio of exendin-4 (uL/mg protein) | 50 ug/ml | 2h | 37ºC | ELISA | Uptake | GGGGRRRRRRRR |
Crotamine | P. falciparum-infected erythrocytes | Cy3-labeled Crotamine | 35074306 | 46.0 | % Internalization | 5 uM | 30 min | 37ºC | Flow cytometry | Internalization | YKQCHKKGGHCFPKEKICLPPSSDFGKMDCRWRWKCCKKGSG |
CKRRMKWKK | HepG2 cells | siRNA | 35024246 | 3600 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | HepG2 cells | siRNA-TSL | 35024246 | 1600 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | HepG2 cells | siRNA-MTSL | 35024246 | 2100 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | HepG2 cells | siRNA-MTSLR | 35024246 | 2550 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | HepG2 cells | siRNA-MTSLR-H | 35024246 | 3900 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | RAW264.7 cells | siRNA-TSL | 35024246 | 1200 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | RAW264.7 cells | siRNA-MTSL | 35024246 | 750 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
CKRRMKWKK | RAW264.7 cells | siRNA-MTSLR | 35024246 | 875 | Mean Fluorescence intensity | 100 uM | 4h | nan | Flow cytometry | Cellular uptake | CKRRMKWKK-Cys |
TmP(Glu)4 | HeLa cells | (alpha-D-glucose)4-TAMRA | 34994362 | 545 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
TmP(Glu)6 | HeLa cells | (alpha-D-glucose)6-TAMRA | 34994362 | 660 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
TmP(Man)4 | HeLa cells | (alpha-D-mannose)4-TAMRA | 34994362 | 860 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
TmP(Man)6 | HeLa cells | (alpha-D-mannose)6-TAMRA | 34994362 | 720 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
TmP(Gal)4 | HeLa cells | (alpha-D-galactose)4-TAMRA | 34994362 | 845 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | RKLRRLLRRLKRL |
TmP(Gal)6 | HeLa cells | (alpha-D-galactose)6-TAMRA | 34994362 | 730 | RFU | 10 uM | 30 min | nan | Flow cytometry | Internalization efficency | KRKLRRLLRRLKRL |
Arg | HeLa cells | Carboxyfluorescein | 30718681 | 180 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Arg | HeLa cells | Carboxyfluorescein | 30718681 | 180 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Arg | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Leu | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
Leu | HeLa cells | Carboxyfluorescein | 30718681 | 35 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
Leu | HeLa cells | Carboxyfluorescein | 30718681 | 25 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
(?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 70 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
(?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 135 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
(?Me)Leu | HeLa cells | Carboxyfluorescein | 30718681 | 120 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 30 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 45 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5cdOM | HeLa cells | Carboxyfluorescein | 30718681 | 60 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 50 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 70 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
Ac5c | HeLa cells | Carboxyfluorescein | 30718681 | 60 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 18 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 12 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Arg | CHO-K1 cells | Carboxyfluorescein | 30718681 | 1 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RRR)3-NH2 |
Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 1 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RRL)3-NH2 |
(?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 15 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
(?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 22 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
(?Me)Leu | CHO-K1 cells | Carboxyfluorescein | 30718681 | 11 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-(S)-(?Me)Leu)3-NH2 |
Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 5 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 11 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5cdOM | CHO-K1 cells | Carboxyfluorescein | 30718681 | 10 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-(S,S)-Ac5cdOM)3-NH2 |
Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 20 | Mean Fluorescence intensity | 1 uM | 2h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 40 | Mean Fluorescence intensity | 1 uM | 6h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
Ac5c | CHO-K1 cells | Carboxyfluorescein | 30718681 | 10 | Mean Fluorescence intensity | 1 uM | 24h | nan | Flow cytometry | Uptake | CF-G(RR-Ac5c)3-NH2 |
KFE8-Tat | BMDC | FITC | 32686113 | 10 | % Positive cells | 0.5uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
KFE8-Tat | BMDC | FITC | 32686113 | 25 | % Positive cells | 1uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
KFE8-Tat | BMDC | FITC | 32686113 | 35 | % Positive cells | 2uM | 4h | 37ºC | Flow cytometry | Nanofiber uptake | FKFEFKFESGSGSG-RKKRRQRRRPQ |
CyLoP-1 | HeLa cells | FITC | 27836642 | 250 | Mean Fluorescence intensity | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
CyLoP-1 | HeLa cells | FITC | 27836642 | 260 | Mean Fluorescence intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
CyLoP-1 | HeLa cells | FITC | 27836642 | 350 | Mean Fluorescence intensity | 15uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
CyLoP-1 | HeLa cells | FITC | 27836642 | 400 | Mean Fluorescence intensity | 20uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
CyLoP-1 | HeLa cells | FITC | 27836642 | 450 | Mean Fluorescence intensity | 30uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
CyLoP-1 | HeLa cells | FITC | 27836642 | 500 | Mean Fluorescence intensity | 40uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CRWRWKCCKK |
diTatBim | HeLa cells | AT520 | 29275934 | 50 | Mean Fluorescence intensity | 5uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-EIWIAQELRRIGDEFNAYYARLL-C-C-LLRAYYANFEDGIRRLEQAIWIE-RRRQRRKKR |
mTatBim | HeLa cells | AT521 | 29275934 | 90 | Mean Fluorescence intensity | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-EIWIAQELRRIGDEFNAYYARLL-C |
NP1-EPT | CHO-K1 cells | EPT | 30673275 | 25 | Mean Fluorescence intensity | nan | nan | nan | FACS | Cellular uptake | stearyl-HHHHHHHHHHHHHHHH-RRRRRRRR-NH2 |
NP1-EPT-2X | CHO-K1 cells | EPT | 30673275 | 15 | Mean Fluorescence intensity | nan | nan | nan | FACS | Cellular uptake | stearyl-HHHHHHHHHHHHHHHH-RRRRRRRR-NH3 |
RRCPP | B16 cells | RRCPP/siRNA | 34375118 | 0 | nan | nan | nan | nan | FACS | Cellular uptake | RGDRRRRRRRRR |
Cys-Trp-Trp-Arg8-Cys-Arg8- Cys-Arg8-Cys | Dendritic cells | peptide/OVA-Cy5.5 | 29359945 | 18 000 | Fluorescence intensity | nan | 4h | nan | Flow cytometry | Antigen Uptake | CWWRRRRRRRRCRRRRRRRRCRRRRRRRRC |
CLIP6 | Dendritic cells | FITC | 31339694 | 50 | Fluorescence intensity | 10uM | 24h | 37ºC | FACS | Cellular uptake | KVRVRVRVDPPTRVRERVKC |
[(RW)5K](RW) | CCRF-CEM cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)2 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 100 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)3 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 200 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)4 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 300 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)5 | CCRF-CEM cells | F'-GpYEEI | 34491768 | 500 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW) | SK-OV-3 cells | F'-GpYEEI | 34491768 | 100 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)2 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)3 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 120 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)4 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 130 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
[(RW)5K](RW)5 | SK-OV-3 cells | F'-GpYEEI | 34491768 | 130 | Mean Fluorescence intensity | 10uM | 3h | nan | FACS | Cellular uptake | RWRWRWRWRWKRWRWRWRWRW |
PLL | Caco-2 cells | TPP | 33360901 | 18 | Cellular uptake | nan | 3h | nan | CLSM | Cellular uptake | poly-L-lysine |
PLL | Caco-2 cells | PA | 33360901 | 15 | Cellular uptake | nan | 3h | nan | CLSM | Cellular uptake | poly-L-lysine |
P1 | HSC-T6 | FITC | 34338123 | 800 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
P1 | A549 cells | FITC | 34338123 | 750 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
P1 | BV2 | FITC | 34338123 | 750 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
P1 | MCF7 cells | FITC | 34338123 | 900 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | (Acp)-KKKKKRFSFKKSFKLSGFSFKKNKK |
r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 2,60E+05 | Mean Fluorescence intensity | 0.5uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRC |
r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 2,80E+05 | Mean Fluorescence intensity | 1uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRC |
r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 4,80E+05 | Mean Fluorescence intensity | 2uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRC |
Deca-r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 1,30E+05 | Mean Fluorescence intensity | 0.25uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRKC |
Deca-r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 1,50E+05 | Mean Fluorescence intensity | 0.5uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRKC |
Deca-r8-PNA | HeLa pLuc/705 cells | AlexaFluor555 (AF555) | 31581514 | 3,50E+05 | Mean Fluorescence intensity | 1uM | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRRKC |
GO-PEI-PEG-CPP | MDA-MB-231 cells | siRNA | 34916779 | 1,00E+02 | Fluorescence intensity | nan | 24h | nan | Flow cytometry | Cellular uptake | RRRXRRRR |
Sc18 | HeLa cells | daunorubicin (Dau) | 34959356 | 1,00E+00 | Relative fluorescence | nan | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB1-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 0 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB2-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 1000 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB3-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 2500 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB4-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 11000 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB5-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 2500 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB1-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 100 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB2-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 300 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB3-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 350 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB4-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 1100 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
CB5-sC18 | HeLa cells | daunorubicin (Dau) | 34959356 | 200 | Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 500 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 600 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 1500 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 1000 | Hoechst fluorescence intensity | 10uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 2500 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 2000 | Hoechst fluorescence intensity | 20uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 3000 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 3200 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 4000 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 3750 | Hoechst fluorescence intensity | 30uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 4750 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 5500 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 3500 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 5400 | Hoechst fluorescence intensity | 40uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-1 | HeLa cells | Carboxyfluorescein | 30665017 | 5800 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-2 | HeLa cells | Carboxyfluorescein | 30665017 | 6600 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
SARTHI-3 | HeLa cells | Carboxyfluorescein | 30665017 | 7500 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | KRKIFLRCKILV |
SARTHI-4 | HeLa cells | Carboxyfluorescein | 30665017 | 7000 | Hoechst fluorescence intensity | 50uM | 4h | 37ºC | Fluorescence spectroscopy | Cellular uptake | VLIKCRLFIKRK |
P2 | HeLa cells | FITC | 34463179 | 1700 | Fluorescence intensity | 5 uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
P2 | MCF7 cells | FITC | 34463179 | 1400 | Fluorescence intensity | 5 uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
P2 | HepG2 cells | FITC | 34463179 | 1400 | Fluorescence intensity | 5 uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
P2 | A549 cells | FITC | 34463179 | 1000 | Fluorescence intensity | 5 uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
P2 | HSC-T6 | FITC | 34463179 | 800 | Fluorescence intensity | 5 uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | (Acp)-RKRRQTSMTDFYHSKRRLIFS |
R8 | U87 cells | LP | 30591464 | 7 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
R8 | U87 cells | PLP | 30591464 | 12 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR |
Tat | CHO cells | icg-labeled lactosomes | 27877876 | 0.38 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | YGRKKRRQRRR-C |
PTD4 | CHO cells | icg-labeled lactosomes | 27877876 | 0.1 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | YARAAARQARA-C |
DPV3 | CHO cells | icg-labeled lactosomes | 27877876 | 0.4 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRRESRKKRRRES-C |
MPG?nlS | CHO cells | icg-labeled lactosomes | 27877876 | 0.39 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | GALFLGFLGAAGSTMGAWSQPKSKRKV-C |
R9MPG | CHO cells | icg-labeled lactosomes | 27877876 | 0.5 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRGALFLAFLAAALSLMG-C |
Pep1 | CHO cells | icg-labeled lactosomes | 27877876 | 0.6 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | KETWWETWWTEWSQPKKKRKV-C |
EB1 | CHO cells | icg-labeled lactosomes | 27877876 | 1 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | LIRLWSHLIHIWFQNRRLKWKKK-C |
PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 2.7 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 5.2 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
PB1-F2 fragment 1 | HEK293T cells | luciferin | 28284862 | 11.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-GSLKTRVLKR-NH2 |
PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 2.3 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 3.1 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 5.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
PB1-F2 fragment 2 | HEK293T cells | luciferin | 28284862 | 16.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-SLKTRVLKRW-NH2 |
PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 2.1 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 3.1 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 7.5 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
PB1-F2 fragment 3 | HEK293T cells | luciferin | 28284862 | 30.1 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKTRVLKRWK-NH2 |
PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 3.2 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 9.8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
PB1-F2 fragment 4 | HEK293T cells | luciferin | 28284862 | 30.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KTRVLKRWKL-NH2 |
PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 2.3 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 18.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
PB1-F2 fragment 5 | HEK293T cells | luciferin | 28284862 | 216.3 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-TRVLKRWKLF-NH2 |
PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 3.4 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 12 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
PB1-F2 fragment 6 | HEK293T cells | luciferin | 28284862 | 198.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RVLKRWKLFN-NH2 |
PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 1.9 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 2.8 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 6.2 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
PB1-F2 fragment 7 | HEK293T cells | luciferin | 28284862 | 30.3 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-VLKRWKLFNK-NH2 |
PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 2.5 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 3.3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
PB1-F2 fragment 8 | HEK293T cells | luciferin | 28284862 | 34.5 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-LKRWKLFNKQ-NH2 |
PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 6.5 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
PB1-F2 fragment 9 | HEK293T cells | luciferin | 28284862 | 13.6 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KRWKLFNKQE-NH2 |
PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 2.7 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 3.5 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 7.3 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
PB1-F2 fragment 10 | HEK293T cells | luciferin | 28284862 | 18.2 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-RWKLFNKQEW-NH2 |
PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 3.3 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 8 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
PB1-F2 fragment 11 | HEK293T cells | luciferin | 28284862 | 14.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-WKLFNKQEWT-NH2 |
PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 1.8 | Cellular uptake | 1.9 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 2.4 | Cellular uptake | 5.6 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 4.7 | Cellular uptake | 16.7 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
PB1-F2 fragment 12 | HEK293T cells | luciferin | 28284862 | 9.7 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Mpa(luc)-KLFNKQEWTN-NH2 |
1-luc | HEK293T cells | luciferin | 28284862 | 5.8 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
1-luc | HEK293T cells | luciferin | 28284862 | 8.7 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
1-luc | HEK293T cells | luciferin | 28284862 | 14.5 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
1-luc | HEK293T cells | luciferin | 28284862 | 22.8 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-NH2 |
2-luc | HEK293T cells | luciferin | 28284862 | 6.2 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
2-luc | HEK293T cells | luciferin | 28284862 | 10.6 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
2-luc | HEK293T cells | luciferin | 28284862 | 22.3 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
2-luc | HEK293T cells | luciferin | 28284862 | 61 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-RRRRR-NH2 |
5-luc | HEK293T cells | luciferin | 28284862 | 11.6 | Cellular uptake | 6.3 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
5-luc | HEK293T cells | luciferin | 28284862 | 21.3 | Cellular uptake | 12.5 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
5-luc | HEK293T cells | luciferin | 28284862 | 36.1 | Cellular uptake | 25 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
5-luc | HEK293T cells | luciferin | 28284862 | 66.8 | Cellular uptake | 50 uM | 1h | 37ºC | Cytotoxicity analysis | Cellular uptake | Ac-CVAKYHGYPWCRRR-TRVLKRWKLF-NH2 |
Tf-LPs | U87 cells | Doxorubicin | 31574945 | 40 | Fluorescence intensity | nan | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRR |
Tf-LPs | GL261 cells | Doxorubicin | 31574945 | 45 | Fluorescence intensity | nan | 4h | nan | Flow cytometry | Cellular uptake | RRRRRRRR |
PAS-pHK | MCF7 cells | miR-126 | 32491855 | 95 | % Internalization | 25 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GKPILFF |
CAAKA | A375 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | A375 cells | QDs | 30240193 | 17 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | MSTO cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | MSTO cells | QDs | 30240193 | 25 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | LN18 cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
CAAKA | U87 cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | CAAKA |
HSV1-VP22 | A375 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | A375 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | MSTO cells | QDs | 30240193 | 13 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | MSTO cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | 9L cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | 9L cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | LN18 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HSV1-VP22 | U87 cells | QDs | 30240193 | 36 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*DAATATRGRSAASRPTERPRAPARSASRPRRPVD |
HIV-TAT | A375 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | MSTO cells | QDs | 30240193 | 4 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | MSTO cells | QDs | 30240193 | 22 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | 9L cells | QDs | 30240193 | 2 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | 9L cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | LN18 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-TAT | U87 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*YGRKKRRQRRR |
HIV-gp41 | A375 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | A375 cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | MSTO cells | QDs | 30240193 | 21 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | MSTO cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | 9L cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | 9L cells | QDs | 30240193 | 8 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | LN18 cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
HIV-gp41 | U87 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*GALFLGWLGAAGSTMGA |
Ku-70 | A375 cells | QDs | 30240193 | 30 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | A375 cells | QDs | 30240193 | 75 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | MSTO cells | QDs | 30240193 | 50 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | 9L cells | QDs | 30240193 | 26 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | 9L cells | QDs | 30240193 | 30 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | LN18 cells | QDs | 30240193 | 45 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
Ku-70 | U87 cells | QDs | 30240193 | 50 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*PMLKE |
hCT(9-32) | A375 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | A375 cells | QDs | 30240193 | 90 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | MSTO cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | 9L cells | QDs | 30240193 | 55 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | 9L cells | QDs | 30240193 | 100 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | LN18 cells | QDs | 30240193 | 20 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
hCT(9-32) | U87 cells | QDs | 30240193 | 40 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*LGTYTQDFNKFHTFPQTAIGVGAP |
integrin ß3 | A375 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | MSTO cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | 9L cells | QDs | 30240193 | 2 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | 9L cells | QDs | 30240193 | 4 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | LN18 cells | QDs | 30240193 | 3 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
integrin ß3 | U87 cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*VTVLALGALAGVGVG |
K-FGF | A375 cells | QDs | 30240193 | 6 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | A375 cells | QDs | 30240193 | 10 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | MSTO cells | QDs | 30240193 | 15 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | MSTO cells | QDs | 30240193 | 18 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | 9L cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | 9L cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | LN18 cells | QDs | 30240193 | 5 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
K-FGF | U87 cells | QDs | 30240193 | 23 | Microscopic fluorescence intensity | 1 nM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | C*AAVALLPAVLLAHLLAP |
His8 | N. tabacum cells | MBP-RFP | 33791772 | 400 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
His12 | N. tabacum cells | MBP-RFP | 33791772 | 1000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
His16 | N. tabacum cells | MBP-RFP | 33791772 | 1500 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
His20 | N. tabacum cells | MBP-RFP | 33791772 | 2800 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
His8 | O. Sativa cells | MBP-RFP | 33791772 | 1000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
His12 | O. Sativa cells | MBP-RFP | 33791772 | 1100 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
His16 | O. Sativa cells | MBP-RFP | 33791772 | 3000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
His20 | O. Sativa cells | MBP-RFP | 33791772 | 2900 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
His8 | C. japonica cells | MBP-RFP | 33791772 | 800 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHH |
His12 | C. japonica cells | MBP-RFP | 33791772 | 2000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHH |
His16 | C. japonica cells | MBP-RFP | 33791772 | 6000 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHH |
His20 | C. japonica cells | MBP-RFP | 33791772 | 10100 | Fluorescence intensity | 5 uM | 24h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
His6 | N. tabacum cells | MBP-RFP-CyaA | 33791772 | 180 | Fluorescence intensity | 2 uM | 6h | 27ºC | CLSM | Cellular uptake | HHHHHH |
His20 | N. tabacum cells | MBP-RFP-CyaA | 33791772 | 350 | Fluorescence intensity | 2 uM | 6h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
His6 | O. Sativa cells | MBP-RFP-CyaA | 33791772 | 150 | Fluorescence intensity | 2 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHH |
His20 | O. Sativa cells | MBP-RFP-CyaA | 33791772 | 380 | Fluorescence intensity | 2 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
His6 | C. japonica cells | MBP-RFP-CyaA | 33791772 | 100 | Fluorescence intensity | 0.5 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHH |
His20 | C. japonica cells | MBP-RFP-CyaA | 33791772 | 160 | Fluorescence intensity | 0.5 uM | 1h | 27ºC | CLSM | Cellular uptake | HHHHHHHHHHHHHHHHHHHH |
Xentry-KALA (XK) | ARPE-19 cells | Cx43AsODN) | 30050146 | 0 | Fluorescence | 1 uM | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | (biotin)-lclrpvgggweaklakalakalakhlakalakalkacea |
Xentry-Protamine (XP) | ARPE-19 cells | Cx43AsODN) | 30050146 | 0 | Fluorescence | 1 uM | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | (biotin)-lclrpvggrsqsrsryyrqrqrsrrrrrrs |
WRAP1 | U87 cells | siRNA | 32135145 | 0 | nan | nan | 24h | nan | CLSM | Cellular uptake | NH2-LLWRLWRLLW-RLWRLL-CONH2 |
WRAP5 | U87 cells | siRNA | 32135145 | 0 | nan | nan | 24h | nan | CLSM | Cellular uptake | NH2-LLRLLRWWWRLLRLL-CONH2 |
pHK-PASA488 | HeLa cells | HKII | 28183803 | 1,50E+03 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | HeLa cells | HKII | 28183803 | 1,00E+04 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | HeLa cells | HKII | 28183803 | 1,70E+04 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | HeLa cells | HKII | 28183803 | 1,60E+04 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHKA489 | HeLa cells | HKII | 28183803 | 1,80E+02 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | HeLa cells | HKII | 28183803 | 1,20E+03 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA489 | HeLa cells | HKII | 28183803 | 1,80E+03 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | HeLa cells | HKII | 28183803 | 1,90E+03 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHK-PASA488 | CHO-K1 cells | HKII | 28183803 | 1,20E+03 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | CHO-K1 cells | HKII | 28183803 | 1,50E+03 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | CHO-K1 cells | HKII | 28183803 | 1,00E+04 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | CHO-K1 cells | HKII | 28183803 | 1,10E+04 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHKA489 | CHO-K1 cells | HKII | 28183803 | 1,70E+02 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | CHO-K1 cells | HKII | 28183803 | 1,90E+02 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA489 | CHO-K1 cells | HKII | 28183803 | 1,10E+03 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | CHO-K1 cells | HKII | 28183803 | 1,30E+03 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHK-PASA488 | pgsA-745 cells | HKII | 28183803 | 1,40E+03 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | pgsA-745 cells | HKII | 28183803 | 1,50E+03 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | pgsA-745 cells | HKII | 28183803 | 1.63 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHK-PASA488 | pgsA-745 cells | HKII | 28183803 | 1,00E+04 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELNGKPILFF-NH2 |
pHKA489 | pgsA-745 cells | HKII | 28183803 | 1,30E+02 | Fluorescence intensity | 5uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | pgsA-745 cells | HKII | 28183803 | 1,50E+02 | Fluorescence intensity | 10uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA489 | pgsA-745 cells | HKII | 28183803 | 1,80E+02 | Fluorescence intensity | 25uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
pHKA490 | pgsA-745 cells | HKII | 28183803 | 1,00E+03 | Fluorescence intensity | 50uM | 2h | 37ºC | FACS | Cellular uptake | A488-MIASHLLAYFFTELN-NH2 |
R16-CD63-GFP | CHO-K1 cells | EVs | 31810935 | 100 | Relative Cellular uptake | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CH3CO-NH-CGRRRRRRRRRRRRRRRR-NH2 |
R16-CD63-GFP | CHO-K1 cells | Evs w/ lyophilization | 31810935 | 100 | Relative Cellular uptake | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CH3CO-NH-CGRRRRRRRRRRRRRRRR-NH2 |
R16-CD63-GFP | CHO cells | EVs | 31810935 | 55 | Relative Cellular uptake | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CH3CO-NH-CGRRRRRRRRRRRRRRRR-NH2 |
R16-CD63-GFP | CHO cells | Evs w/ lyophilization | 31810935 | 49 | Relative Cellular uptake | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CH3CO-NH-CGRRRRRRRRRRRRRRRR-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 1.6 | Cellular retention (mol/cell x 10-16) | 37 kBq | 1h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 1.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 2h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 4.5 | Cellular retention (mol/cell x 10-16) | 37 kBq | 4h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 6.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 6h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 11.24 | Cellular retention (mol/cell x 10-16) | 37 kBq | 12h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
AMO/PF6 | A549 cells | 99mTc | 33480702 | 10.42 | Cellular retention (mol/cell x 10-16) | 37 kBq | 24h | 37ºC | CLSM | Cellular uptake | AMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 1.3 | Cellular retention (mol/cell x 10-16) | 37 kBq | 1h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 1.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 2h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 3.3 | Cellular retention (mol/cell x 10-16) | 37 kBq | 4h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 5.8 | Cellular retention (mol/cell x 10-16) | 37 kBq | 6h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 10.66 | Cellular retention (mol/cell x 10-16) | 37 kBq | 12h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
misAMO/PF6 | A549 cells | 99mTc | 33480702 | 9.2 | Cellular retention (mol/cell x 10-16) | 37 kBq | 24h | 37ºC | CLSM | Cellular uptake | misAMO-Stearoyl-AGYLLGK(-QN)4INLKALAALAKKIL-NH2 |
LDP-NLS | HeLa cells | FITC | 28159722 | 50100 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWRRKLKKLRPKKKRKV |
LDP | HeLa cells | FITC | 28159722 | 8000 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWRRKLKKLR |
NLS | HeLa cells | FITC | 28159722 | 0 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | PKKKRKV |
Mut-LDP-NLS | HeLa cells | FITC | 28159722 | 0 | FITC Mean Intensity | 20 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | AWRRKLKALAPAKKAKV |
cR10 | U2OS cells | FITC | 33615660 | 0 | FITC signal | 6 uM | 15 min | nan | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCG |
cR10DABCYL | U2OS cells | FITC | 33615660 | 0 | FITC signal | 6 uM | 15 min | nan | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCG-DABCYL |
Ub-SScR10 | U2OS cells | TAMPA | 33615660 | 18 | TAMPA intensity | 2 uM | 1h | nan | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCGRRRRRRRRRR |
Ub-SScR10D | U2OS cells | TAMPA | 33615660 | 50 | TAMPA intensity | 12 uM | 1h | nan | CLSM | Cellular uptake | LYRAGLYRAGLYKAGCGRRRRRRRRRR |
Tat-PTD | HDF cells | FITC | 32374475 | 264.6±23.21 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
Tat-PTD | HDF cells | FITC | 32374475 | 209.00±29.67 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
Ara-27 | HDF cells | FITC | 32374475 | 210.33±17.90 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
Ara-27 | HDF cells | FITC | 32374475 | 1800.33±590.46 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
Tat-PTD | hDPSC cells | FITC | 32374475 | 174.67±8.45 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
Tat-PTD | hDPSC cells | FITC | 32374475 | 231.00±42.12 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GRKKRRQRRK |
Ara-27 | hDPSC cells | FITC | 32374475 | 240.00±27.75 | Relative fluorescence | 0.2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
Ara-27 | hDPSC cells | FITC | 32374475 | 4985.67±335.33 | Relative fluorescence | 2uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RNQRKTVRCFRCRQAGHWISDCRLKSK |
MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 0.65 | Relative Mean Fluorescence intensity | nan | 1h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 1.35 | Relative Mean Fluorescence intensity | nan | 3h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
MSN@PLA–PEG-CPP | HT29 cells | FITC | 32697099 | 2.6 | Relative Mean Fluorescence intensity | nan | 6h | 37ºC | CLSM | Cellular uptake | VSRRRRRRGGRRRRC |
CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1100 | Fluorescence intensity | 2.5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KARKKKLNKKGRKMAGRKRGRPKK |
CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1400 | Fluorescence intensity | 5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KARKKKLNKKGRKMAGRKRGRPKK |
CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1450 | Fluorescence intensity | 7.5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KARKKKLNKKGRKMAGRKRGRPKK |
CPP-Dot1l | MCF7 cells | FITC | 32024261 | 1900 | Fluorescence intensity | 10uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KARKKKLNKKGRKMAGRKRGRPKK |
NCO | MCF7 cells | FITC | 32024261 | 200 | Fluorescence intensity | 2.5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KALGISYGRKK |
NCO | MCF7 cells | FITC | 32024261 | 100 | Fluorescence intensity | 5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KALGISYGRKK |
NCO | MCF7 cells | FITC | 32024261 | 300 | Fluorescence intensity | 7.5uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KALGISYGRKK |
NCO | MCF7 cells | FITC | 32024261 | 300 | Fluorescence intensity | 10uM | 1h | nan | Fluorescent Microscopy | Cellular uptake | FITC-(Acp)-KALGISYGRKK |
NLS-A | PK15 cells | FITC | 30108178 | 690 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
NLS-A | HeLa cells | FITC | 30108178 | 580 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
NLS-A | NIH-3T3 cells | FITC | 30108178 | 750 | Fluorescence intensity | 6uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | MTYPRRRFRRRRHRPRS |
TAT0 | HeLa cells | HPMA | 31936737 | 8 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT0 | HeLa cells | HPMA | 31936737 | 7 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT0 | HeLa cells | HPMA | 31936737 | 32 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT0 | HeLa cells | HPMA | 31936737 | 28 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT4 | HeLa cells | HPMA | 31936737 | 7 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT4 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT4 | HeLa cells | HPMA | 31936737 | 50 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT4 | HeLa cells | HPMA | 31936737 | 53 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT12 | HeLa cells | HPMA | 31936737 | 5 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT12 | HeLa cells | HPMA | 31936737 | 22 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT12 | HeLa cells | HPMA | 31936737 | 58 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
TAT12 | HeLa cells | HPMA | 31936737 | 75 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GRKKRRQRRR |
PEN0 | HeLa cells | HPMA | 31936737 | 11 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN0 | HeLa cells | HPMA | 31936737 | 18 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN0 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN0 | HeLa cells | HPMA | 31936737 | 12 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN4 | HeLa cells | HPMA | 31936737 | 8 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN4 | HeLa cells | HPMA | 31936737 | 17 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN4 | HeLa cells | HPMA | 31936737 | 13 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN4 | HeLa cells | HPMA | 31936737 | 13 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN12 | HeLa cells | HPMA | 31936737 | 10 | Relative Median Fluorescence | 1uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN12 | HeLa cells | HPMA | 31936737 | 27 | Relative Median Fluorescence | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN12 | HeLa cells | HPMA | 31936737 | 26 | Relative Median Fluorescence | 25uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
PEN12 | HeLa cells | HPMA | 31936737 | 25 | Relative Median Fluorescence | 50uM | 1h | 4ºC | Flow cytometry | Cellular uptake | RRMKWKK |
d-Pen | C2C12 cells | Streptavidin-Alexa555 | 29045142 | 0 | nan | 50uM | 10min | nan | BCARS Imaging | Cellular uptake | GGGGGGRQIKIWFQNRRMKWKKK-biotinyl-NH2 |
rEETI-II | HeLa cells | Alexa488 | 27734922 | 0 | nan | 20uM | 45min | 37ºC | Fluorescence imaging | Cellular uptake | GSGCPRILMRCKQDSDCLAGCVCGPNGFCGGNS |
R8-Alexa488 | A431 cells | Cyt D | 29743505 | 0 | nan | 2uM | 15 min | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
R8-Alexa488 | HeLa cells | Cyt D | 29743505 | 0 | nan | 2uM | 15 min | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
EGFP-R8 | A431 cells | Lat B | 29743505 | 0 | nan | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
EGFP-R8 | A431 cells | JAS | 29743505 | 0 | nan | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRR-GC |
RFFR | SH-SY5Y cells | TAMPA | 35019611 | 0 | nan | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | TAMRA-RFFR |
RFFR | NIH-3T3 cells | TAMPA | 35019611 | 0 | nan | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | TAMRA-RFFR |
RFFR | HeLa cells | TAMPA | 35019611 | 0 | nan | 100 ug/mL | 30min | 37ºC | CLSM | Cellular uptake | TAMRA-RFFR |
Tat | HeLa cells | Alexa488 | 34152716 | 1 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRRPPQG |
Tat-G | HeLa cells | Alexa488 | 34152716 | 0.2 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGGGKGGQGGGPPQG |
MCNr-2 | HeLa cells | Alexa488 | 34152716 | 0.3 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CPKILKKCRRDSDCPGACICRGNGYCGSGSDEETGEGGV |
MCNr-2c | HeLa cells | Alexa488 | 34152716 | 0.4 | Mean Fluorescence intensity | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CPFWRRRRCKRDSDCPGACICRGNGYCGSGCDEETGECGV |
R2W4R2 | MCF7 cells | FITC | 32116040 | 25 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
R2W4R2 | MCF7 cells | FITC | 32116040 | 72 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
R2W4R2 | MCF7 cells | FITC | 32116040 | 70 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
R2W4R2 | MCF7 cells | FITC | 32116040 | 93 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR |
W3R4W3 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
W3R4W3 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
W3R4W3 | MCF7 cells | FITC | 32116040 | 8 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
W3R4W3 | MCF7 cells | FITC | 32116040 | 12 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW |
R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 10 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 18 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 41 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
R2W4R2-E12 | MCF7 cells | FITC | 32116040 | 45 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWWWWRR-E12 |
W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 3 | Cell fluorescence (%) | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 2 | Cell fluorescence (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 4 | Cell fluorescence (%) | 15uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
W3R4W3-E12 | MCF7 cells | FITC | 32116040 | 23 | Cell fluorescence (%) | 25uM | 1h | 37ºC | Flow cytometry | Cellular uptake | WWWRRRRWWW-E12 |
TP | CHO cells | AgNPs | 33920021 | 300 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | CHO cells | AuNPs | 33920021 | 85 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | CHO cells | IONPs | 33920021 | 38 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | CHO cells | QDs | 33920021 | 135 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | CHO cells | BSA | 33920021 | 270 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | CHO cells | Dextran | 33920021 | 22 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | AgNPs | 33920021 | 400 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | AuNPs | 33920021 | 40 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | IONPs | 33920021 | 29 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | QDs | 33920021 | 190 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | BSA | 33920021 | 210 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | H1975 cells | Dextran | 33920021 | 18 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | AgNPs | 33920021 | 70 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | AuNPs | 33920021 | 15 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | IONPs | 33920021 | 10 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | QDs | 33920021 | 110 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | BSA | 33920021 | 60 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
TP | HeLa cells | Dextran | 33920021 | 19 | Relative Cellular uptake | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | FAM-Ahx-GWTLNSAGYLLGKINLKALAALAKKIL |
sC18 | HEK293 cells | actinomycin D | 27860402 | 70000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
sC18 | HEK293 cells | actinomycin D | 27860402 | 50000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
(sC18)2 | HEK293 cells | actinomycin D | 27860402 | 300000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
(sC18)2 | HEK293 cells | actinomycin D | 27860402 | 600000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
sC18 | MCF7 cells | actinomycin D | 27860402 | 100000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
sC18 | MCF7 cells | actinomycin D | 27860402 | 200000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
(sC18)2 | MCF7 cells | actinomycin D | 27860402 | 1800000 | Relative fluorescence | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
(sC18)2 | MCF7 cells | actinomycin D | 27860402 | 1500000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEKGLRKRLRKFRNKIKEK |
TAT | HeLa cells | FITC | 34101293 | 70 | Cellular uptake (%) | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRR-NH2 |
TAT | HeLa cells | FITC | 34101293 | 100 | Cellular uptake (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | YGRKKRRQRRR-NH2 |
HNLS-3 | HeLa cells | FITC | 34101293 | 20 | Cellular uptake (%) | 10uM | 1h | 4ºC | Flow cytometry | Cellular uptake | PFVYLIPKKKRKVHHHHHHGC-NH2 |
HNLS-3 | HeLa cells | FITC | 34101293 | 100 | Cellular uptake (%) | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | PFVYLIPKKKRKVHHHHHHGC-NH2 |
AF-cGm | HeLa cells | Alexa488 | 32979382 | 0.5 | Relative Cellular uptake | 4uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GCRRLCYK*QRCVTYCRGR |
AF-cGm | HeLa cells | Alexa488 | 32979382 | 2.1 | Relative Cellular uptake | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GCRRLCYK*QRCVTYCRGR |
AF-[R4A,R18A]cGm | HeLa cells | Alexa488 | 32979382 | 0.2 | Relative Cellular uptake | 4uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GCRALCYK*QRCVTYCRGA |
AF-[R4A,R18A]cGm | HeLa cells | Alexa488 | 32979382 | 2.3 | Relative Cellular uptake | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GCRALCYK*QRCVTYCRGA |
AF-[G1K,K8R]cGm | HeLa cells | Alexa488 | 32979382 | 0.5 | Relative Cellular uptake | 4uM | 1h | 4ºC | Flow cytometry | Cellular uptake | K*CRRLCYRQRCVTYCRGR |
AF-[G1K,K8R]cGm | HeLa cells | Alexa488 | 32979382 | 4.5 | Relative Cellular uptake | 4uM | 1h | 37ºC | Flow cytometry | Cellular uptake | K*CRRLCYRQRCVTYCRGR |
Mel-lip | bEnd.3 cells | DiI | 32561686 | 5 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-lip | bEnd.3 cells | DiI | 32561686 | 10 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-lip | bEnd.3 cells | DiI | 32561686 | 20 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-lip | bEnd.3 cells | DiI | 32561686 | 39 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-lip | bEnd.3 cells | DiI | 32561686 | 70 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 5 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 25 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 37 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
Mel-Tf-lip | bEnd.3 cells | DiI | 32561686 | 70 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | GIGAVLKVLTTGLPALISWIKRKRQ |
kFGF-lip | bEnd.3 cells | DiI | 32561686 | 10 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-lip | bEnd.3 cells | DiI | 32561686 | 17 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-lip | bEnd.3 cells | DiI | 32561686 | 39 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-lip | bEnd.3 cells | DiI | 32561686 | 72 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 8 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 18 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 22 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 40 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
kFGF-Tf-lip | bEnd.3 cells | DiI | 32561686 | 72 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | AAVALLPAVLLALLAP |
PasR8-lip | bEnd.3 cells | DiI | 32561686 | 4 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-lip | bEnd.3 cells | DiI | 32561686 | 7 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-lip | bEnd.3 cells | DiI | 32561686 | 30 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-lip | bEnd.3 cells | DiI | 32561686 | 42 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-lip | bEnd.3 cells | DiI | 32561686 | 67 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 4 | Cellular uptake (%) | 100nM | 0.1h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 7 | Cellular uptake (%) | 100nM | 0.25h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 28 | Cellular uptake (%) | 100nM | 0.5h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 40 | Cellular uptake (%) | 100nM | 1h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
PasR8-Tf-lip | bEnd.3 cells | DiI | 32561686 | 73 | Cellular uptake (%) | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | FFLIPKGRRRRRRRRGC |
Agl-AA 1a | MDA-MB-231 cells | fluorescent tag | 28863239 | 50 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXR |
Agl-AA 1b | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXRXRXR |
Agl-AA 1c | MDA-MB-231 cells | fluorescent tag | 28863239 | 60 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XRXRXRXRXRXR |
Agl-AA 2a | MDA-MB-231 cells | fluorescent tag | 28863239 | 50 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXW |
Agl-AA 2b | MDA-MB-231 cells | fluorescent tag | 28863239 | 150 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXWXWXW |
Agl-AA 2c | MDA-MB-231 cells | fluorescent tag | 28863239 | 650 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XWXWXWXWXWXW |
Agl-AA 3a | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXR |
Agl-AA 3b | MDA-MB-231 cells | fluorescent tag | 28863239 | 30 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXRXFXR |
Agl-AA 3c | MDA-MB-231 cells | fluorescent tag | 28863239 | 40 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | XFXRXFXRXFXR |
Agl-AA 4a | MDA-MB-231 cells | fluorescent tag | 28863239 | 100 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | RQIKIWFQNRRMKWKKGG |
Agl-AA 4b | MDA-MB-231 cells | fluorescent tag | 28863239 | 190 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | RRWWRRWRR |
Agl-AA 5a | MDA-MB-231 cells | fluorescent tag | 28863239 | 40 | Cellular uptake | 10uM | 3h | 37ºC | FT-IR | Cellular uptake | AWARAWARAWAR |
BRC4wt | HeLa cells | TAMRA | 29654063 | 30 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | LLGFHTASGKKVKIAK |
R9 | HeLa cells | TAMRA | 29654063 | 5000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR |
R9-BRC4wt | HeLa cells | TAMRA | 29654063 | 4000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGFHTASGKKVKIAK |
R9-BRC4mut | HeLa cells | TAMRA | 29654063 | 2000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGATHFSGKKVKIAK |
BRC4wt | U2OS cells | TAMRA | 29654063 | 50 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | LLGFHTASGKKVKIAK |
R9 | U2OS cells | TAMRA | 29654063 | 10000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR |
R9-BRC4wt | U2OS cells | TAMRA | 29654063 | 4000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGFHTASGKKVKIAK |
R9-BRC4mut | U2OS cells | TAMRA | 29654063 | 10000 | Median TAMRA intensity | 10 umol/L | 1h | nan | Flow cytometry | Cellular uptake | RRRRRRRRR-LLGATHFSGKKVKIAK |
GBPECP | A549 cells | FITC | 27936565 | 0 | nan | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYRWRCKNQN |
GBPEDN | A549 cells | FITC | 27936565 | 0 | nan | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYQRRCKNQN |
GBPECP(W4R) | A549 cells | FITC | 27936565 | 0 | nan | 5 uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | NYRRRCKNQN |
IgG-colpep | HeLa cells | FITC | 26725435 | 20 | Fluorescence intensity | 40 ug /mL | 3h | 37ºC | Flow cytometry | Cellular uptake | GPXGPXGPXGPRGPRGPRGPXGPXGPXGP |
IgG-?R8 | HeLa cells | FITC | 26725435 | 14 | Fluorescence intensity | 40 ug /mL | 3h | 37ºC | Flow cytometry | Cellular uptake | XRRRRRRRR |
PepB2 | CHO-K1 cells | PA | 29247010 | 600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | CROP | 29247010 | 900 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | SLO | 29247010 | 1300 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | CT-B | 29247010 | 600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | Tf | 29247010 | 1500 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | SA | 29247010 | 1600 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | Dextran | 29247010 | 1500 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
PepB2 | CHO-K1 cells | MS | 29247010 | 1000 | Median Fluorescence intensity | 50 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | NVFKGNTISDKISFNFSDK |
IMT-P8 | HeLa cells | KLA | 27189051 | 300000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
IMT-P8 | MDA-MB-231 cells | KLA | 27189051 | 200000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
IMT-P8 | PC3 cells | KLA | 27189051 | 1100000 | Median Fluorescence intensity | 2.5 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
IMT-P8 | HeLa cells | GFP | 27189051 | 25000 | Median Fluorescence intensity | 5 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RRWRRWNRFNRRRCR |
CMR19 | SJSA-1 cells | cR10 | 34977581 | 0 | nan | 5uM | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | FSDMeSSSVPNBBRNCG |
SI-ULK1 micelle | HepG2 cells | Rho | 29787814 | 0 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
Rhodamine micelle | HepG2 cells | Rho | 29787814 | 115 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
SI-ULK1/Rhodamine micelle | HepG2 cells | Rho | 29787814 | 175 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
SI-ULK1 micelle | HepG2 cells | FITC | 29787814 | 85 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
Rhodamine micelle | HepG2 cells | FITC | 29787814 | 10 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
SI-ULK1/Rhodamine micelle | HepG2 cells | FITC | 29787814 | 100 | Relative fluorescence | 5uM | 24h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRR-NH2 |
Cf | HEK293T cells | FITC | 34277705 | 0 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | Cf-RRPPWLRLDIRR-NH2 |
Cf | HEK293T cells | FITC | 34277705 | 5 | Fluorescence intensity | 5uM | 24h | 37ºC | Flow cytometry | Cellular uptake | Cf-RRPPWLRLDIRR-NH2 |
Cf | HEK293T cells | FITC | 34277705 | 2 | Fluorescence intensity | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | Cf-RRPPWLRLDIRR-NH2 |
Dabcyl | HEK293T cells | FITC | 34277705 | 40 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
Dabcyl | HEK293T cells | FITC | 34277705 | 10 | Fluorescence intensity | 5uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
Dabcyl | HEK293T cells | FITC | 34277705 | 120 | Fluorescence intensity | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | RRRPPWLRLDIRRK |
E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | nan | nan | 1h | 37ºC | CLSM | Cellular uptake | MSGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
Tat-E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | nan | nan | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
Tat-A1E28 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | nan | nan | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGRKRLDRNGGGPGVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPVGVPGVGVPGVGVPGFGVPGVGVPGVGVPGFGVPGVGVPGGGVPGGGVPGVGVPGAGVPGVGVPGGGVPGWPC |
Tat-A4V48 | MDA-MB-231 cells | Alexa488 | 31952530 | 0 | nan | nan | 1h | 37ºC | CLSM | Cellular uptake | MSGYGRKKRRQRRRGGGPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPGVGRKRLDRNGVGVPGVGVPGVGVPGVGVPGVGVPGVGVPG |
(KW)4 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
(KW)4 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
(KW)4 | MCF7 cells | FITC | 28933182 | 70 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKW |
(KW)5 | MCF7 cells | FITC | 28933182 | 60 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
(KW)5 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
(KW)5 | MCF7 cells | FITC | 28933182 | 75 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KWKWKWKWKW |
K2W4K2 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
K2W4K2 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
K2W4K2 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKWWWWKK |
K3W4K3 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
K3W4K3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
K3W4K3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KKKWWWWKKK |
W2K4W2 | MCF7 cells | FITC | 28933182 | 35 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
W2K4W2 | MCF7 cells | FITC | 28933182 | 20 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
W2K4W2 | MCF7 cells | FITC | 28933182 | 30 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWKKKKWW |
W3K4W3 | MCF7 cells | FITC | 28933182 | 80 | Cell fluorescence (%) | 10 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
W3K4W3 | MCF7 cells | FITC | 28933182 | 90 | Cell fluorescence (%) | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
W3K4W3 | MCF7 cells | FITC | 28933182 | 85 | Cell fluorescence (%) | 50uM | 2h | 37ºC | Flow cytometry | Cellular uptake | WWWKKKKWWW |
CPP-siRNA | HT1080 cells | siRNA | 27012462 | 120 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
CPP-siRNA/N-NB | HT1080 cells | siRNA | 27012462 | 30 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
CPP-siRNA/N-NB(+US) | HT1080 cells | siRNA | 27012462 | 110 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
CPP-DOX | MCF7 cells | Doxorubicin | 26176270 | 83 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX | HT1080 cells | Doxorubicin | 26176270 | 80 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX/N-NB | MCF7 cells | Doxorubicin | 26176270 | 22 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX/N-NB | HT1080 cells | Doxorubicin | 26176270 | 20 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX/NGR-NB | MCF7 cells | Doxorubicin | 26176270 | 22 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
CPP-DOX/NGR-NB | HT1080 cells | Doxorubicin | 26176270 | 40 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
CPP-DOX/N-NB (+US) | MCF7 cells | Doxorubicin | 26176270 | 82 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX/N-NB (+US) | HT1080 cells | Doxorubicin | 26176270 | 85 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX |
CPP-DOX/NGR-NB (+US) | MCF7 cells | Doxorubicin | 26176270 | 80 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
CPP-DOX/NGR-NB (+US) | HT1080 cells | Doxorubicin | 26176270 | 82 | Mean Fluorescence intensity | nan | 24h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-DOX/CYGGRGNG |
ENCP | Caco-2 cells | Insulin | 29518466 | 50 | Cellular uptake (%) | nan | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
NCP | Caco-2 cells | Insulin | 29518466 | 80 | Cellular uptake (%) | nan | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
Insulin+R8 | Caco-2 cells | Insulin | 29518466 | 0 | Cellular uptake (%) | nan | 2h | 37ºC | Liquid chromatography | Cellular uptake | RRRRRRRR |
TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 160 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 200 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
?-CT 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 170 | Internalization | 5uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
?-CT 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 180 | Internalization | 10uM | 2h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 110 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
TAT | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 100 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | GRKKRRQRRRPQ |
?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 165 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
?-CC 15 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 250 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPP |
?-CT 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 160 | Internalization | 5uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
?-CT 16 | Leishmania donovani promastigotes | Doxorubicin | 33053805 | 210 | Internalization | 10uM | 4h | 26ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPPPPPPP |
[RW]3 | A549 cells | FITC | 28694765 | 32 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
[RW]3 | A549 cells | FITC | 28694765 | 63 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
[RW]3 | A549 cells | FITC | 28694765 | 90 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRW |
[RW]4 | A549 cells | FITC | 28694765 | 57 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
[RW]4 | A549 cells | FITC | 28694765 | 79 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
[RW]4 | A549 cells | FITC | 28694765 | 80 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRW |
[RW]5 | A549 cells | FITC | 28694765 | 35 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
[RW]5 | A549 cells | FITC | 28694765 | 49 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
[RW]5 | A549 cells | FITC | 28694765 | 68 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRW |
[RW]6 | A549 cells | FITC | 28694765 | 60 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
[RW]6 | A549 cells | FITC | 28694765 | 71 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
[RW]6 | A549 cells | FITC | 28694765 | 79 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
R5W3R4 | A549 cells | FITC | 28694765 | 47 | Cell fluorescence (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
R5W3R4 | A549 cells | FITC | 28694765 | 59 | Cell fluorescence (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
R5W3R4 | A549 cells | FITC | 28694765 | 88 | Cell fluorescence (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 30min | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 1h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 4h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 8h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)1 | COS-1 cells | QDs | 28703833 | 1,00E+05 | Fluorescence intensity | 100 nM | 24h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)2 | COS-1 cells | QDs | 28703833 | 5,00E+04 | Fluorescence intensity | 100 nM | 30min | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGPPPPPPPPPGRRRRRRRRRFGPPPPPPPPPGWGHHHHHH |
QD-(Arg9)2 | COS-1 cells | QDs | 28703833 | 1,50E+05 | Fluorescence intensity | 100 nM | 1h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGPPPPPPPPPGRRRRRRRRRFGPPPPPPPPPGWGHHHHHH |
QD-(Arg9)2 | COS-1 cells | QDs | 28703833 | 1,00E+05 | Fluorescence intensity | 100 nM | 4h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGPPPPPPPPPGRRRRRRRRRFGPPPPPPPPPGWGHHHHHH |
QD-(Arg9)2 | COS-1 cells | QDs | 28703833 | 5,00E+05 | Fluorescence intensity | 100 nM | 8h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGPPPPPPPPPGRRRRRRRRRFGPPPPPPPPPGWGHHHHHH |
QD-(Arg9)2 | COS-1 cells | QDs | 28703833 | 3,80E+05 | Fluorescence intensity | 100 nM | 24h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGPPPPPPPPPGRRRRRRRRRFGPPPPPPPPPGWGHHHHHH |
QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 0 | Fluorescence intensity | 100 nM | 30min | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 8,00E+04 | Fluorescence intensity | 100 nM | 1h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 1,00E+05 | Fluorescence intensity | 100 nM | 4h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 2,30E+05 | Fluorescence intensity | 100 nM | 8h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)4 | COS-1 cells | QDs | 28703833 | 1,30E+05 | Fluorescence intensity | 100 nM | 24h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)8 | COS-1 cells | QDs | 28703833 | 1,00E+04 | Fluorescence intensity | 100 nM | 30min | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)8 | COS-1 cells | QDs | 28703833 | 2,20E+05 | Fluorescence intensity | 100 nM | 1h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)8 | COS-1 cells | QDs | 28703833 | 6,80E+05 | Fluorescence intensity | 100 nM | 4h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)8 | COS-1 cells | QDs | 28703833 | 3,50E+05 | Fluorescence intensity | 100 nM | 8h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)8 | COS-1 cells | QDs | 28703833 | 2,00E+05 | Fluorescence intensity | 100 nM | 24h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)16 | COS-1 cells | QDs | 28703833 | 1,00E+05 | Fluorescence intensity | 100 nM | 30min | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)16 | COS-1 cells | QDs | 28703833 | 1,90E+05 | Fluorescence intensity | 100 nM | 1h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)16 | COS-1 cells | QDs | 28703833 | 4,40E+05 | Fluorescence intensity | 100 nM | 4h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)16 | COS-1 cells | QDs | 28703833 | 1,80E+05 | Fluorescence intensity | 100 nM | 8h | nan | Fluorescent Microscopy | Cellular uptake | RRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGRRRRRRRRRFGWPPPPPPPPPGGHHHHHH |
QD-(Arg9)16 | COS-1 cells | QDs | 28703833 | 9,50E+05 | Fluorescence intensity | 100 nM | 24h | nan | Fluorescent Microscopy | Cellular uptake | REDVYGRKKRRQRRRPKKKRKV |
REDV-TAT-NLS-H0 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 23 | Cellular uptake (%) | nan | 4h | nan | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHH |
REDV-TAT-NLS-H4 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 30 | Cellular uptake (%) | nan | 4h | nan | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHHHHHH |
REDV-TAT-NLS-H8 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 40 | Cellular uptake (%) | nan | 4h | nan | Flow cytometry | Cellular uptake | REDVYGRKKRRQRRRPKKKRKVHHHHHHHHHHHH |
REDV-TAT-NLS-H12 | HUVEC cells | Cy5-oligonucleotide | 29580233 | 88 | Cellular uptake (%) | nan | 4h | nan | Flow cytometry | Cellular uptake | REDV-YGRKKRRQRRR-PKK-KRKV-HHHHHHHHHHHH |
CVP1-N2 | HCT116 cells | FITC | 33141296 | 10 | Relative internalization (%) | 0.1uM | nan | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
CVP1-N2 | HCT116 cells | FITC | 33141296 | 75 | Relative internalization (%) | 1uM | nan | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
CVP1-N2 | HCT116 cells | FITC | 33141296 | 100 | Relative internalization (%) | 10uM | nan | 37ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
CVP1-N2 | HCT116 cells | FITC | 33141296 | 88 | Relative internalization (%) | 10uM | nan | 4ºC | Flow cytometry | Cellular uptake | LKRLRRRYKFRHRRRQRYRRR |
Scp01-b | Caski cells | FITC | 30230543 | 350 | Fluorescence intensity | 2.5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Scp01-b | Caski cells | FITC | 30230543 | 1100 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Scp01-b | Caski cells | FITC | 30230543 | 1350 | Fluorescence intensity | 7.5uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Scp01-b | Caski cells | FITC | 30230543 | 1400 | Fluorescence intensity | 10uM | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
R4-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 1361 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRR |
R8-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 2890 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRR |
R12-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 2862 | Relative Cellular uptake | 20uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRRRRRR |
R16-EMCS | CHO-K1 cells | CD63-GFP Evs | 28512335 | 1823 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GRRRRRRRRRRRRRRRR |
cyc-hCT(9-32) | MCF7 cells | Carboxyfluorescein | 27197760 | 15000 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | CF-Cys-BLGTYTQDFNXFHTFPQTAIGVGAP |
cyc-hCT(9-32) | MCF7 cells | Carboxyfluorescein | 27197760 | 52000 | Relative fluorescence | 50uM | 30min | 37ºC | Flow cytometry | Cellular uptake | CF-Cys-BLGTYTQDFNXFHTFPQTAIGVGAP |
iCREKA | U87 cells | FITC | 29686590 | 14110 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CREKAPLGLAGRKKRRQRRRC |
CREKA | U87 cells | FITC | 29686590 | 2569.5 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | CREKA |
ALD5MTS (2–17) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17)-sC18 | HeLa cells | TAM | 30367921 | 0.65 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
ALD5MTS (2–17)-sC18 | HeLa cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14)-sC18 | HeLa cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14)-sC18 | HeLa cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7) | HeLa cells | TAM | 30367921 | 0.05 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7) | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7)-sC18 | HeLa cells | TAM | 30367921 | 0.75 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7)-sC18 | HeLa cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | HeLa cells | TAM | 30367921 | 0.4 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | HeLa cells | TAM | 30367921 | 0.15 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
sC18 | HeLa cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
sC18 | HeLa cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
ALD5MTS (2–17) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17)-sC18 | MCF7 cells | TAM | 30367921 | 0.35 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
ALD5MTS (2–17)-sC18 | MCF7 cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14) | MCF7 cells | TAM | 30367921 | 0.02 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14) | MCF7 cells | TAM | 30367921 | 0.01 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14)-sC18 | MCF7 cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14)-sC18 | MCF7 cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7) | MCF7 cells | TAM | 30367921 | 0.04 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7) | MCF7 cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7)-sC18 | MCF7 cells | TAM | 30367921 | 0.8 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7)-sC18 | MCF7 cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | MCF7 cells | TAM | 30367921 | 0.15 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | MCF7 cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
sC18 | MCF7 cells | TAM | 30367921 | 0.1 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
sC18 | MCF7 cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
ALD5MTS (2–17) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTR |
ALD5MTS (2–17)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
ALD5MTS (2–17)-sC18 | TDA cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLR |
HSP60MTS (2–14)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
HSP60MTS (2–14)-sC18 | TDA cells | TAM | 30367921 | 0.1 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7) | TDA cells | TAM | 30367921 | 0.01 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7) | TDA cells | TAM | 30367921 | 0 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIR |
BNA3MTS (2–7)-sC18 | TDA cells | TAM | 30367921 | 0.3 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
BNA3MTS (2–7)-sC18 | TDA cells | TAM | 30367921 | 0.08 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KQRFIRGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | TDA cells | TAM | 30367921 | 0.25 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
CalpMTS (2–19)-sC18 | TDA cells | TAM | 30367921 | 0.2 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
sC18 | TDA cells | TAM | 30367921 | 0.15 | Internalization | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
sC18 | TDA cells | TAM | 30367921 | 0.05 | Internalization | 1uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRKFRNKIKEK |
MTX-SCPP-PS | A549 cells | FITC | 29280317 | 0 | nan | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | RLWMRWYSPRTRAYGC |
TI | MDA-MB-435S cells | Alexa488 | 31714739 | 6000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
[Y8SI11S]cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 5000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
[F4S-Y13S]cTI | MDA-MB-435S cells | Alexa488 | 31714739 | 500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
TI | MM96L cells | Alexa488 | 31714739 | 5500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
cTI | MM96L cells | Alexa488 | 31714739 | 2500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
[Y8SI11S]cTI | MM96L cells | Alexa488 | 31714739 | 4500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
[F4S-Y13S]cTI | MM96L cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
TI | HeLa cells | Alexa488 | 31714739 | 3000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
cTI | HeLa cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
[Y8SI11S]cTI | HeLa cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
[F4S-Y13S]cTI | HeLa cells | Alexa488 | 31714739 | 500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
TI | HaCaT cells | Alexa488 | 31714739 | 2500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCR |
cTI | HaCaT cells | Alexa488 | 31714739 | 1500 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCYRGICYRRCRG |
[Y8SI11S]cTI | HaCaT cells | Alexa488 | 31714739 | 2000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCFRVCSRGSCYRRCRG |
[F4S-Y13S]cTI | HaCaT cells | Alexa488 | 31714739 | 1000 | Fluorescence intensity | 2uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KWCSRVCYRGICSRRCRG |
SynB1–ELP1–dnMAML | D54 cells | Fluorescein | 28140690 | 9 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP1–dnMAML | D54 cells | Fluorescein | 28140690 | 37 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP2–dnMAML | D54 cells | Fluorescein | 28140690 | 5 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP2–dnMAML | D54 cells | Fluorescein | 28140690 | 8 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP1–dnMAML | U251 cells | Fluorescein | 28140690 | 8 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP1–dnMAML | U251 cells | Fluorescein | 28140690 | 24 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP2–dnMAML | U251 cells | Fluorescein | 28140690 | 7 | Relative fluorescence | 30 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
SynB1–ELP2–dnMAML | U251 cells | Fluorescein | 28140690 | 10 | Relative fluorescence | 30 uM | 1h | 42ºC | Flow cytometry | Cellular uptake | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
KT2 | HCT116 cells | FITC | 31073999 | 100 | Mean Fluorescence intensity | 1.25uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
KT2 | HCT116 cells | FITC | 31073999 | 200 | Mean Fluorescence intensity | 2.5uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
KT2 | HCT116 cells | FITC | 31073999 | 500 | Mean Fluorescence intensity | 5uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
KT2 | HCT116 cells | FITC | 31073999 | 800 | Mean Fluorescence intensity | 10uM | 4h | 37ºC | Flow cytometry | Cellular uptake | NGVQPKYKWWKWWKKWW-NH2 |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 100 | Mean Fluorescence intensity | 9.0 uM | 30min | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 300 | Mean Fluorescence intensity | 9.0 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 1000 | Mean Fluorescence intensity | 9.0 uM | 2h | 37ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 50 | Mean Fluorescence intensity | 9.0 uM | 30min | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 50 | Mean Fluorescence intensity | 9.0 uM | 1h | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
palmitoyl-cyclic-(D-Arg)12 | HeLa cells | FITC | 29530390 | 200 | Mean Fluorescence intensity | 9.0 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | C37H66N7O17P3S-rrrrrrrrrrrr |
P-(dNP2)-DOX | HeLa cells | Doxorubicin | 30205127 | 2.5 | Fluorescence intensity | 10 ug/ml | 2h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
P-(dNP2)-DOX | HeLa cells | Doxorubicin | 30205127 | 3.5 | Fluorescence intensity | 10 ug/ml | 4h | 37ºC | Flow cytometry | Cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
hybrid ?,?-peptide 9 | HeLa cells | Carboxyfluorescein | 34065025 | 4 | % Fluorescence | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPP |
hybrid ?,?-peptide 9 | HeLa cells | Carboxyfluorescein | 34065025 | 2 | % Fluorescence | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPP |
hybrid ?,?-peptide 10 | HeLa cells | Carboxyfluorescein | 34065025 | 4.5 | % Fluorescence | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPPP |
hybrid ?,?-peptide 10 | HeLa cells | Carboxyfluorescein | 34065025 | 2.5 | % Fluorescence | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPPP |
hybrid ?,?-peptide 11 | HeLa cells | Carboxyfluorescein | 34065025 | 5 | % Fluorescence | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPP |
hybrid ?,?-peptide 11 | HeLa cells | Carboxyfluorescein | 34065025 | 3 | % Fluorescence | 25uM | 2h | 37ºC | Flow cytometry | Cellular uptake | PPPPPPPPPPP |
KD3 | MCF7 cells | Alexa488 | 33533253 | 5 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
cTAT | MCF7 cells | Alexa488 | 33533253 | 10 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
cR10 | MCF7 cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
cTAT-KD3 | MCF7 cells | Alexa488 | 33533253 | 25 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
cR10-KD3 | MCF7 cells | Alexa488 | 33533253 | 45 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
KD3 | HeLa cells | Alexa488 | 33533253 | 3 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
cTAT | HeLa cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
cR10 | HeLa cells | Alexa488 | 33533253 | 18 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
cTAT-KD3 | HeLa cells | Alexa488 | 33533253 | 18 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
cR10-KD3 | HeLa cells | Alexa488 | 33533253 | 20 | Relative Cellular uptake | 2 uM | 1h | 37ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
KD3 | MCF7 cells | Alexa488 | 33533253 | 0 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
cTAT | MCF7 cells | Alexa488 | 33533253 | 1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
cR10 | MCF7 cells | Alexa488 | 33533253 | 15 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
cTAT-KD3 | MCF7 cells | Alexa488 | 33533253 | 0 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrDLTFKEYWDQLTSAA |
cR10-KD3 | MCF7 cells | Alexa488 | 33533253 | 1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRELTFKEYWDQLTSAA |
KD3 | HeLa cells | Alexa488 | 33533253 | 0.2 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | LTFKEYWDQLTSAA |
cTAT | HeLa cells | Alexa488 | 33533253 | 1.3 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD |
cR10 | HeLa cells | Alexa488 | 33533253 | 3 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE |
cTAT-KD3 | HeLa cells | Alexa488 | 33533253 | 0.8 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrGgKkRrD-LTFKEYWDQLTSAA |
cR10-KD3 | HeLa cells | Alexa488 | 33533253 | 2.1 | Relative Cellular uptake | 2 uM | 2h | 4ºC | Flow cytometry | Cellular uptake | KrRrRrRrRrRE-LTFKEYWDQLTSAA |
N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 15000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 7000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
N50-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 1000 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 13000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 10000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
NrTP-sC18* | HeLa cells | Carboxyfluorescein | 29977402 | 2900 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 17000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 13000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
N50-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 16000 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | VQRKRQKLMPGLRKRLRKFRNK |
NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 21000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 7000 | Fluorescence intensity | 10uM | 120min | 37ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
NrTP-sC18* | MCF7 cells | Carboxyfluorescein | 29977402 | 7500 | Fluorescence intensity | 10uM | 30min | 4ºC | Flow cytometry | Cellular uptake | YKQCHKKGGKKGSGGLRKRLRKFRNK |
Conjugate 1a | U87 cells | Carboxyfluorescein | 31243977 | 0.4 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 1a | HT29 cells | Carboxyfluorescein | 31243977 | 0.38 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 1a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.3 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | U87 cells | Carboxyfluorescein | 31243977 | 1 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | HT29 cells | Carboxyfluorescein | 31243977 | 0.37 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.35 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 1a | U87 cells | Carboxyfluorescein | 31243977 | 0.8 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 1a | HT29 cells | Carboxyfluorescein | 31243977 | 0.75 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 1a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.4 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | c[DKP-RGD]-PEG4-GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | U87 cells | Carboxyfluorescein | 31243977 | 1.2 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | HT29 cells | Carboxyfluorescein | 31243977 | 0.43 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
Conjugate 2a | MCF7 cells | Carboxyfluorescein | 31243977 | 0.6 | Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GLRKRLRK(CF)FRNKIKEK-CONH2 |
R8-Lip | C6 cells | CFPE | 26877777 | 40 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
R8-RGD-Lip | C6 cells | CFPE | 26877777 | 60 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
R8-EGR-Lip | C6 cells | CFPE | 26877777 | 80 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
R8-dGR-Lip | C6 cells | CFPE | 26877777 | 90 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
R8-Lip | bEnd.3 cells | CFPE | 26877777 | 10 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
R8-RGD-Lip | bEnd.3 cells | CFPE | 26877777 | 20 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
R8-EGR-Lip | bEnd.3 cells | CFPE | 26877777 | 18 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
R8-dGR-Lip | bEnd.3 cells | CFPE | 26877777 | 25 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
R8-Lip | HeLa cells | CFPE | 26877777 | 6 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRR-Lip |
R8-RGD-Lip | HeLa cells | CFPE | 26877777 | 7 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-RGD-Lip |
R8-EGR-Lip | HeLa cells | CFPE | 26877777 | 8 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-EGR-Lip |
R8-dGR-Lip | HeLa cells | CFPE | 26877777 | 9 | Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | Cys-RRRRRRRR-dGR-Lip |
HL6 | A549 cells | FITC | 31253836 | 0 | nan | nan | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | CHHHHHRRWQWRHHHHHC |
hPep1 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 25nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
hPep2 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 25nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
hPep3 | HeLa cells | AF568-SSO | 34440250 | 300 | Relative fluorescence | 25nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
hPep1 | HeLa cells | AF568-SSO | 34440250 | 100 | Relative fluorescence | 50nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
hPep2 | HeLa cells | AF568-SSO | 34440250 | 300 | Relative fluorescence | 50nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
hPep3 | HeLa cells | AF568-SSO | 34440250 | 1000 | Relative fluorescence | 50nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
hPep1 | HeLa cells | AF568-SSO | 34440250 | 1000 | Relative fluorescence | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
hPep2 | HeLa cells | AF568-SSO | 34440250 | 1500 | Relative fluorescence | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
hPep3 | HeLa cells | AF568-SSO | 34440250 | 2500 | Relative fluorescence | 100nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
hPep1 | HeLa cells | AF568-SSO | 34440250 | 5500 | Relative fluorescence | 200nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S5)AKAL-NH2 |
hPep2 | HeLa cells | AF568-SSO | 34440250 | 6000 | Relative fluorescence | 200nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-LAKLAKA(R8)AKLLKA(S8)AKAL-NH2 |
hPep3 | HeLa cells | AF568-SSO | 34440250 | 7000 | Relative fluorescence | 200nM | 4h | nan | Fluorescence spectroscopy | Cellular uptake | H-L(R8)KLAKA(R8)AKLLKA(R8)AKAL-NH2 |
VaspinN | HEK293 cells | TAMRA | 33866927 | 150 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | LKPSFSPRNY |
VaspinHA1 | HEK293 cells | TAMRA | 33866927 | 80 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KALSEVQGWKQRMAAKELAR |
VaspinHA2 | HEK293 cells | TAMRA | 33866927 | 150 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KQRMAAKELAR |
VaspinN | NIH-3T3 cells | TAMRA | 33866927 | 2500 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | LKPSFSPRNY |
VaspinHA1 | NIH-3T3 cells | TAMRA | 33866927 | 2000 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KALSEVQGWKQRMAAKELAR |
VaspinHA2 | NIH-3T3 cells | TAMRA | 33866927 | 2000 | Relative fluorescence | 10uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | KQRMAAKELAR |
NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 70 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 50 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 60 | Fluorescence intensity | 0.002ug/mL | 30min | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 210 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 160 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 120 | Fluorescence intensity | 0.002ug/mL | 2h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 250 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 230 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 200 | Fluorescence intensity | 0.002ug/mL | 4h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
NLC-RGE | MDA-MB-231 cells | Cou-6 | 29528244 | 342.34 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | RGERPPR |
NLC-cRGD | MDA-MB-231 cells | Cou-6 | 29528244 | 254.4 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | CRGDRGPDC |
NLC-RGE/cRG | MDA-MB-231 cells | Cou-6 | 29528244 | 245.8 | Fluorescence intensity | 0.002ug/mL | 12h | 37ºC | Flow cytometry | Cellular uptake | RGERPPRCRGDRGPDC |
CPP–siRNA/N-NB | MCF7 cells | siRNA | 26492155 | 30 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
CPP–siRNA/YSA-NB | MCF7 cells | siRNA | 26492155 | 40 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-YSAYPDSVPMMS |
CPP-siRNA/N-NB (+US) | MCF7 cells | siRNA | 26492155 | 110 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK |
CPP–siRNA/YSA-NB (+US) | MCF7 cells | siRNA | 26492155 | 130 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | Cellular uptake | CKRRMKWKK-YSAYPDSVPMMS |
I-LCP | HCT116 cells | Radiolabelled Iodine (125I) | 31445852 | 10 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAANVGrrrrrrrrrXk([125I]IB)-NH2 |
I-NCP | HCT116 cells | Radiolabelled Iodine (125I) | 31445852 | 2 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAACtVGrrrrrrrrrXk([125I]IB)-NH2 |
LPC | HCT116 cells | FL | 31445852 | 5 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAANVGrrrrrrrrrXk(FL)-NH2 |
NCP | HCT116 cells | FL | 31445852 | 7 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-eeeeeeeeeXPAACtVGrrrrrrrrrXk(FL)-NH2 |
LCP-r | HCT116 cells | FL | 31445852 | 31 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-XPAANVGrrrrrrrrrXk(FL)-NH2 |
NCP-r | HCT116 cells | FL | 31445852 | 33 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | Cellular uptake | Ac-XPAACtVGrrrrrrrrrXk(FL)-NH2 |
R9 | A549 cells | FITC | 27074859 | 65 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
R5W3R4 | A549 cells | FITC | 27074859 | 70 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
[RW]6 | A549 cells | FITC | 27074859 | 72 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
R9 | A549 cells | FITC | 27074859 | 73 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
R5W3R4 | A549 cells | FITC | 27074859 | 80 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
[RW]6 | A549 cells | FITC | 27074859 | 79 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
R9 | A549 cells | FITC | 27074859 | 88 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR |
R5W3R4 | A549 cells | FITC | 27074859 | 95 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR |
[RW]6 | A549 cells | FITC | 27074859 | 85 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW |
R9/E9 | A549 cells | FITC | 27074859 | 52 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
R5W3R4/E9 | A549 cells | FITC | 27074859 | 55 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
[RW]6/E9 | A549 cells | FITC | 27074859 | 56 | Relative fraction of positive cells (%) | 10uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
R9/E9 | A549 cells | FITC | 27074859 | 72 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
R5W3R4/E9 | A549 cells | FITC | 27074859 | 75 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
[RW]6/E9 | A549 cells | FITC | 27074859 | 78 | Relative fraction of positive cells (%) | 25uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
R9/E9 | A549 cells | FITC | 27074859 | 82 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRRRRR-EEEEEEEEE |
R5W3R4/E9 | A549 cells | FITC | 27074859 | 85 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RRRRRWWWRRRR-EEEEEEEEE |
[RW]6/E9 | A549 cells | FITC | 27074859 | 86 | Relative fraction of positive cells (%) | 50uM | 1.5h | 37ºC | Flow cytometry | Cellular uptake | RWRWRWRWRWRW-EEEEEEEEE |
Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 200000 | Fluorescence intensity | 2.5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 800000 | Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
Dabcyl–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 1050000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | Dabcyl-RRRRRRK-Rho-NH2 |
H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 0 | Fluorescence intensity | 2.5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 5000 | Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
H–Arg6–Lys(Rh)–NH2 | HeLa cells | Carboxyfluorescein | 34032919 | 5000 | Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | H-RRRRRRK-Rho-NH2 |
biotinyl-GM3BP | HeLa cells | GFP | 28051846 | 8 | Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | Cellular uptake | GWWYKGRARPVSAVAK(biotin)-NH2 |
biotinyl-GM3BP | HeLa cells | GFP | 28051846 | 1 | Fluorescence intensity | 5uM | 1h | 4ºC | Flow cytometry | Cellular uptake | GWWYKGRARPVSAVAK(biotin)-NH2 |
biotinyl-TAT | HeLa cells | GFP | 28051846 | 0 | nan | nan | nan | nan | Flow cytometry | Cellular uptake | YGRKKRRQRRRK(biotin)-NH2 |
biotinyl-CP8 | HeLa cells | GFP | 28051846 | 0 | nan | nan | nan | nan | Flow cytometry | Cellular uptake | AETVESCLAKPHTENK- (biotin)-NH2 |
GGL27 | A375 cells | TAMRA | 31672541 | 25 | Corrected total cell fluorescence | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
GGL27 | A375 cells | TAMRA | 31672541 | 8 | Corrected total cell fluorescence | 5uM | 2h | 4ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
GGL27 | HeLa cells | TAMRA | 31672541 | 35 | Corrected total cell fluorescence | 5uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
GGL27 | HeLa cells | TAMRA | 31672541 | 18 | Corrected total cell fluorescence | 5uM | 2h | 4ºC | Flow cytometry | Cellular uptake | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
GA-TAT | EJ cells | nan | 29670331 | 1 | Cellular uptake | 0.25uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | EJ cells | nan | 29670331 | 2 | Cellular uptake | 1uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | EJ cells | nan | 29670331 | 5 | Cellular uptake | 2.5uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | EJ cells | nan | 29670331 | 6 | Cellular uptake | 5uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | SV-HUC-1 cells | nan | 29670331 | 1 | Cellular uptake | 0.25uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | SV-HUC-1 cells | nan | 29670331 | 2 | Cellular uptake | 1uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | SV-HUC-1 cells | nan | 29670331 | 5 | Cellular uptake | 2.5uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
GA-TAT | SV-HUC-1 cells | nan | 29670331 | 7 | Cellular uptake | 5uM | 2h | nan | Flow cytometry | Cellular uptake | GA-YGRKKRRQRRR |
SNEDDS F-1 | Caco-2 cells | sodium fluorescein | 27458781 | 1.5 | Cellular uptake (%) | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-pDNA |
SNEDDS F-1 | Caco-2 cells | sodium fluorescein | 27458781 | 2 | Cellular uptake (%) | nan | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-pDNA |
SNEDDS F-2 | Caco-2 cells | sodium fluorescein | 27458781 | 3 | Cellular uptake (%) | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-OL-Pdna |
SNEDDS F-2 | Caco-2 cells | sodium fluorescein | 27458781 | 5 | Cellular uptake (%) | nan | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RKKRRQRRR-OL-Pdna |
L1 | HeLa cells | Carboxyfluorescein | 27966361 | 14 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-MIILIIGSTSRDHMVLHEYVNAAGIT-NH2 |
L2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-FLLIRRVLGSTSRDHMVLHEYVNAAGIT-NH2 |
L3 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-PWPRVPWRWGSTSRDHMVLHEYVNAAGIT-NH2 |
L4 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-LKRAIWLIKGSTSRDHMVLHEYVNAAGIT-NH2 |
C1 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-FIDLKRKIWLIK-NH2 |
C2 | HeLa cells | Carboxyfluorescein | 27966361 | 5 | Normalized Mean Fluorescence intensity | 5uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-YLKFIPLKDAIWKIK-NH2 |
L1 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-MIILIIGSTSRDHMVLHEYVNAAGIT-NH2 |
L2 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-FLLIRRVLGSTSRDHMVLHEYVNAAGIT-NH2 |
L3 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-PWPRVPWRWGSTSRDHMVLHEYVNAAGIT-NH2 |
L4 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-LKRAIWLIKGSTSRDHMVLHEYVNAAGIT-NH2 |
C1 | HeLa cells | Carboxyfluorescein | 27966361 | 6 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-FIDLKRKIWLIK-NH2 |
C2 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 2uM | 30 min | nan | Flow cytometry | Cellular uptake | Fluo-YLKFIPLKDAIWKIK-NH2 |
L1 | HeLa cells | Carboxyfluorescein | 27966361 | 13 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-MIILIIGSTSRDHMVLHEYVNAAGIT-NH2 |
L2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-FLLIRRVLGSTSRDHMVLHEYVNAAGIT-NH2 |
L3 | HeLa cells | Carboxyfluorescein | 27966361 | 7 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-PWPRVPWRWGSTSRDHMVLHEYVNAAGIT-NH2 |
L4 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-LKRAIWLIKGSTSRDHMVLHEYVNAAGIT-NH2 |
C1 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-FIDLKRKIWLIK-NH2 |
C2 | HeLa cells | Carboxyfluorescein | 27966361 | 1 | Normalized Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-YLKFIPLKDAIWKIK-NH2 |
L1-1 | HeLa cells | Carboxyfluorescein | 27966361 | 3 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-KIIIIDGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
L1-2 | HeLa cells | Carboxyfluorescein | 27966361 | 4 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-K(Nle)IILIIDGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
L1-3 | HeLa cells | Carboxyfluorescein | 27966361 | 16 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-(Nle)IILIIGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
L1-4 | HeLa cells | Carboxyfluorescein | 27966361 | 5 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-MLILIIGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
L1-5 | HeLa cells | Carboxyfluorescein | 27966361 | 9 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-MIILIIMGVADLIKKFESISKEE-NH2 |
L1-6 | HeLa cells | Carboxyfluorescein | 27966361 | 15 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-PLILLRLLRGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
L1-7 | HeLa cells | Carboxyfluorescein | 27966361 | 35 | Median Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Cellular uptake | Fluo-FIDIIIKILLIGSTSRDH(Nle)VLHEYVNAAGIT-Ado-NH2 |
R8HNPs | R1 ESC cells | nan | 33464088 | 59 | Relative fluorescence | 25 ug/mL | 30 min | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | 43 | Relative fluorescence | 25 ug/mL | 1h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | 38 | Relative fluorescence | 25 ug/mL | 3h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | 27 | Relative fluorescence | 25 ug/mL | 6h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | 20 | Relative fluorescence | 25 ug/mL | 12h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | 19 | Relative fluorescence | 25 ug/mL | 24h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
R8HNPs | R1 ESC cells | nan | 33464088 | -20 | Relative fluorescence | 25 ug/mL | 48h | nan | CLSM | Cellular uptake | RRRRRRRR-H-NPs-siScr |
SialoPen 6 | HeLa cells | Cy5 | 33409387 | 8,00E+03 | Mean Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)6-Ahx-NH2 |
SialoPen 7 | HeLa cells | Cy5 | 33409387 | 9,00E+03 | Mean Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)7-Ahx-NH2 |
SialoPen 8 | HeLa cells | Cy5 | 33409387 | 1,20E+04 | Mean Fluorescence intensity | 1uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)8-Ahx-NH2 |
SialoPen 6 | HeLa cells | Cy5 | 33409387 | 1,70E+04 | Mean Fluorescence intensity | 2.5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)6-Ahx-NH2 |
SialoPen 7 | HeLa cells | Cy5 | 33409387 | 2,00E+04 | Mean Fluorescence intensity | 2.5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)7-Ahx-NH2 |
SialoPen 8 | HeLa cells | Cy5 | 33409387 | 2,50E+04 | Mean Fluorescence intensity | 2.5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)8-Ahx-NH2 |
SialoPen 6 | HeLa cells | Cy5 | 33409387 | 3,50E+04 | Mean Fluorescence intensity | 5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)6-Ahx-NH2 |
SialoPen 7 | HeLa cells | Cy5 | 33409387 | 4,00E+04 | Mean Fluorescence intensity | 5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)7-Ahx-NH2 |
SialoPen 8 | HeLa cells | Cy5 | 33409387 | 4,40E+04 | Mean Fluorescence intensity | 5uM | 30 min | 37ºC | Flow cytometry | Cellular uptake | Cy5-(Neu2en-R)8-Ahx-NH2 |
SR11 | HeLa cells | FITC | 26752214 | 20 | Mean Fluorescence intensity | 20 ug/ml | 30min | nan | Flow cytometry | Cellular uptake | NH2-SGASDDEEIAR-COOH |
SR11 | HeLa cells | FITC | 26752214 | 110 | Mean Fluorescence intensity | 20 ug/ml | 1h | nan | Flow cytometry | Cellular uptake | NH2-SGASDDEEIAR-COOH |
SR11 | HeLa cells | FITC | 26752214 | 130 | Mean Fluorescence intensity | 20 ug/ml | 1.5h | nan | Flow cytometry | Cellular uptake | NH2-SGASDDEEIAR-COOH |
SR11 | HeLa cells | FITC | 26752214 | 140 | Mean Fluorescence intensity | 20 ug/ml | 2h | nan | Flow cytometry | Cellular uptake | NH2-SGASDDEEIAR-COOH |
IR15 | HeLa cells | FITC | 26752214 | 90 | Mean Fluorescence intensity | 20 ug/ml | 30min | nan | Flow cytometry | Cellular uptake | NH2-ICSSHYEPTVRIGGR-COOH |
IR15 | HeLa cells | FITC | 26752214 | 135 | Mean Fluorescence intensity | 20 ug/ml | 1h | nan | Flow cytometry | Cellular uptake | NH2-ICSSHYEPTVRIGGR-COOH |
IR15 | HeLa cells | FITC | 26752214 | 150 | Mean Fluorescence intensity | 20 ug/ml | 1.5h | nan | Flow cytometry | Cellular uptake | NH2-ICSSHYEPTVRIGGR-COOH |
IR15 | HeLa cells | FITC | 26752214 | 170 | Mean Fluorescence intensity | 20 ug/ml | 2h | nan | Flow cytometry | Cellular uptake | NH2-ICSSHYEPTVRIGGR-COOH |
PAK | A375 cells | FITC | 30904618 | 0 | nan | 20uM | 48h | 37ºC | Fluorescent Microscopy | Cellular uptake | GGEEEEEEEEPLGLAGRRRRRRRRGG |
?1H | HeLa cells | FITC | 28096156 | 18 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HeLa cells | FITC | 28096156 | 18 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HeLa cells | FITC | 28096156 | 19 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HeLa cells | FITC | 28096156 | 12 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?2H | HeLa cells | FITC | 28096156 | 13 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HeLa cells | FITC | 28096156 | 14 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HeLa cells | FITC | 28096156 | 12 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HeLa cells | FITC | 28096156 | 8 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?1H | HBMEC cells | FITC | 28096156 | 25 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HBMEC cells | FITC | 28096156 | 30 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HBMEC cells | FITC | 28096156 | 23 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?1H | HBMEC cells | FITC | 28096156 | 30 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | KSKTEYYNAWAVWERNAP |
?2H | HBMEC cells | FITC | 28096156 | 40 | Fluorescence intensity | 1uM | 2h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HBMEC cells | FITC | 28096156 | 45 | Fluorescence intensity | 1uM | 4h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HBMEC cells | FITC | 28096156 | 35 | Fluorescence intensity | 1uM | 6h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
?2H | HBMEC cells | FITC | 28096156 | 40 | Fluorescence intensity | 1uM | 24h | 37ºC | Flow cytometry | Cellular uptake | GNGEQREMAVSRLRDCLDRQA |
R8-CM?CD | MCF7 cells | FITC | 32589088 | 12 | Mean fluorescence intensity (%) | nan | 2h | nan | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
R8-CM?CD | MCF7 cells | FITC | 32589088 | 15 | Mean fluorescence intensity (%) | nan | 6h | nan | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
R8-CM?CD | MCF7 cells | FITC | 32589088 | 35 | Mean fluorescence intensity (%) | nan | 12h | nan | CLSM | Cellular uptake | RRRRRRRR-CM?CD |
Cf-OT20 | MonoMac6 cells | FITC | 30099595 | 5000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-TKPKGTKPKGTKPKGTKPKG |
Cf-Crot(1-9,38-42) | MonoMac6 cells | FITC | 30099595 | 15000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-YKQCHKKGGKKGSG |
Cf-Penetratin | MonoMac6 cells | FITC | 30099595 | 140000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-RQIKIWFQNRRMKWKK |
Cf-Dhvar4 | MonoMac6 cells | FITC | 30099595 | 200000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-KRLFKKLLFSLRKY |
Cf-Transportan | MonoMac6 cells | FITC | 30099595 | 40000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-AGYLLGKINLKALAALAKKIL |
Cf-Magainin | MonoMac6 cells | FITC | 30099595 | 10000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-GIGKFLHSAKKFGKAFVGEIMNS |
Cf-Melittin | MonoMac6 cells | FITC | 30099595 | 175000 | FITC Mean Intensity | 10uM | 2h | 37ºC | Flow cytometry | Cellular uptake | CF-GIGAVLKVLTTGLPALISWIKRKRQQ |
Pas2r12 | HEK293 cells | EGFP, immunoglobulin G | 30893557 | 1400 | Fluorescence intensity | 40uM | 45min | 37ºC | Flow cytometry | Cellular uptake | FFLIG-FFLIG-rrrrrrrrrrrr-NH2 |
A1 | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKKRRQRRR |
A2 | HeLa cells | FITC | 33355559 | 210 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | S5GRKS5RRQRRR |
A3 | HeLa cells | FITC | 33355559 | 220 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | R8GRKKRRS5RRR |
A4 | HeLa cells | FITC | 33355559 | 410 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKS5RRQS5RR |
A5 | HeLa cells | FITC | 33355559 | 80 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKERRQKRR |
A6 | HeLa cells | FITC | 33355559 | 370 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRAS5RRQS5RA |
A7 | HeLa cells | FITC | 33355559 | 120 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRAS5RRQS5RA |
A8 | HeLa cells | FITC | 33355559 | 25 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRAS5ARQS5RA |
A9 | HeLa cells | FITC | 33355559 | 200 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKR8RRQS5RR |
A10 | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKR8RRQXRR |
A11 | HeLa cells | FITC | 33355559 | 90 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKS5RRQXRR |
A3u | HeLa cells | FITC | 33355559 | 80 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | R8GRRKKRRS5RRR |
A4u | HeLa cells | FITC | 33355559 | 100 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRKS5RRQS5RR |
A6u | HeLa cells | FITC | 33355559 | 90 | Relative Mean Fluorescence intensity (%) | 2uM | 2h | nan | Flow cytometry | Cellular uptake | YGRAS5RRQS5RR |
C6M3 | CHO-K1 cells | siRNA-Cy3 labeled | 28349343 | 90 | Fluorescent cells (%) | nan | nan | nan | Flow cytometry | Cellular uptake | Ac-RLWHLLWRLWRRLHRLLR-NH2 |
AntpOVA | Dendritic cells | FITC | 27138940 | 50 | Cellular uptake (%) | 100ug/ml | 30min | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
AntpOVA | Dendritic cells | FITC | 27138940 | 45 | Cellular uptake (%) | 100ug/ml | 1h | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
AntpOVA | Dendritic cells | FITC | 27138940 | 45 | Cellular uptake (%) | 100ug/ml | 2h | 37ºC | Flow cytometry | Cellular uptake | RQIKIWFQNRRMKWKK-SIINFEKL |
Tylotoin-sC18* | HaCaT cells | Carboxyfluorescein | 30389988 | 1400 | Relative fluorescence | 10uM | 30min | 37ºC | Flow cytometry | Cellular uptake | KCVRQNNKRVCKGLRKRLRKFRNK-NH2 |
TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 13 | Cellular uptake | nan | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 10 | Cellular uptake | nan | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 9 | Cellular uptake | nan | 1h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 15 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 13 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 12 | Cellular uptake | nan | 2h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
TDCS-Tat NPs | Caco-2 cells | Cou-6 | 30672923 | 26 | Cellular uptake | nan | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | GRKKRRQRRRPQ |
TDCS-Pen NPs | Caco-2 cells | Cou-6 | 30672923 | 23 | Cellular uptake | nan | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RQIKIWFQNRRMKWKKGG |
TDCS-R8 NPs | Caco-2 cells | Cou-6 | 30672923 | 21 | Cellular uptake | nan | 4h | 37ºC | Fluorescent Microscopy | Cellular uptake | RRRRRRRR |
DsC18 | MCF7 cells | Carboxyfluorescein | 28332260 | 39 | Relative fluorescence | 25uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-GLRKRLRKFRNKIKEK |
DsC18(NIA)2 | MCF7 cells | Carboxyfluorescein | 28332260 | 40 | Relative fluorescence | 25uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-?A-GLRK-?A?A-NIA-RLRKFRNK-?A?A-NIA-IKEK |
DsC18 | MCF7 cells | Carboxyfluorescein | 28332260 | 130 | Relative fluorescence | 50uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-GLRKRLRKFRNKIKEK |
DsC18(NIA)2 | MCF7 cells | Carboxyfluorescein | 28332260 | 150 | Relative fluorescence | 50uM | 30min | 37ºC | Fluorescent Microscopy | Cellular uptake | CF-?A-GLRK-?A?A-NIA-RLRKFRNK-?A?A-NIA-IKEK |
BR2-Lp | HepG2 cells | Cou-6 | 28644728 | 125 | Mean Fluorescence intensity | 0.1ug/ml | 3h | 37ºC | Flow cytometry | Cellular uptake | RAGLQFPVGRLLRRL |
BR2-Lp | Miha cells | Cou-6 | 28644728 | 100 | Mean Fluorescence intensity | 0.1ug/ml | 3h | 37ºC | Flow cytometry | Cellular uptake | RAGLQFPVGRLLRRL |
CCMV | HeLa cells | Cy5 | 31257379 | 4000 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | Cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL |
SPIONs-PEG-gH625 | MDA-MB-231 cells | Cy5.5 | 28388503 | 384.8 | Fluorescence intensity | 100 mg/L | 15min | nan | Fluorescent Microscopy | Cellular uptake | AcHGLASTLTRWAHYNALIRAFC-CONH2 |
SPIONs-PEG-gH625 | MDA-MB-231 cells | Cy5.5 | 28388503 | 656.2 | Fluorescence intensity | 100 mg/L | 30min | nan | Fluorescent Microscopy | Cellular uptake | AcHGLASTLTRWAHYNALIRAFC-CONH2 |
Lp-PEI | HeLa cells | 5'-Cy3, LOR-2501 | 31544540 | 5 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
Lp-PP | HeLa cells | 5'-Cy3, LOR-2502 | 31544540 | 10 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
p-PPRP | HeLa cells | 5'-Cy3, LOR-2503 | 31544540 | 15.67 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
Lp-PEI | A549 cells | 5'-Cy3, LOR-2504 | 31544540 | 5 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
Lp-PP | A549 cells | 5'-Cy3, LOR-2505 | 31544540 | 12 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
p-PPRP | A549 cells | 5'-Cy3, LOR-2506 | 31544540 | 19.6 | Mean Fluorescence intensity | nan | 4h | 37ºC | CLSM | Cellular uptake | RRRRRRRR |
9R | HEK293 cells | dsRED | 30293549 | 0 | nan | nan | nan | nan | Fluorescent Microscopy | Penetration | RRRRRRRRR |
9K | HEK293 cells | dsRED | 30293549 | 0.7 | Mean Intensity | 20ug | 30min | nan | Fluorescent Microscopy | Penetration | KKKKKKKKK |
9K | HEK293 cells | dsRED | 30293549 | 1.3 | Mean Intensity | 20ug | 1h | nan | Fluorescent Microscopy | Penetration | KKKKKKKKK |
9K | HEK293 cells | dsRED | 30293549 | 1.4 | Mean Intensity | 20ug | 4h | nan | Fluorescent Microscopy | Penetration | KKKKKKKKK |
9K | HEK293 cells | dsRED | 30293549 | 1.8 | Mean Intensity | 20ug | 12h | nan | Fluorescent Microscopy | Penetration | KKKKKKKKK |
9K | HEK293 cells | dsRED | 30293549 | 1.6 | Mean Intensity | 20ug | 24h | nan | Fluorescent Microscopy | Penetration | KKKKKKKKK |
F6G6(rR)3R2 | HeLa cells | 4CzIPN | 30525541 | 97.2 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
F6G6(rR)3R2 | HeLa cells | NAI-DPAC | 30525541 | 44.1 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
F6G6(rR)3R2 | HeLa cells | BTZ-DMAC | 30525541 | 59.7 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
F6G6(rR)3R2 | NIH-3T3 cells | 4CzIPN | 30525541 | 57 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
F6G6(rR)3R2 | NIH-3T3 cells | NAI-DPAC | 30525541 | 10.3 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
F6G6(rR)3R2 | NIH-3T3 cells | BTZ-DMAC | 30525541 | 18 | Fluorescence intensity (%) | 2ug/mL | 5min | 37ºC | Flow cytometry | cellular internalization of NPs | FFFFFFGGGGGGrrrRR |
RLA | C6 cells | DB | 31617510 | 42.6 | Cellular uptake | 25uM | 30min | 37ºC | ELISA | cellular uptake | B12H11S(CH2)2COOH-rlarlarrlarlar |
r8 | C6 cells | DB | 31617510 | 4.6 | Cellular uptake | 25uM | 30min | 37ºC | ELISA | cellular uptake | B12H11S(CH2)2COOH-rrrrrrrr |
PEP-1 | HEK293T cells | GFP | 27516189 | 57.58 | GFP-positive population (%) | 20uM | 4h | nan | Flow cytometry | transfection | Ac-KETWWETWWTEWSQPKKKRKV-Cya |
CADY-2 | HEK293T cells | GFP | 27516189 | 58.7 | GFP-positive population (%) | 20uM | 4h | nan | Flow cytometry | transfection | Ac-GLWWRLWWRLRSWFRLWFRA-Cya |
R9 | Endothelial cells | CmLN | 26748549 | 18 | Mean Fluorescence intensity | 10uM | 4h | 37ºC | Flow cytometry | cellular uptake | RRRRRRRRR |
R9 | Endothelial cells | CmLN | 26748549 | 35 | Mean Fluorescence intensity | 25uM | 4h | 37ºC | Flow cytometry | cellular uptake | RRRRRRRRR |
R9 | Endothelial cells | CmLN | 26748549 | 50 | Mean Fluorescence intensity | 50uM | 4h | 37ºC | Flow cytometry | cellular uptake | RRRRRRRRR |
HBD | HeLa cells | rTCS, FITC | 27050721 | 0 | nan | 10uM | 10h | nan | CLSM | nan | GPGLWERQAREHSERKKRRRESECKAA |
pHLIP | MCF7 cells | SS-DOX | 25853477 | 20 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
pHLIP | MCF7 cells | SS-DOX | 25853477 | 40 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
pHLIP | MCF7 cells | SS-DOX | 25853477 | 24 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
pHLIP | MCF7 cells | SS-DOX | 25853477 | 35 | Mean Fluorescence intensity | 7uM | 3h | 37ºC | Flow cytometry | Cellular uptake | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
HSF | HTB-55 cells | FP | 30465781 | 0.15 | Drug transport | 1uM | 3h | nan | Fluorescent Microscopy | Drug transport | AcetlyNH-KCFQWQRNMRKVRGPPVSCIKR-CONH2 |
HSF | HTB-55 cells | SX/FP | 30465781 | 0.14 | Drug transport | 1uM | 3h | nan | Fluorescent Microscopy | Drug transport | AcetlyNH-KCFQWQRNMRKVRGPPVSCIKR-CONH2 |
Tpl | T98G cell | FITC | 31726199 | 40 | Percentage of FITC | 3uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Tpl | T98G cell | FITC | 31726199 | 55 | Percentage of FITC | 5uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Tpl | T98G cell | FITC | 31726199 | 70 | Percentage of FITC | 7uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Tpl | L929 cells | FITC | 31726199 | 3 | Percentage of FITC | 3uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Tpl | L929 cells | FITC | 31726199 | 5 | Percentage of FITC | 5uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Tpl | L929 cells | FITC | 31726199 | 2 | Percentage of FITC | 7uM | 1h | 37ºC | Flow cytometry | CPP activity | NH2-KWCFRVCYRGICYRRCR-CONH2 |
Hpp3 | ECV304 cells | FITC | 27070736 | 3000 | Fluorescence intensity | 2.5uM | 1h | 37ºC | Fluorescence spectroscopy | cellular uptake | KPKRKRRKKKGHGWSR |
Hpp3 | ECV304 cells | FITC | 27070736 | 5000 | Fluorescence intensity | 5uM | 1h | 37ºC | Fluorescence spectroscopy | cellular uptake | KPKRKRRKKKGHGWSR |
Hpp3 | ECV304 cells | FITC | 27070736 | 5200 | Fluorescence intensity | 7.5uM | 1h | 37ºC | Fluorescence spectroscopy | cellular uptake | KPKRKRRKKKGHGWSR |
Hpp3 | ECV304 cells | FITC | 27070736 | 5800 | Fluorescence intensity | 10uM | 1h | 37ºC | Fluorescence spectroscopy | cellular uptake | KPKRKRRKKKGHGWSR |
Kkd-5 | HeLa cells | FITC | 28349160 | 30 | Relative Mean Fluorescence intensity (%) | 5uM | 4h | 37ºC | Flow cytometry | cellular uptake | nan |
Kkd-5 | HeLa cells | FITC | 28349160 | 70 | Relative Mean Fluorescence intensity (%) | 10uM | 4h | 37ºC | Flow cytometry | cellular uptake | nan |
Kkd-5 | HeLa cells | FITC | 28349160 | 97 | Relative Mean Fluorescence intensity (%) | 25uM | 4h | 37ºC | Flow cytometry | cellular uptake | nan |
Fol-Pep1 | HeLa cells | FITC | 26544061 | 17 | Mean Fluorescence intensity | nan | 2h | 37ºC | Flow cytometry | cellular uptake | folate-KETWWETWWTEWSQPKKKRKVC |
Fol-Pep2 | HaCaT cells | FITC | 26544061 | 8 | Mean Fluorescence intensity | nan | 2h | 37ºC | Flow cytometry | cellular uptake | folate-KETWWETWWTEWSQPKKKRKVC |
R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 28 | Cellular uptake | 2.5 | nan | 37ºC | Flow cytometry | cellular uptake | RRRRRRRR |
RP/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 58 | Cellular uptake | 2.5 | nan | 37ºC | Flow cytometry | cellular uptake | RRRRRRRR |
MRP/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 35 | Cellular uptake | 2.5 | nan | 37ºC | Flow cytometry | cellular uptake | RRRRRRRR |
D-arm/R8-modified MITO-Porter | HeLa cells | NBD | 27056631 | 40 | Cellular uptake | 2.5 | nan | 37ºC | Flow cytometry | cellular uptake | RRRRRRRR |
CPP 2 | RAW264.7 cells | FITC | 30095906 | 71.9 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | cellular uptake | GFAWNVCVYRNGVRVCHRRAN |
CPP 6 | RAW264.7 cells | FITC | 30095906 | 95.8 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | cellular uptake | YGRKKRRQRRR-C-MC-VC-PABC-GFAWNVCVYRNGVRVCHRRAN |
CPP 7 | RAW264.7 cells | FITC | 30095906 | 75.2 | Intracellular FITC-labeled peptides (%) | 5uM | 2h | 37ºC | Flow cytometry | cellular uptake | GFAWNVCVYRNGVRVCHRRAN-NH2 |
gH625 | HeLa cells | PtNPs | 28758654 | 0 | nan | nan | nan | nan | STEM | cellular uptake | Ac-HGLASTLTRWAHYNALIRAFK(Mtt)GGGC-NH2 |
DEN-K(GALA)-TAT-K(STR) | HeLa cells | Alexa488–eGFP siRNA | 28093948 | 7,50E+05 | Mean Fluorescence intensity | 100 | 4h | 37ºC | Flow cytometry | cellular uptake | DEN-K(WEAALAEALAEALAEHLAEALAEALEALAA)-GRKKRRQRRRPPQ-K(STR) |
MPG | Caco-2 cells | TAMRA, iCAL36 | 31283917 | 39 | Normalized Fluorescence | nan | 1.5h | 37ºC | Flow cytometry | cellular uptake | GALFLGWLGAAGSTMGAWSQPKKKRKV-ANSRWPTSII |
C6M1 | Caco-2 cells | TAMRA, iCAL36 | 31283917 | 93 | Normalized Fluorescence | nan | 1.5h | 37ºC | Flow cytometry | cellular uptake | RLWRLLWRLWRRLWRLLR-ANSRWPTSII |
WRAP5 | Caco-2 cells | TAMRA, iCAL36 | 31283917 | 257 | Normalized Fluorescence | nan | 1.5h | 37ºC | Flow cytometry | cellular uptake | LLRLLRWWWRLLRLL-ANSRWPTSI |
SAP(E) | nan | nan | 27237727 | 0 | nan | nan | nan | nan | nan | nan | AcCGGWVELPPPVELPPPVELPPP-NH2 |
CGA-N9 | C. tropicaliscells | Propidium iodide (PI) | 30610128 | 2.25 | Fluorescence intensity | 3.9mg/ml | 2h | 28ºC | Flow cytometry | cellular uptake | NH2-RILSILRHQ-COOH |
MeG10 | HeLa cells | FITC | 27039278 | 2200 | Mean Fluorescence intensity | 5uM | nan | 37ºC | CLSM | cellular uptake | RRRRRRRR |
dG5 | HeLa cells | FITC | 27039278 | 200 | Mean Fluorescence intensity | 5uM | nan | 37ºC | CLSM | cellular uptake | RRRRRRRR |
dG10 | HeLa cells | FITC | 27039278 | 1500 | Mean Fluorescence intensity | 5uM | nan | 37ºC | CLSM | cellular uptake | RRRRRRRR |
PGON20 | HeLa cells | FITC | 27039278 | 2200 | Mean Fluorescence intensity | 5uM | nan | 37ºC | CLSM | cellular uptake | RRRRRRRR |
MePh10-b-dG5 | HeLa cells | FITC | 27039278 | 500 | Mean Fluorescence intensity | 5uM | nan | 37ºC | CLSM | cellular uptake | RRRRRRRR |
RG301 | HeLa cells | Carboxyfluorescein | 34333729 | 100 | Cellular uptake (%) | 10uM | 4h | 37ºC | Flow cytometry | cellular uptake | RaDPAYQaRFLGKrKfIcL |
RG302 | HeLa cells | Carboxyfluorescein | 34333729 | 100 | Cellular uptake (%) | 10uM | 4h | 37ºC | Flow cytometry | cellular uptake | KrKfIcLGRaDPAYQaRFL |
CTX-M1 | HeLa cells | Alexa488 | 28459137 | 40 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
CTX-M2 | HeLa cells | Alexa488 | 28459137 | 38 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
CTX-M1 | HeLa cells | Cy5.5 | 28459137 | 49 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
CTX-M2 | HeLa cells | Cy5.5 | 28459137 | 75 | Relative fluorescence (%) | 6uM | 1h | 37ºC | Flow cytometry | internalization of fluorescently labeled peptides | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
HBHAc | HepG2 cells | eGFP | 31524004 | 55 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
HBHAc | HepG2 cells | eGFP | 31524004 | 30 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
HBHAc | HepG2 cells | eGFP | 31524004 | 20 | Mean Fluorescence intensity | 3uM | 1h | 37ºC | Flow cytometry | cellular uptake | KKAAPAKKAAAKKAPAKKAAAKK |
[WR]5 | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1000 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | FACS | cellular uptake | WRWRWRWRWR |
c[C(WR)4C] | CCRF-CEM cells | F'-GpYEEI | 32498339 | 200 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | FACS | cellular uptake | CWRWRWRWRC |
l(C(WR)4C) | CCRF-CEM cells | F'-GpYEEI | 32498339 | 700 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | FACS | cellular uptake | CWRWRWRWRC |
c[C(WR)5C] | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1050 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | FACS | cellular uptake | CWRWRWRWRWRC |
l(C(WR)5C) | CCRF-CEM cells | F'-GpYEEI | 32498339 | 1100 | Mean Fluorescence intensity | 25uM | 3h | 37ºC | FACS | cellular uptake | CWRWRWRWRWRC |
CPP 12 | HeLa cells | Carboxyfluorescein | 33838611 | 550 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac6cNH2-RR-Ac6cNH2-RR-Ac6cNH2-NH2 |
CPP 13 | HeLa cells | Carboxyfluorescein | 33838611 | 400 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac5cNH2-RR-Ac5cNH2-RR-Ac5cNH2-NH2 |
CPP 14 | HeLa cells | Carboxyfluorescein | 33838611 | 2600 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRRRRRRRRR-NH2 |
CPP 12 | HEK293 cells | Carboxyfluorescein | 33838611 | 110 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac6cNH2-RR-Ac6cNH2-RR-Ac6cNH2-NH2 |
CPP 13 | HEK293 cells | Carboxyfluorescein | 33838611 | 1200 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRR-Ac5cNH2-RR-Ac5cNH2-RR-Ac5cNH2-NH2 |
CPP 14 | HEK293 cells | Carboxyfluorescein | 33838611 | 2800 | Mean Fluorescence intensity | 2uM | 2h | nan | Flow cytometry | Intracellular levels of peptides | CF-GRRRRRRRRR-NH2 |
SAHM1 | HeLa cells | FITC | 28757184 | 16 | Mean Fluorescence intensity | 5uM | 90min | nan | Flow cytometry | cellular uptake | ?A1a-ERLRRRI-S5-LCR-S5-HHST |
StAx | HeLa cells | FITC | 28757184 | 3 | Mean Fluorescence intensity | 5uM | 90min | nan | Flow cytometry | cellular uptake | RRWPRXILDXHVRRVWR |
LMWP | HT1080 cells | mCherry, His-tag | 29058417 | 0 | nan | nan | nan | nan | Flow cytometry | cellular uptake | VSRRRRRRGGRRRR |
PI | A549 cells | siRNA | 27480031 | 90 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KLULKLULKULKAULKLUGC(cRGDfC)-NH2 |
PI-acetamide | A549 cells | siRNA | 27480031 | 50 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KLULKLULKULKAULKLUGC(CH2CONH2)-NH2 |
PII | A549 cells | siRNA | 27480031 | 20 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KLULKLULKULKAC(cRGDfC)LKLUG-NH2 |
PIII | A549 cells | siRNA | 27480031 | 92 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KC(cRGDfC)ULKLULKULKAC(cRGDfC)LKLUG-NH2 |
PIV | A549 cells | siRNA | 27480031 | 5 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KLULKLUC(cRGDfC)KULKAC(cRGDfC)LKLUG-NH2 |
PV | A549 cells | siRNA | 27480031 | 15 | Mean Fluorescence intensity/mg protein | 2.5uM | 8h | 37ºC | Fluorometer | cellular uptake | Acetyl-KC(cRGDfC)ULKLUC(cRGDfC)KULKAC(cRGDfC)LKLUG-NH2 |
Lys-peptide 1 | HeLa cells | nan | 26814673 | 90 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | cellular uptake | TMR-GKKKKKKKKK-NH2 |
Arg-peptide 2 | HeLa cells | nan | 26814673 | 500 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | cellular uptake | TMR-GRRRRRRRRR-NH2 |
Lys(AEt)-peptide 3 | HeLa cells | nan | 26814673 | 10 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | cellular uptake | TMR-G(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)(AEt)-NH2 |
Lys(GEt)-peptide 4 | HeLa cells | nan | 26814673 | 200 | RFU/mg | 1uM | 2h | 4ºC | Fluorescence spectroscopy | cellular uptake | TMR-G(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)(GEt)-NH2 |
KIW7 | HeLa cells | pDNA | 32329496 | 0 | nan | nan | nan | nan | CLSM | nan | NH2-KIWFQNR-COOH |
mPrPA488 | N2a cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | cellular uptake | ALFVKLMGTPLDNAKWTLCPVLRGMWKY |
bPrPA488 | N2a cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | cellular uptake | KPACVIKMVS-WKIGPVSDLKLVKSFGLMRW |
mPrPA488 | HeLa cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | cellular uptake | ALFVKLMGTPLDNAKWTLCPVLRGMWKY |
bPrPA488 | HeLa cells | Alexa488 | 27818203 | 1 | Cellular uptake | 1uM | 24h | 4ºC | CLSM | cellular uptake | KPACVIKMVS-WKIGPVSDLKLVKSFGLMRW |
stearyl-r8 | HeLa cells | CD63-GFP Evs | 27748399 | 3340 | Relative Cellular uptake | 16uM | 24h | 37ºC | CLSM | cellular uptake | CH3(CH2)16-CO-NH-D(Arg)8-NH2 |
stearyl-sC18 | MCF7 cells | CD63-GFP Evs | 34365796 | 692 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | cellular uptake | CH3(CH2)16-CONH-GGGGLRKRLRKFRNKIKEK-NH2 |
stearyl-(sC18)2 | MCF7 cells | CD63-GFP Evs | 34365796 | 777 | Relative Cellular uptake | 2uM | 24h | 37ºC | Flow cytometry | cellular uptake | NH2-GLRK(KEKIKNRFKRLRKRLGGGG-NH2CO-CH3(CH2)16)RLRKFRNKIKEK-NH2 |
sC18 | MCF7 cells | CD63-GFP Evs | 34365796 | 128 | Relative Cellular uptake | 10uM | 24h | 37ºC | Flow cytometry | cellular uptake | NH2-GLRKRLRKFRNKIKEK-amide |
(sC18)2 | MCF7 cells | CD63-GFP Evs | 34365796 | 78 | Relative Cellular uptake | 2uM | 24h | 37ºC | Flow cytometry | cellular uptake | NH2-GLRK(RLRKFRKEKIKNRFKRLRKRLG-NH2)NKIKEK-amide |
T-hNP | B16 cells | Rh-PE | 28954191 | 9 | Mean Fluorescence intensity | nan | 15 min | 37ºC | Flow cytometry | cellular uptake | GRKKRRQRRRPQ |
peptide 1 | HeLa cells | DUB | 32831622 | 0 | nan | nan | nan | nan | nan | nan | Ac-RWVRVpGO(FAM)WIRQ-LRGG-AFC |
peptide 2 | HeLa cells | DUB | 32831622 | 0 | nan | nan | nan | nan | nan | nan | Ac-RWVRVpGO(FAM)WIRQ-LVLRLRGG-AFC |
peptide 3 | HeLa cells | DUB | 32831622 | 0 | nan | nan | nan | nan | nan | nan | Z-LRGGAMC |
peptide 4 | HeLa cells | DUB | 32831622 | 0 | nan | 30uM | 1h | 37ºC | Flow cytometry | cellular uptake | Ac-RWVRVpGO(FAM)WIRQLRGG-NH2 |
COSS 4 | HeLa cells | TAMRA | 27774725 | 150 | Mean Fluorescence intensity | nan | 1h | 37ºC | Flow cytometry | cellular uptake | nan |
POSS-(PEG-NLS-G-TAT)8 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 2000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CPKKKRKVEDPGGRKKRRQRRRPQ |
POSS-(PEG-NLS-G-TAT-G-REDV)8 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 2100 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CPKKKRKVEDPGGRKKRRQRRRPQGREDV |
TP-H12 | Endothelial cells | Cy5-oligonucleotide | 32254599 | 7000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | REDVGRKKRRQRRRPQCPKKKRKVEDPHHHHHHHHHHHH |
L6 | A549 cells | FITC | 30360131 | 0 | nan | nan | nan | nan | Fluorescent Microscopy | Cellular internalization of CPP-FITC | RRWQWR |
H6 | BY-2 plant cells | TAMRA | 27885926 | 9000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHH-NH2 |
H8 | BY-2 plant cells | TAMRA | 27885926 | 15000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHH-NH2 |
H10 | BY-2 plant cells | TAMRA | 27885926 | 12000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHH-NH2 |
H12 | BY-2 plant cells | TAMRA | 27885926 | 5000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHH-NH2 |
H14 | BY-2 plant cells | TAMRA | 27885926 | 6000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHH-NH2 |
H16 | BY-2 plant cells | TAMRA | 27885926 | 6000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHHHH-NH2 |
H18 | BY-2 plant cells | TAMRA | 27885926 | 3000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHHHHHH-NH2 |
H20 | BY-2 plant cells | TAMRA | 27885926 | 3000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHHHHHHHH-NH2 |
H22 | BY-2 plant cells | TAMRA | 27885926 | 1000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHHHHHHHHHH-NH2 |
H24 | BY-2 plant cells | TAMRA | 27885926 | 2000 | Cellular uptake | 1uM | 12h | 27ºC | CLSM | cellular uptake | HHHHHHHHHHHHHHHHHHHHHHHH-NH2 |
Lip-Cou6 | MCF7 cells | Cou-6 | 35539172 | 40 | Mean Fluorescence intensity | nan | 1h | 37ºC | Flow cytometry | cellular uptake | PFVYL-Cou6 |
PFV-Lip-Cou6 | MCF7 cells | Cou-6 | 35539172 | 90 | Mean Fluorescence intensity | nan | 1h | 37ºC | Flow cytometry | cellular uptake | PFVYL-Lip-Cou6 |
His16-Lyso | HT1080 cells | lysosomes | 31426598 | 100 | Relative cellular uptake (%) | nan | nan | 37ºC | Flow cytometry | cellular uptake | stearly-His6-HHHHHHHHHHHHHHHH–NH2 |
R9 | A549 cells | chitosan/siRNA | 26568525 | 70 | Cellular uptake (%) | nan | nan | nan | Flow cytometry | cellular uptake | RRRRRRRRR |
R9G4 | A549 cells | chitosan/siRNA | 26568525 | 80 | Cellular uptake (%) | nan | nan | nan | Flow cytometry | cellular uptake | RRRRRRRRRGGGG |
R9G10 | A549 cells | chitosan/siRNA | 26568525 | 90 | Cellular uptake (%) | nan | nan | nan | Flow cytometry | cellular uptake | RRRRRRRRRGGGGGGGGGG |
RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 350 | Mean Fluorescence intensity | 6ug/mL | 1h | 37ºC | Flow cytometry | cellular uptake | HHHHHH-RRRRRRRRRRR |
RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 800 | Mean Fluorescence intensity | 12ug/mL | 2h | 37ºC | Flow cytometry | cellular uptake | HHHHHH-RRRRRRRRRRR |
RhB-NLC-R11 | HaCaT cells | RhB | 31447556 | 1050 | Mean Fluorescence intensity | 25ug/mL | 4h | 37ºC | Flow cytometry | cellular uptake | HHHHHH-RRRRRRRRRRR |
ppTG21 | HepG2 cells | GFP | 30994954 | 0.3 | Fluorescence intensity | 30uM | 90min | nan | CLSM | cellular uptake | NH2-GLFHALLHLLHSLWHLLLHA-CONH2 |
ppTG21 | HepG2 cells | GFP, 1TAG-3CIY | 30994954 | 0.5 | Fluorescence intensity | 30uM | 90min | nan | CLSM | cellular uptake | NH2-GLFHALLHLLHSLWHLLLHA-CONH2 |
ppTG21 | HepG2 cells | GFP, 1TAG-3BrY | 30994954 | 0.6 | Fluorescence intensity | 30uM | 90min | nan | CLSM | cellular uptake | NH2-GLFHALLHLLHSLWHLLLHA-CONH2 |
ppTG21 | HepG2 cells | GFP, 1TAG-3IY | 30994954 | 1.3 | Fluorescence intensity | 30uM | 90min | nan | CLSM | cellular uptake | NH2-GLFHALLHLLHSLWHLLLHA-CONH2 |
ppTG21 | HepG2 cells | GFP, 2TAG-3IY | 30994954 | 1.5 | Fluorescence intensity | 30uM | 90min | nan | CLSM | cellular uptake | NH2-GLFHALLHLLHSLWHLLLHA-CONH2 |
Cys-penetratin | TR146 cell | Alexa 647-sCT | 35210769 | 3800 | Relative Mean Fluorescence intensity | nan | 24h | 37ºC | FACS | cellular uptake | CRQIKIWFQNRRMKWKK |
PFV | U87 cells | Doxorubicin | 30261346 | 52 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
PFV | bEnd.3 cells | Doxorubicin | 30261346 | 50 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
PFV | Glial cells | Doxorubicin | 30261346 | 50 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
Tf-PFV | U87 cells | Doxorubicin | 30261346 | 65 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
Tf-PFV | bEnd.3 cells | Doxorubicin | 30261346 | 5 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
Tf-PFV | Glial cells | Doxorubicin | 30261346 | 62 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
PFV | U87 cells | Erlo | 30261346 | 45 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
PFV | bEnd.3 cells | Erlo | 30261346 | 47 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
PFV | Glial cells | Erlo | 30261346 | 43 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | PFVYLI |
Tf-PFV | U87 cells | Erlo | 30261346 | 70 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
Tf-PFV | bEnd.3 cells | Erlo | 30261346 | 69 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
Tf-PFV | Glial cells | Erlo | 30261346 | 65 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | Tf-PFVYLI |
PPP | MCF7 cells | NPs | 27043442 | 90 | Mean Fluorescence intensity | nan | 30min | nan | Flow cytometry | cellular uptake | CGRRMKWKK-Psaa-GGGG-EEEERRRR |
PPP | MCF7 cells | NPs | 27043442 | 110 | Mean Fluorescence intensity | nan | 30min | nan | Flow cytometry | cellular uptake | CGRRMKWKK-Psaa-GGGG-EEEERRRR |
Rq | HeLa cells | PTX, FITC | 29026300 | 62.65 | Percentage (%) | 10uM | 30min | 37ºC | Flow cytometry | cellular uptake | RRRRQWWQW |
Rq | HeLa cells | PTX, FITC | 29026300 | 73.35 | Percentage (%) | 100uM | 30min | 37ºC | Flow cytometry | cellular uptake | RRRRQWWQW |
KALA | BMDC | ssPalmE,DiD | 31386869 | 11000 | Geo Mean Fluorescence intensity | nan | 2h | nan | FACS | cellular uptake | WEAKLAKALAKALAKHLAKALAKALK |
KALA | BMDC | ssPalmM,DiD | 31386869 | 12000 | Geo Mean Fluorescence intensity | nan | 2h | nan | FACS | cellular uptake | WEAKLAKALAKALAKHLAKALAKALK |
RU006 | HeLa cells | Doxorubicin | 29113134 | 0.4 | Fluorescence intensity | 10uM | 6h | 25ºC | CLSM | Dox encapsulation | Ac-AIAKAXKIA-NH2 |
RU006 | HeLa cells | Doxorubicin | 29113134 | 0.6 | Fluorescence intensity | 20uM | 6h | 25ºC | CLSM | Dox encapsulation | Ac-AIAKAXKIA-NH2 |
RU006 | HeLa cells | Doxorubicin | 29113134 | 0.8 | Fluorescence intensity | 50uM | 6h | 25ºC | CLSM | Dox encapsulation | Ac-AIAKAXKIA-NH2 |
BP9 | HepG2 cells | Doxorubicin | 31452330 | 0 | nan | nan | 3h | 37ºC | CLSM | cellular uptake | AHLHNRS |
COL-CPP | A549 cells | FITC | 28835794 | 1,50E+04 | Mean Fluorescence intensity | 15uM | 30min | 37ºC | Flow cytometry | cellular uptake | FITC-A?-GG-(P-Hyp-G)8-RRGRRG |
COL-CPP | A549 cells | FITC | 28835794 | 2,40E+04 | Mean Fluorescence intensity | 30uM | 30min | 37ºC | Flow cytometry | cellular uptake | FITC-A?-GG-(P-Hyp-G)8-RRGRRG |
COL-CPP | A549 cells | FITC | 28835794 | 5,00E+05 | Mean Fluorescence intensity | 90uM | 30min | 37ºC | Flow cytometry | cellular uptake | FITC-A?-GG-(P-Hyp-G)8-RRGRRG |
TH | HeLa cells | FITC | 28603674 | 1600 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
TH | HeLa cells | FITC | 28603674 | 1700 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
TH | HeLa cells | FITC | 28603674 | 2750 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHINLHHLAHL(Aib)HHIL-NH2 |
Methly-TH | HeLa cells | FITC | 28603674 | 1550 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
Methly-TH | HeLa cells | FITC | 28603674 | 1600 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
Methly-TH | HeLa cells | FITC | 28603674 | 1900 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHMINLHMHMLAHML(Aib)HMHMIL-NH2 |
Ethyl-TH | HeLa cells | FITC | 28603674 | 1200 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
Ethyl-TH | HeLa cells | FITC | 28603674 | 1100 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
Ethyl-TH | HeLa cells | FITC | 28603674 | 2250 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHEINLHEHELAHEL(Aib)HEHEIL-NH2 |
Isopropyl-TH | HeLa cells | FITC | 28603674 | 1750 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
Isopropyl-TH | HeLa cells | FITC | 28603674 | 1500 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
Isopropyl-TH | HeLa cells | FITC | 28603674 | 2250 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHIINLHIHILAHIL(Aib)HIHIIL-NH2 |
Butyl-TH | HeLa cells | FITC | 28603674 | 2200 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
Butyl-TH | HeLa cells | FITC | 28603674 | 2800 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
Butyl-TH | HeLa cells | FITC | 28603674 | 2500 | Fluorescence intensity | 5uM | 1h | 37ºC | FACS | cellular uptake | AGYLLGHBINLHBHBLAHBL(Aib)HBHBIL-NH2 |
NC-2 | hPSC cells | FAM-labeled AMO | 28524768 | 155 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | cellular uptake | RRRRGGRRRRRRSV-C-S-SC-VSRRRRRRGGRRRR |
NC-2 | BJ-fibroblasts | FAM-labeled AMO | 28524768 | 15 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | cellular uptake | RRRRGGRRRRRRSV-C-S-SC-VSRRRRRRGGRRRR |
NC-2 | Panc-1 | FAM-labeled AMO | 28524768 | 10 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | cellular uptake | RRRRGGRRRRRRSV-C-S-SC-VSRRRRRRGGRRRR |
NC-2 | AsPc-1 | FAM-labeled AMO | 28524768 | 3 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | cellular uptake | RRRRGGRRRRRRSV-C-S-SC-VSRRRRRRGGRRRR |
NC-2 | MiaPaCa-2 | FAM-labeled AMO | 28524768 | 3 | Mean Fluorescence intensity | nan | 6h | 37ºC | Flow cytometry | cellular uptake | RRRRGGRRRRRRSV-C-S-SC-VSRRRRRRGGRRRR |
dNP2 | HeLa cells | FITC | 32254889 | 100 | Fluorescence intensity | nan | 4h | nan | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | HeLa cells | FITC | 32254889 | 350 | Fluorescence intensity | nan | 18h | nan | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
SAH-P53-8 | HeLa cells | Rho | 29150077 | 700 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | QSQQTFNLWKLLQN |
SAH-p53-4 | HeLa cells | Rho | 29150077 | 500 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | LSQETFDLWKLLEN |
BP1.2 | HeLa cells | Rho | 29150077 | 1200 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | RSQRRFRLWRLLEN |
BP1.3 | HeLa cells | Rho | 29150077 | 1700 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | RRRRRFDLWKLLEN |
BP1.4 | HeLa cells | Rho | 29150077 | 3500 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | RSQERFDLWKLLEN |
BP1.5 | HeLa cells | Rho | 29150077 | 1500 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | LRRETFDRWKRLRR |
BP1.6 | HeLa cells | Rho | 29150077 | 2500 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | LSQETFRLWRRLRR |
BP1.7 | HeLa cells | Rho | 29150077 | 1600 | Cellular uptake | nan | 30min | 37ºC | Flow cytometry | cellular uptake | LRRETFDLWKRLRR |
rEETI-II | HeLa cells | Xfect, Alexa488, Noco | 31061420 | 50 | FITC per cell (%) | 5uM | 1h | 37ºC | Flow cytometry | cellular uptake | CPRILMRCKQDSDCLAGCVCGPNGFCG |
rEETI-II | HeLa cells | Xfect, Alexa488, IKA | 31061420 | 40 | FITC per cell (%) | 5uM | 1h | 37ºC | Flow cytometry | cellular uptake | CPRILMRCKQDSDCLAGCVCGPNGFCG |
RP7 | bEnd.3 cells | NRP1, FITC | 33508290 | 3,20E+05 | Cell Count | nan | 1h | 37ºC | Flow cytometry | cellular uptake | RPARPAR |
Tat-C-RP7 | bEnd.3 cells | NRP1, FITC | 33508290 | 2,80E+06 | Cell Count | nan | 1h | 37ºC | Flow cytometry | cellular uptake | RKKRRQRRRCRPARPAR |
NR2B9c | BCECs cells | TAMRA | 32674358 | 0.02 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | live cell peptide uptake | KLSSIESDV |
Tat-NR2B9c | BCECs cells | TAMRA | 32674358 | 0.09 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | live cell peptide uptake | YGRKKRRQRRRKLSSIESDV |
Tat-N-dimer | BCECs cells | TAMRA | 32674358 | 0.05 | Cell peptide accumulation (mol*cm^-2) | 100uM | 3h | 37ºC | Fluorescent Microscopy | live cell peptide uptake | YGRKKRRQRRRNPEG4(IETDV)2 |
CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 1500 | Mean value of cellular uptake | 1uM | 4h | 37ºC | Flow cytometry | cellular uptake | KLKLALALALAVQRKRQKLMPC |
CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 500 | Mean value of cellular uptake | 0.1uM | 4h | 37ºC | Flow cytometry | cellular uptake | KLKLALALALAVQRKRQKLMPC |
CB5005-Cy | U87 cells | Carboxyfluorescein | 30243823 | 70 | Mean value of cellular uptake | 0.01uM | 4h | 37ºC | Flow cytometry | cellular uptake | KLKLALALALAVQRKRQKLMPC |
Dox-SS[C(WR)4K] | HT1080 cells | Doxorubicin | 30396106 | 8000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | cellular uptake | CWRWRWRWRK |
Dox-SS[C(WR)4K] | HEK293 cells | Doxorubicin | 30396106 | 6000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | cellular uptake | CWRWRWRWRK |
Dox-SS[C(WR)4K] | SK-OV-3 cells | Doxorubicin | 30396106 | 13000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | cellular uptake | CWRWRWRWRK |
Dox-SS[C(WR)4K] | CCRF-CEM cells | Doxorubicin | 30396106 | 5000 | Mean Fluorescence intensity | 50uM | 3h | 37ºC | Flow cytometry | cellular uptake | CWRWRWRWRK |
KL4 | A549 cells | siRNA | 32352853 | 75 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | cellular uptake | KLLLLKLLLLKLLLLKLLLLK-NH2 |
KA2 | A549 cells | siRNA | 32352853 | 0 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | cellular uptake | KAALLKAALLKAALLKAALLK-NH2 |
KV4 | A549 cells | siRNA | 32352853 | 90 | Cellular uptake (%) | 3000 pmol | 4h | 37ºC | Flow cytometry | cellular uptake | KVVVVKVVVVKVVVVKVVVVK-NH2 |
DNP | Caco-2 cells | Carboxyfluorescein | 28757359 | 2 | Uptake amount (x10^3 pfu/ug protein) | 10uM | 10min | 37ºC | CLSM | uptake stude | C-DNPGNET-C |
DRIM | HEK293 cells | nan | 28921993 | 8 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | QQRKRKIWSILAPLGTTLVKLVAGIG-NH2 |
WWSP | HEK293 cells | nan | 28921993 | 10 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | PLILLRLLRGQF-NH2 |
KFGF | HEK293 cells | nan | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | AAVLLPVLLAAP-NH2 |
MAP-1 | HEK293 cells | nan | 28921993 | 20 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | KLALKALKALKAALKLA-NH2 |
sDRIM | HEK293 cells | nan | 28921993 | 5 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | QQRKRKIWSKLAPDGTTLVKLVAGIG-NH2 |
sWWSP | HEK293 cells | nan | 28921993 | 2 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | PLIKLRLDRGQF-NH2 |
sKFGF | HEK293 cells | nan | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | AAKLLPDLLAAP-NH2 |
sMAP-1 | HEK293 cells | nan | 28921993 | 18 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | KLALKALKKLKADLKLA-NH2 |
DRIM | HeLa cells | nan | 28921993 | 20 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | QQRKRKIWSILAPLGTTLVKLVAGIG-NH2 |
WWSP | HeLa cells | nan | 28921993 | 10 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | PLILLRLLRGQF-NH2 |
KFGF | HeLa cells | nan | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | AAVLLPVLLAAP-NH2 |
MAP-1 | HeLa cells | nan | 28921993 | 25 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | KLALKALKALKAALKLA-NH2 |
sDRIM | HeLa cells | nan | 28921993 | 3 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | QQRKRKIWSKLAPDGTTLVKLVAGIG-NH2 |
sWWSP | HeLa cells | nan | 28921993 | 2 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | PLIKLRLDRGQF-NH2 |
sKFGF | HeLa cells | nan | 28921993 | 1 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | AAKLLPDLLAAP-NH2 |
sMAP-1 | HeLa cells | nan | 28921993 | 15 | Normalized fluorescence intensities | 2uM | 4h | 37ºC | FACS | cellular uptake | KLALKALKKLKADLKLA-NH2 |
Cur | MCF7 cells | NPs | 31691601 | 5500 | Fluorescence intensity | 25ug/ml | 4h | 37ºC | Flow cytometry | cellular uptake | (ACP)-GPLGIAGQrrrrrrrrr-(ACP) |
Cur | MCF7 cells | P-NPs | 31691601 | 9000 | Fluorescence intensity | 25ug/ml | 4h | 37ºC | Flow cytometry | cellular uptake | (ACP)-GPLGIAGQrrrrrrrrr-(ACP) |
C9-PNA | U87 cells | FITC | 31497713 | 6,00E+05 | FITC count | 0.5uM | 2h | 37ºC | Flow cytometry | cellular uptake | FfRrRrE |
PEG2k-ppTAT-PEG1k-PE | A549 cells | MMP2 | 28870072 | 280 | PTX | 2mg/ml | 4h | 37ºC | Flow cytometry | cellular uptake | GPLGIAGQYGRKKRRQRRRC |
PEG2k-ppTAT-PEG1k-PE | MCF7 cells | MMP2 | 28870072 | 200 | PTX | 2mg/ml | 4h | 37ºC | Flow cytometry | cellular uptake | GPLGIAGQYGRKKRRQRRRC |
StA-R8 | HepG2 cells | Cy3-siRNA | 27354583 | 40 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CH3(CH2)16-CONH-RRRRRRRR |
StA-R8 | A549 cells | Cy3-siRNA | 27354583 | 48 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CH3(CH2)16-CONH-RRRRRRRR |
StA-R8 liposome | HepG2 cells | Cy3-siRNA | 27354583 | 45 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CH3(CH2)16-CONH-RRRRRRRRRR |
StA-R8 liposome | A549 cells | Cy3-siRNA | 27354583 | 50 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CH3(CH2)16-CONH-(Arg)10 |
vaults 1a | RAW264.7 cells | FITC | 28029784 | 10000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Cleavable 8 | RAW264.7 cells | FITC | 28029784 | 20000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Noncleavable 12 | RAW264.7 cells | FITC | 28029784 | 80000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
vaults 1a | HeLa cells | FITC | 28029784 | 3500 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Cleavable 8 | HeLa cells | FITC | 28029784 | 4500 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Noncleavable 12 | HeLa cells | FITC | 28029784 | 6000 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
vaults 1a | CHO-K1 cells | FITC | 28029784 | 1800 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Cleavable 8 | CHO-K1 cells | FITC | 28029784 | 2300 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
Vault-r8Noncleavable 12 | CHO-K1 cells | FITC | 28029784 | 2600 | Mean Fluorescence intensity | 10ug | 16h | 37ºC | Flow cytometry | cellular uptake | MAGCGCPCGCGA |
C6M1 | CHO-K1 cells | Cy3-siRNA | 26682443 | 100 | Relative fluorescence (%) | nan | 4h | 37ºC | Flow cytometry | cellular uptake | Acetyl-RLWRLLWRLWRRLWRLLR-NH2 |
DM1 | CHO-K1 cells | Cy3-siRNA | 26682443 | 95 | Relative fluorescence (%) | nan | 4h | 37ºC | Flow cytometry | cellular uptake | DEG-RLWRLLWRLWRRLWRLLR-NH2 |
R1PECL | HeLa cells | nan | 27532744 | 1000 | Fluorescence intensity | nan | 24h | nan | Flow cytometry | cellular uptake | RC-PEG-b-PCL |
R4PECL | HeLa cells | nan | 27532744 | 2500 | Fluorescence intensity | nan | 24h | nan | Flow cytometry | cellular uptake | RRRRC-PEG-b-PCL |
R8PECL | HeLa cells | nan | 27532744 | 8000 | Fluorescence intensity | nan | 24h | nan | Flow cytometry | cellular uptake | RRRRRRRRC-PEG-b-PCL |
R7E7 | MDA-MB-231 cells | FITC | 30774914 | 40 | Intensity | 10uM | 10min | nan | Flow cytometry | cellular uptake | RRRRRRREEEEEEE |
R7E7 | MDA-MB-231 cells | FITC | 30774914 | 160 | Intensity | 50uM | 10min | nan | Flow cytometry | cellular uptake | RRRRRRREEEEEEE |
R7E7 | MDA-MB-231 cells | FITC | 30774914 | 200 | Intensity | 100uM | 10min | nan | Flow cytometry | cellular uptake | RRRRRRREEEEEEE |
P-01 | 293T cells | YOYO-1 | 35542475 | 2,20E+04 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-CLLHHLLHHLLHHC-RRRRRRRRR |
P-02 | 293T cells | YOYO-1 | 35542475 | 1,80E+04 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-cllhhllhhllhhc-rrrrrrrrr |
P-03 | 293T cells | YOYO-1 | 35542475 | 2,20E+04 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-CLLKKLLKKLLKKC-HHHHHH-RRRRRRRRR |
P-04 | 293T cells | YOYO-1 | 35542475 | 2,00E+04 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-cllkkllkkllkkc-hhhhhh-rrrrrrrrr |
P-05 | 293T cells | YOYO-1 | 35542475 | 1,80E+03 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-CLLHHLLHHLLHHC-GRKKRRQRRR |
P-06 | 293T cells | YOYO-1 | 35542475 | 1,70E+03 | Count | nan | 30min | 37ºC | FACS | cellular uptake | C18-cllhhllhhllhhc-grkkrrqrrr |
PLGA/R6LRVG | Caco-2 cells | FITC | 34239301 | 1500 | Mean Fluorescence intensity | 600 ug/ml | 3h | nan | Flow cytometry | cellular uptake | RRRRRRLRVG |
HPRP-A1 | A549 cells | FITC | 29396568 | 25 | Fluorescence intensity | 16uM | 100s | 37ºC | Flow cytometry | cellular uptake | Ac-FKKLKKLFSKLWNWK-NH2 |
HPRP-A1-iRGD | A549 cells | FITC | 29396568 | 35 | Fluorescence intensity | 16uM | 100s | 37ºC | Flow cytometry | cellular uptake | Ac-FKKLKKLFSKLWNWK-NH2-Ac-CRGDKGPDC-NH2 |
RCCNPs | HepG2 cells | nan | 34893294 | 8000 | Mean Fluorescence intensity | nan | 3h | 37ºC | Flow cytometry | cellular uptake | RRRRRRHHHH |
RCCNPs | HepG2 cells | nan | 34893294 | 11000 | Mean Fluorescence intensity | nan | 3h | 37ºC | Flow cytometry | cellular uptake | RRRRRRHHHH |
NFL-TBS.40-63 | J3T cells | LNC-(DiD) | 34144141 | 17 | Fluorescent cells (%) | 1 mg/ml | 12h | 37ºC | Flow cytometry | cellular uptake of LNC-(DiD) | YSSYSAPVSSSLSVRRSYSSSSGS |
R-NLC | A549 cells | Cou-6 | 32104313 | 3500 | Cou 6/protein /ug/mg) | 2ug/ml | 2h | nan | Flow cytometry | cellular uptake | RRRRRRRRNLC |
dNP2 | MDA-MB-231 cells | Cou-6-NLC | 33921919 | 2300 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | MDA-MB-231 cells | Cou-6-NLC | 33921919 | 2200 | Mean Fluorescence intensity | nan | 8h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | 4T1 cells | Cou-6-NLC | 33921919 | 2000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | 4T1 cells | Cou-6-NLC | 33921919 | 2200 | Mean Fluorescence intensity | nan | 8h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | MCF7 cells | Cou-6-NLC | 33921919 | 3000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
dNP2 | MCF7 cells | Cou-6-NLC | 33921919 | 3400 | Mean Fluorescence intensity | nan | 8h | 37ºC | Flow cytometry | cellular uptake | CKIKKVKKKGRKKIKKVKKKGRK |
tLyP-1-HFtn | MDA-MB-231 cells | FITC | 33568906 | 120 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGNKRTR |
M-tLyP-1-HFtn | MDA-MB-231 cells | FITC | 33568906 | 20 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGNARTA |
P7 | A549 cells | Carboxyfluorescein | 33995950 | 100 | Cell Fluorescence | 25uM | 90min | 37ºC | Flow cytometry | cellular uptake | COOH-RRRRRRRRRR-NH2 |
P8 | A549 cells | Carboxyfluorescein | 33995950 | 75 | Cell Fluorescence | 25uM | 90min | 37ºC | Flow cytometry | cellular uptake | COOH-KKKKKKKKKK-NH2 |
Pep-1 | U87 cells | PeCNL, Cou6 | 28672205 | 89.8 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | CGEMGWVRC |
Pep-1 | U87 cells | CNL, Cou6 | 28672205 | 47.5 | Cellular uptake (%) | nan | 2h | 37ºC | Flow cytometry | cellular uptake | CGEMGWVRC |
TAT-ASA-MNP-CDDP | HNE-1 cells | FITC | 30826059 | 1800 | Fluorescence intensity | 5ug/ml | 2h | nan | Flow cytometry | intracellular uptake | YGRKKRRQRRR |
TAT-ASA-MNP-CDDP | CNE-2 cells | FITC | 30826059 | 800 | Fluorescence intensity | 5ug/ml | 2h | nan | Flow cytometry | intracellular uptake | YGRKKRRQRRR |
IF-7 | A549 cells | CMNC | 31686810 | 5000 | Mean Fluorescence intensity | 100ug | 30min | 37ºC | Flow cytometry | cellular uptake | IFLLWQ |
IF-7 | A549 cells | CMNC | 31686810 | 10000 | Mean Fluorescence intensity | 100ug | 1h | 37ºC | Flow cytometry | cellular uptake | IFLLWQ |
IF-7 | A549 cells | CMNC | 31686810 | 16000 | Mean Fluorescence intensity | 100ug | 2h | 37ºC | Flow cytometry | cellular uptake | IFLLWQ |
IF-7 | A549 cells | CMNC | 31686810 | 17000 | Mean Fluorescence intensity | 100ug | 4h | 37ºC | Flow cytometry | cellular uptake | IFLLWQ |
PP1 | HUVEC cells | Cy5 | 30855618 | 1000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
PP1 | HUVEC cells | BCPs | 30855618 | 5000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
PP1 | HUVEC cells | TCPs-1 | 30855618 | 3800 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
PP1 | HUVEC cells | TCPs-2 | 30855618 | 3500 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
PP1 | HUVEC cells | TCPs-3 | 30855618 | 3000 | Mean Fluorescence intensity | nan | 4h | 37ºC | Flow cytometry | cellular uptake | CGPKKKRKVGYGRKKRRQRRR |
DP7-C | GL261 cells | siRNA | 34973309 | 130000 | Mean Fluorescence intensity | nan | 4h | nan | Flow cytometry | cellular uptake | VQWRIRVAVIRK |
DP7-C | GL261 cells | HA, siRNA | 34973309 | 140000 | Mean Fluorescence intensity | nan | 4h | nan | Flow cytometry | cellular uptake | VQWRIRVAVIRK |
GBP(L) | A549 cells | L-DOX | 32241176 | 1.1 | Cellular uptake | nan | 24h | 37ºC | Flow cytometry | cellular uptake | NYRWRCKN |
GBP(M) | A549 cells | L-DOX | 32241176 | 2.6 | Cellular uptake | nan | 24h | 37ºC | Flow cytometry | cellular uptake | NYRWRCKN |
GBP(H) | A549 cells | L-DOX | 32241176 | 5.7 | Cellular uptake | nan | 24h | 37ºC | Flow cytometry | cellular uptake | NYRWRCKN |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 42 | Mean Fluorescence intensity | 5uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 78 | Mean Fluorescence intensity | 10uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 100 | Mean Fluorescence intensity | 15uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 115 | Mean Fluorescence intensity | 20uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 120 | Mean Fluorescence intensity | 25uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
R8NLS | A2780 cells | P-GFLG-FITC | 26784985 | 130 | Mean Fluorescence intensity | 30uM | 1h | 37ºC | Flow cytometry | cellular uptake | CRRRRRRRRVKRKKKP |
LinTT1 | U87 cells | NW, FAM | 31255690 | 11 | Fluorescence | nan | 1h | 37ºC | Flow cytometry | cellular uptake of nanoworms | AKRGARSTA |
LinTT1 | NCH421K cells | NW, FAM | 31255690 | 4 | Fluorescence | nan | 1h | 37ºC | Flow cytometry | cellular uptake of nanoworms | AKRGARSTA |
NT4 | HT29 cells | QDs | 29501065 | 14000 | Mean Fluorescence intensity | 20uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
NT4 | HT29 cells | QDs | 29501065 | 9000 | Mean Fluorescence intensity | 10uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
NT4 | HT29 cells | QDs | 29501065 | 5000 | Mean Fluorescence intensity | 5uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
NT4 | HT29 cells | QDs | 29501065 | 1000 | Mean Fluorescence intensity | 1uM | 30min | 37ºC | Flow cytometry | QD internalization | ELYENKPRRPYIL |
P2 | HeLa cells | FITC-siRNA | 35575337 | 5000 | Relative fluorescence | nan | 6h | nan | Flow cytometry | cellular uptake | P(LAEMA37)-b-P(FPMA2-st-DMA2)-KRRKRRRRRK |
P3 | HeLa cells | FITC-siRNA | 35575337 | 4800 | Relative fluorescence | nan | 6h | nan | Flow cytometry | cellular uptake | P(LAEMA23-st-FPMA3)-KRRKRRRRRK |
P4 | HeLa cells | FITC-siRNA | 35575337 | 5500 | Relative fluorescence | nan | 6h | nan | Flow cytometry | cellular uptake | P(LAEMA25-st-FPMA2-st-DMA2)-KRRKRRRRRK |
L17E | HeLa cells | FITC | 35395514 | 100 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
L17ER2 | HeLa cells | FITC | 35395514 | 200 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GRRGK(FITC)-NH2 |
L17ER4 | HeLa cells | FITC | 35395514 | 900 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | cellular uptake | IWLTALKFLGKHAAKHEAKQQLSKL-GRRRRGK(FITC)-NH2 |
R2L17E | HeLa cells | FITC | 35395514 | 220 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | cellular uptake | RRG-IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
R4L17E | HeLa cells | FITC | 35395514 | 800 | Relative Cellular uptake | 6uM | 1h | 37ºC | Flow cytometry | cellular uptake | RRRRG-IWLTALKFLGKHAAKHEAKQQLSKL-GK(FITC)-NH2 |
JTS-1 | TF cells | FITC | 35601335 | 0 | nan | 1uM | 1h | nan | CLSM | peptide uptake | GLFEALLELLESLWELLLEA |
STRAP-1 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 500 | Mean Fluorescence intensity | 10uM | 4h | nan | Flow cytometry | cellular uptake | KrKiFcL |
STRAP-2 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 400 | Mean Fluorescence intensity | 10uM | 4h | nan | Flow cytometry | cellular uptake | kRkIfCl |
STRAP-3 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 800 | Mean Fluorescence intensity | 10uM | 4h | nan | Flow cytometry | cellular uptake | KrKfIcL |
STRAP-4 | MDA-MB-231 cells | Carboxyfluorescein | 35839086 | 2000 | Mean Fluorescence intensity | 10uM | 4h | nan | Flow cytometry | cellular uptake | kRkFiCl |
Oleyl-(HR)4 | MDA-MB-231 cells | siRNA-A488 | 35456715 | 10 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | HRHRHRHR |
Oleyl-R1-(HR)4 | MDA-MB-231 cells | siRNA-A489 | 35456715 | 50 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | RHRHRHRHR |
Oleyl-R2-(HR)4 | MDA-MB-231 cells | siRNA-A490 | 35456715 | 100 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | RRHRHRHRHR |
Oleyl-R3-(HR)4 | MDA-MB-231 cells | siRNA-A491 | 35456715 | 250 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | RRRHRHRHRHR |
Oleyl-R4-(HR)4 | MDA-MB-231 cells | siRNA-A492 | 35456715 | 400 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | RRRRHRHRHRHR |
Oleyl-R5-(HR)4 | MDA-MB-231 cells | siRNA-A493 | 35456715 | 500 | Mean Fluorescence intensity | 50nM | 24h | 37ºC | Flow cytometry | cellular internalization of oleyl | RRRRRHRHRHRHR |
CyLoP-1 | NIH-3T3 cells | Carboxyfluorescein | 35752142 | 7000 | corr. Fluorescence | 2.5uM | 18h | 37ºC | Flow cytometry | cellular internalization of oleyl | CRWRWKCCKK |
This second table lists the usable information to deploy Machine Learning approaches, such as the POSEIDON predictor. This comprises information on 1.263 peptide samples, as it had to undergo several steps of pre-processing that made the remaining samples unusable for the target purpose. This table informs on:
The values can be sorted by clicking the arrows near the column names. The global search box on top of the table can be used to query the whole table. Additionally, the search boxes on the footer of the table can be used to query the individual columns.
Cell line | PubmedID | Uptake | Conc. | Time | Raw sequence | Sequence |
---|---|---|---|---|---|---|
Cell line | PubmedID | Uptake | Conc. | Time | Raw sequence | Sequence |
A375 cells | 30240193 | 0.7 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
A375-R cells | 30240193 | 0.78 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
MSTO cells | 30240193 | 1.0 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
9L cells | 30240193 | 0.3 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
9L-R cells | 30240193 | 0.6 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
LN18 cells | 30240193 | 0.48 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
U87 cells | 30240193 | 1.26 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
A375 cells | 30240193 | 0.78 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
A375-R cells | 30240193 | 1.0 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
MSTO cells | 30240193 | 1.18 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
9L cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
9L-R cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
LN18 cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
U87 cells | 30240193 | 1.36 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
HeLa cells | 28183803 | 3.18 | 5.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
HeLa cells | 28183803 | 4.0 | 10.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
HeLa cells | 28183803 | 4.23 | 25.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
HeLa cells | 28183803 | 4.2 | 50.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
HeLa cells | 28183803 | 2.26 | 5.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
HeLa cells | 28183803 | 3.08 | 10.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
HeLa cells | 28183803 | 3.26 | 25.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
HeLa cells | 28183803 | 3.28 | 50.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
CHO-K1 cells | 28183803 | 3.08 | 5.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
CHO-K1 cells | 28183803 | 3.18 | 10.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
CHO-K1 cells | 28183803 | 4.0 | 25.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
CHO-K1 cells | 28183803 | 4.04 | 50.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
CHO-K1 cells | 28183803 | 2.23 | 5.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
CHO-K1 cells | 28183803 | 2.28 | 10.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
CHO-K1 cells | 28183803 | 3.04 | 25.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
CHO-K1 cells | 28183803 | 3.11 | 50.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
pgsA-745 cells | 28183803 | 3.15 | 5.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
pgsA-745 cells | 28183803 | 3.18 | 10.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
pgsA-745 cells | 28183803 | 0.21 | 25.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
pgsA-745 cells | 28183803 | 4.0 | 50.0 | 120.0 | MIASHLLAYFFTELNGKPILFF | MIASHLLAYFFTELNGKPILFF |
pgsA-745 cells | 28183803 | 2.11 | 5.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
pgsA-745 cells | 28183803 | 2.18 | 10.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
pgsA-745 cells | 28183803 | 2.26 | 25.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
pgsA-745 cells | 28183803 | 3.0 | 50.0 | 120.0 | MIASHLLAYFFTELN | MIASHLLAYFFTELN |
MCF7 cells | 32024261 | 3.04 | 2.5 | 60.0 | KARKKKLNKKGRKMAGRKRGRPKK | KARKKKLNKKGRKMAGRKRGRPKK |
MCF7 cells | 32024261 | 3.15 | 5.0 | 60.0 | KARKKKLNKKGRKMAGRKRGRPKK | KARKKKLNKKGRKMAGRKRGRPKK |
MCF7 cells | 32024261 | 3.16 | 7.5 | 60.0 | KARKKKLNKKGRKMAGRKRGRPKK | KARKKKLNKKGRKMAGRKRGRPKK |
MCF7 cells | 32024261 | 3.28 | 10.0 | 60.0 | KARKKKLNKKGRKMAGRKRGRPKK | KARKKKLNKKGRKMAGRKRGRPKK |
MCF7 cells | 32024261 | 2.3 | 2.5 | 60.0 | KALGISYGRKK | KALGISYGRKK |
MCF7 cells | 32024261 | 2.0 | 5.0 | 60.0 | KALGISYGRKK | KALGISYGRKK |
MCF7 cells | 32024261 | 2.48 | 7.5 | 60.0 | KALGISYGRKK | KALGISYGRKK |
MCF7 cells | 32024261 | 2.48 | 10.0 | 60.0 | KALGISYGRKK | KALGISYGRKK |
MCF-7 cells | 32116040 | 1.0 | 5.0 | 60.0 | RRWWWWRREEEEEEEEEEEE | RRWWWWRREEEEEEEEEEEE |
MCF-7 cells | 32116040 | 1.26 | 10.0 | 60.0 | RRWWWWRREEEEEEEEEEEE | RRWWWWRREEEEEEEEEEEE |
MCF-7 cells | 32116040 | 1.61 | 15.0 | 60.0 | RRWWWWRREEEEEEEEEEEE | RRWWWWRREEEEEEEEEEEE |
MCF-7 cells | 32116040 | 1.65 | 25.0 | 60.0 | RRWWWWRREEEEEEEEEEEE | RRWWWWRREEEEEEEEEEEE |
MCF-7 cells | 32116040 | 0.48 | 5.0 | 60.0 | WWWRRRRWWWEEEEEEEEEEEE | WWWRRRRWWWEEEEEEEEEEEE |
MCF-7 cells | 32116040 | 0.3 | 10.0 | 60.0 | WWWRRRRWWWEEEEEEEEEEEE | WWWRRRRWWWEEEEEEEEEEEE |
MCF-7 cells | 32116040 | 0.6 | 15.0 | 60.0 | WWWRRRRWWWEEEEEEEEEEEE | WWWRRRRWWWEEEEEEEEEEEE |
MCF-7 cells | 32116040 | 1.36 | 25.0 | 60.0 | WWWRRRRWWWEEEEEEEEEEEE | WWWRRRRWWWEEEEEEEEEEEE |
HeLa cells | 34101293 | 1.85 | 10.0 | 60.0 | YGRKKRRQRRR | YGRKKRRQRRR |
HeLa cells | 34101293 | 2.0 | 10.0 | 60.0 | YGRKKRRQRRR | YGRKKRRQRRR |
HeLa cells | 34101293 | 1.3 | 10.0 | 60.0 | PFVYLIPKKKRKVHHHHHHGC | PFVYLIPKKKRKVHHHHHHGC |
HeLa cells | 34101293 | 2.0 | 10.0 | 60.0 | PFVYLIPKKKRKVHHHHHHGC | PFVYLIPKKKRKVHHHHHHGC |
HepG2 cells | 29787814 | 0.0 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HepG2 cells | 29787814 | 2.06 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HepG2 cells | 29787814 | 2.24 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HepG2 cells | 29787814 | 1.93 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HepG2 cells | 29787814 | 1.0 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HepG2 cells | 29787814 | 2.0 | 5.0 | 1440.0 | GRKKRRQRRR | GRKKRRQRRR |
HEK-293T cell | 34277705 | 0.0 | 1.0 | 1440.0 | RRPPWLRLDIRR | RRPPWLRLDIRR |
HEK-293T cell | 34277705 | 0.7 | 5.0 | 1440.0 | RRPPWLRLDIRR | RRPPWLRLDIRR |
HEK-293T cell | 34277705 | 0.3 | 10.0 | 1440.0 | RRPPWLRLDIRR | RRPPWLRLDIRR |
HEK-293T cell | 34277705 | 1.6 | 1.0 | 1440.0 | RRRPPWLRLDIRRK | RRRPPWLRLDIRRK |
HEK-293T cell | 34277705 | 1.0 | 5.0 | 1440.0 | RRRPPWLRLDIRRK | RRRPPWLRLDIRRK |
HEK-293T cell | 34277705 | 2.08 | 10.0 | 1440.0 | RRRPPWLRLDIRRK | RRRPPWLRLDIRRK |
A549 cells | 28694765 | 1.54 | 10.0 | 90.0 | RWRWRWRWRW | RWRWRWRWRW |
A549 cells | 28694765 | 1.69 | 25.0 | 90.0 | RWRWRWRWRW | RWRWRWRWRW |
A549 cells | 28694765 | 1.83 | 50.0 | 90.0 | RWRWRWRWRW | RWRWRWRWRW |
CHO-K1 cells | 28512335 | 3.13 | 20.0 | 1440.0 | CGRRRR | CGRRRR |
CHO-K1 cells | 28512335 | 3.46 | 20.0 | 1440.0 | CGRRRRRRRR | CGRRRRRRRR |
CHO-K1 cells | 28512335 | 3.46 | 20.0 | 1440.0 | CGRRRRRRRRRRRR | CGRRRRRRRRRRRR |
CHO-K1 cells | 28512335 | 3.26 | 10.0 | 1440.0 | CGRRRRRRRRRRRRRRRR | CGRRRRRRRRRRRRRRRR |
D54 cells | 28140690 | 0.95 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
D54 cells | 28140690 | 1.57 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
D54 cells | 28140690 | 0.7 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
D54 cells | 28140690 | 0.9 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
U251 cells | 28140690 | 0.9 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
U251 cells | 28140690 | 1.38 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVVVVVGGGAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
U251 cells | 28140690 | 0.85 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
U251 cells | 28140690 | 1.0 | 30.0 | 60.0 | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH | RGGRLSYSRRRFSTSTGRVPGVGGGGGGGAAAAAAAAGLPRHSAVMERLRRRIELCRRHHSTCEARYEAVSPERLELERQHTFALHQRCIQAKAKRAGKH |
HCT 116 cells | 31073999 | 2.0 | 1.25 | 240.0 | NGVQPKYKWWKWWKKWW | NGVQPKYKWWKWWKKWW |
HCT 116 cells | 31073999 | 2.3 | 2.5 | 240.0 | NGVQPKYKWWKWWKKWW | NGVQPKYKWWKWWKKWW |
HCT 116 cells | 31073999 | 2.7 | 5.0 | 240.0 | NGVQPKYKWWKWWKKWW | NGVQPKYKWWKWWKKWW |
HCT 116 cells | 31073999 | 2.9 | 10.0 | 240.0 | NGVQPKYKWWKWWKKWW | NGVQPKYKWWKWWKKWW |
MCF7 cells | 33533253 | 1.0 | 2.0 | 60.0 | KRRRGGKKRRD | KRRRGGKKRRD |
MCF7 cells | 33533253 | 1.18 | 2.0 | 60.0 | KRRRRRRRRRRE | KRRRRRRRRRRE |
MCF7 cells | 33533253 | 1.4 | 2.0 | 60.0 | KRRRGGKKRRDLTFKEYWDQLTSAA | KRRRGGKKRRDLTFKEYWDQLTSAA |
MCF7 cells | 33533253 | 1.65 | 2.0 | 60.0 | KRRRRRRRRRRELTFKEYWDQLTSAA | KRRRRRRRRRRELTFKEYWDQLTSAA |
HeLa cells | 33533253 | 1.18 | 2.0 | 60.0 | KRRRGGKKRRD | KRRRGGKKRRD |
HeLa cells | 33533253 | 1.26 | 2.0 | 60.0 | KRRRRRRRRRRE | KRRRRRRRRRRE |
HeLa cells | 33533253 | 1.26 | 2.0 | 60.0 | KRRRGGKKRRDLTFKEYWDQLTSAA | KRRRGGKKRRDLTFKEYWDQLTSAA |
HeLa cells | 33533253 | 1.3 | 2.0 | 60.0 | KRRRRRRRRRRELTFKEYWDQLTSAA | KRRRRRRRRRRELTFKEYWDQLTSAA |
MCF7 cells | 33533253 | 0.0 | 2.0 | 120.0 | KRRRGGKKRRD | KRRRGGKKRRD |
MCF7 cells | 33533253 | 1.18 | 2.0 | 120.0 | KRRRRRRRRRRE | KRRRRRRRRRRE |
MCF7 cells | 33533253 | 0.0 | 2.0 | 120.0 | KRRRGGKKRRDLTFKEYWDQLTSAA | KRRRGGKKRRDLTFKEYWDQLTSAA |
MCF7 cells | 33533253 | 0.0 | 2.0 | 120.0 | KRRRRRRRRRRELTFKEYWDQLTSAA | KRRRRRRRRRRELTFKEYWDQLTSAA |
HeLa cells | 33533253 | 0.11 | 2.0 | 120.0 | KRRRGGKKRRD | KRRRGGKKRRD |
HeLa cells | 33533253 | 0.48 | 2.0 | 120.0 | KRRRRRRRRRRE | KRRRRRRRRRRE |
HeLa cells | 33533253 | -0.1 | 2.0 | 120.0 | KRRRGGKKRRDLTFKEYWDQLTSAA | KRRRGGKKRRDLTFKEYWDQLTSAA |
HeLa cells | 33533253 | 0.32 | 2.0 | 120.0 | KRRRRRRRRRRELTFKEYWDQLTSAA | KRRRRRRRRRRELTFKEYWDQLTSAA |
U87 cells | 31243977 | -0.4 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HT-29 cells | 31243977 | -0.42 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF7 cells | 31243977 | -0.52 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
U87 cells | 31243977 | 0.0 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HT-29 cells | 31243977 | -0.43 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF7 cells | 31243977 | -0.46 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
U87 cells | 31243977 | -0.1 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HT-29 cells | 31243977 | -0.12 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF7 cells | 31243977 | -0.4 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
U87 cells | 31243977 | 0.08 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HT-29 cells | 31243977 | -0.37 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF7 cells | 31243977 | -0.22 | 10.0 | 60.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34440250 | 2.0 | 0.025 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 2.0 | 0.025 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 2.48 | 0.025 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 2.0 | 0.05 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 2.48 | 0.05 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.0 | 0.05 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.0 | 0.1 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.18 | 0.1 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.4 | 0.1 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.74 | 0.2 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.78 | 0.2 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
HeLa cells | 34440250 | 3.85 | 0.2 | 240.0 | LAKLAKAAAKLLKAAAKAL | LAKLAKAAAKLLKAAAKAL |
A549 cells | 27074859 | 1.72 | 10.0 | 90.0 | RRRRRRRRREEEEEEEEE | RRRRRRRRREEEEEEEEE |
A549 cells | 27074859 | 1.74 | 10.0 | 90.0 | RRRRRWWWRRRREEEEEEEEE | RRRRRWWWRRRREEEEEEEEE |
A549 cells | 27074859 | 1.75 | 10.0 | 90.0 | RWRWRWRWRWRWEEEEEEEEE | RWRWRWRWRWRWEEEEEEEEE |
A549 cells | 27074859 | 1.86 | 25.0 | 90.0 | RRRRRRRRREEEEEEEEE | RRRRRRRRREEEEEEEEE |
A549 cells | 27074859 | 1.88 | 25.0 | 90.0 | RRRRRWWWRRRREEEEEEEEE | RRRRRWWWRRRREEEEEEEEE |
A549 cells | 27074859 | 1.89 | 25.0 | 90.0 | RWRWRWRWRWRWEEEEEEEEE | RWRWRWRWRWRWEEEEEEEEE |
A549 cells | 27074859 | 1.91 | 50.0 | 90.0 | RRRRRRRRREEEEEEEEE | RRRRRRRRREEEEEEEEE |
A549 cells | 27074859 | 1.93 | 50.0 | 90.0 | RRRRRWWWRRRREEEEEEEEE | RRRRRWWWRRRREEEEEEEEE |
A549 cells | 27074859 | 1.93 | 50.0 | 90.0 | RWRWRWRWRWRWEEEEEEEEE | RWRWRWRWRWRWEEEEEEEEE |
HeLa cells | 34032919 | 0.0 | 2.5 | 30.0 | RRRRRRK | RRRRRRK |
HeLa cells | 34032919 | 3.7 | 5.0 | 30.0 | RRRRRRK | RRRRRRK |
HeLa cells | 34032919 | 3.7 | 10.0 | 30.0 | RRRRRRK | RRRRRRK |
HeLa cells | 28051846 | 0.9 | 5.0 | 60.0 | GWWYKGRARPVSAVAK | GWWYKGRARPVSAVAK |
HeLa cells | 28051846 | 0.0 | 5.0 | 60.0 | GWWYKGRARPVSAVAK | GWWYKGRARPVSAVAK |
EJ cells | 29670331 | 0.0 | 0.25 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
EJ cells | 29670331 | 0.3 | 1.0 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
EJ cells | 29670331 | 0.7 | 2.5 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
EJ cells | 29670331 | 0.78 | 5.0 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
SV-HUC-1 cells | 29670331 | 0.0 | 0.25 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
SV-HUC-1 cells | 29670331 | 0.3 | 1.0 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
SV-HUC-1 cells | 29670331 | 0.7 | 2.5 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
SV-HUC-1 cells | 29670331 | 0.85 | 5.0 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
HeLa cells | 27966361 | 1.15 | 5.0 | 30.0 | MIILIIGSTSRDHMVLHEYVNAAGIT | MIILIIGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.6 | 5.0 | 30.0 | FLLIRRVLGSTSRDHMVLHEYVNAAGIT | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.48 | 5.0 | 30.0 | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.48 | 5.0 | 30.0 | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.85 | 5.0 | 30.0 | FIDLKRKIWLIK | FIDLKRKIWLIK |
HeLa cells | 27966361 | 0.7 | 5.0 | 30.0 | YLKFIPLKDAIWKIK | YLKFIPLKDAIWKIK |
HeLa cells | 27966361 | 0.0 | 2.0 | 30.0 | MIILIIGSTSRDHMVLHEYVNAAGIT | MIILIIGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.0 | 2.0 | 30.0 | FLLIRRVLGSTSRDHMVLHEYVNAAGIT | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.0 | 2.0 | 30.0 | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.0 | 2.0 | 30.0 | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.78 | 2.0 | 30.0 | FIDLKRKIWLIK | FIDLKRKIWLIK |
HeLa cells | 27966361 | 0.85 | 2.0 | 30.0 | YLKFIPLKDAIWKIK | YLKFIPLKDAIWKIK |
HeLa cells | 27966361 | 1.11 | 2.0 | 120.0 | MIILIIGSTSRDHMVLHEYVNAAGIT | MIILIIGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.6 | 2.0 | 120.0 | FLLIRRVLGSTSRDHMVLHEYVNAAGIT | FLLIRRVLGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.85 | 2.0 | 120.0 | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT | PWPRVPWRWGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.6 | 2.0 | 120.0 | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT | LKRAIWLIKGSTSRDHMVLHEYVNAAGIT |
HeLa cells | 27966361 | 0.0 | 2.0 | 120.0 | FIDLKRKIWLIK | FIDLKRKIWLIK |
HeLa cells | 27966361 | 0.0 | 2.0 | 120.0 | YLKFIPLKDAIWKIK | YLKFIPLKDAIWKIK |
HeLa cells | 27966361 | 0.48 | 2.0 | 120.0 | KIIIIDGSTSRDHLVLHEYVNAAGITA | KIIIIDGSTSRDHLVLHEYVNAAGITA |
HeLa cells | 27966361 | 0.6 | 2.0 | 120.0 | KLIILIIDGSTSRDHLVLHEYVNAAGITA | KLIILIIDGSTSRDHLVLHEYVNAAGITA |
HeLa cells | 27966361 | 1.2 | 2.0 | 120.0 | LIILIIGSTSRDHLVLHEYVNAAGITA | LIILIIGSTSRDHLVLHEYVNAAGITA |
HeLa cells | 27966361 | 0.7 | 2.0 | 120.0 | MIILIIGSTSRDHLVLHEYVNAAGITA | MIILIIGSTSRDHLVLHEYVNAAGITA |
HeLa cells | 27966361 | 0.95 | 2.0 | 120.0 | MIILIIMGVADLIKKFESISKEE | MIILIIMGVADLIKKFESISKEE |
HeLa cells | 27966361 | 1.18 | 2.0 | 120.0 | PLILLRLLRGSTSRDHLVLHEYVNAAGITA | PLILLRLLRGSTSRDHLVLHEYVNAAGITA |
HeLa cells | 27966361 | 1.54 | 2.0 | 120.0 | FIDIIIKILLIGSTSRDHLVLHEYVNAAGITA | FIDIIIKILLIGSTSRDHLVLHEYVNAAGITA |
MonoMac6 cells | 30099595 | 3.7 | 10.0 | 120.0 | TKPKGTKPKGTKPKGTKPKG | TKPKGTKPKGTKPKGTKPKG |
MonoMac6 cells | 30099595 | 4.18 | 10.0 | 120.0 | YKQCHKKGGKKGSG | YKQCHKKGGKKGSG |
MonoMac6 cells | 30099595 | 5.15 | 10.0 | 120.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
MonoMac6 cells | 30099595 | 4.6 | 10.0 | 120.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
MonoMac6 cells | 30099595 | 4.0 | 10.0 | 120.0 | GIGKFLHSAKKFGKAFVGEIMNS | GIGKFLHSAKKFGKAFVGEIMNS |
MonoMac6 cells | 30099595 | 5.24 | 10.0 | 120.0 | GIGAVLKVLTTGLPALISWIKRKRQQ | GIGAVLKVLTTGLPALISWIKRKRQQ |
HEK293 cells | 30893557 | 3.15 | 40.0 | 45.0 | FFLIGFFLIGRRRRRRRRRRRR | FFLIGFFLIGRRRRRRRRRRRR |
HeLa cells | 33355559 | 2.32 | 2.0 | 120.0 | AGRKARRQRRR | AGRKARRQRRR |
HeLa cells | 33355559 | 2.34 | 2.0 | 120.0 | AGRKKRRARRR | AGRKKRRARRR |
HeLa cells | 33355559 | 2.61 | 2.0 | 120.0 | YGRKARRQARR | YGRKARRQARR |
HeLa cells | 33355559 | 2.57 | 2.0 | 120.0 | YGRAARRQARA | YGRAARRQARA |
HeLa cells | 33355559 | 2.08 | 2.0 | 120.0 | YGRAARRQARA | YGRAARRQARA |
HeLa cells | 33355559 | 1.4 | 2.0 | 120.0 | YGRAAARQARA | YGRAAARQARA |
HeLa cells | 33355559 | 2.3 | 2.0 | 120.0 | YGRKARRQARR | YGRKARRQARR |
HeLa cells | 33355559 | 2.0 | 2.0 | 120.0 | YGRKARRQRR | YGRKARRQRR |
HeLa cells | 33355559 | 1.95 | 2.0 | 120.0 | YGRKARRQRR | YGRKARRQRR |
HeLa cells | 33355559 | 1.9 | 2.0 | 120.0 | AGRRKKRRARRR | AGRRKKRRARRR |
HeLa cells | 33355559 | 2.0 | 2.0 | 120.0 | YGRKARRQARR | YGRKARRQARR |
HeLa cells | 33355559 | 1.95 | 2.0 | 120.0 | YGRAARRQARR | YGRAARRQARR |
HaCaT cells | 30389988 | 3.15 | 10.0 | 30.0 | KCVRQNNKRVCKGLRKRLRKFRNK | KCVRQNNKRVCKGLRKRLRKFRNK |
MCF-7 cells | 28332260 | 1.59 | 25.0 | 30.0 | FLRKRLRKFRNKIKEK | FLRKRLRKFRNKIKEK |
MCF-7 cells | 28332260 | 1.6 | 25.0 | 30.0 | AGLRKAAARLRKFRNKAAAIKEK | AGLRKAAARLRKFRNKAAAIKEK |
MCF-7 cells | 28332260 | 2.11 | 50.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF-7 cells | 28332260 | 2.18 | 50.0 | 30.0 | AGLRKAAARLRKFRNKAAAIKEK | AGLRKAAARLRKFRNKAAAIKEK |
HEK-293 T-cell | 27516189 | 1.76 | 20.0 | 240.0 | KETWWETWWTEWSQPKKKRKV | KETWWETWWTEWSQPKKKRKV |
HEK-293 T-cell | 27516189 | 1.77 | 20.0 | 240.0 | GLWWRLWWRLRSWFRLWFRA | GLWWRLWWRLRSWFRLWFRA |
RAW264.7 cells | 30095906 | 1.98 | 5.0 | 120.0 | YGRKKRRQRRRCAGFAWNVCVYRNGVRVCHRRAN | YGRKKRRQRRRCAGFAWNVCVYRNGVRVCHRRAN |
RAW264.7 cells | 30095906 | 1.88 | 5.0 | 120.0 | GFAWNVCVYRNGVRVCHRRAN | GFAWNVCVYRNGVRVCHRRAN |
HeLa cells | 34333729 | 2.0 | 10.0 | 240.0 | RADPAYQARFLGKRKFICL | RADPAYQARFLGKRKFICL |
HeLa cells | 34333729 | 2.0 | 10.0 | 240.0 | KRKFICLGRADPAYQARFL | KRKFICLGRADPAYQARFL |
HeLa cells | 33838611 | 2.74 | 2.0 | 120.0 | GRRARRARRA | GRRARRARRA |
HeLa cells | 33838611 | 2.6 | 2.0 | 120.0 | GRRARRARRA | GRRARRARRA |
HeLa cells | 33838611 | 3.41 | 2.0 | 120.0 | GRRRRRRRRR | GRRRRRRRRR |
HEK293 cells | 33838611 | 2.04 | 2.0 | 120.0 | GRRARRARRA | GRRARRARRA |
HEK293 cells | 33838611 | 3.08 | 2.0 | 120.0 | GRRARRARRA | GRRARRARRA |
HEK293 cells | 33838611 | 3.45 | 2.0 | 120.0 | GRRRRRRRRR | GRRRRRRRRR |
A549 cells | 27480031 | 1.95 | 2.5 | 480.0 | KLALKLALKALKAALKLAGCRGDFC | KLALKLALKALKAALKLAGCRGDFC |
A549 cells | 27480031 | 1.7 | 2.5 | 480.0 | KLALKLALKALKAALKLAGCA | KLALKLALKALKAALKLAGCA |
A549 cells | 27480031 | 1.3 | 2.5 | 480.0 | KLALKLALKALKACRGDFCLKLAG | KLALKLALKALKACRGDFCLKLAG |
A549 cells | 27480031 | 1.96 | 2.5 | 480.0 | KCRGDFCALKLALKALKACRGDFCLKLAG | KCRGDFCALKLALKALKACRGDFCLKLAG |
A549 cells | 27480031 | 0.7 | 2.5 | 480.0 | KLALKLACRGDFCKALKACRGDFCLKLAG | KLALKLACRGDFCKALKACRGDFCLKLAG |
A549 cells | 27480031 | 1.18 | 2.5 | 480.0 | KCRGDFCALKLACRGDFCKALKACRGDFCLKLAG | KCRGDFCALKLACRGDFCKALKACRGDFCLKLAG |
HeLa cells | 26814673 | 1.95 | 1.0 | 120.0 | AGKKKKKKKKK | AGKKKKKKKKK |
HeLa cells | 26814673 | 2.7 | 1.0 | 120.0 | AGRRRRRRRRR | AGRRRRRRRRR |
HeLa cells | 26814673 | 1.0 | 1.0 | 120.0 | AGKKKKKKKKK | AGKKKKKKKKK |
HeLa cells | 26814673 | 2.3 | 1.0 | 120.0 | AGKKKKKKKKK | AGKKKKKKKKK |
A549 cells | 28835794 | 4.18 | 15.0 | 30.0 | AGGPPGPPGPPGPPGPPGPPGPPGPPGRRGRRG | AGGPPGPPGPPGPPGPPGPPGPPGPPGRRGRRG |
A549 cells | 28835794 | 4.38 | 30.0 | 30.0 | AGGPPGPPGPPGPPGPPGPPGPPGPPGRRGRRG | AGGPPGPPGPPGPPGPPGPPGPPGPPGRRGRRG |
HeLa cells | 28603674 | 3.2 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.23 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.44 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.19 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.2 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.28 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.08 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.04 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.35 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.24 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.18 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.35 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.34 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.45 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 28603674 | 3.4 | 5.0 | 60.0 | AGYLLGHINLHHLAHLAHHIL | AGYLLGHINLHHLAHLAHHIL |
HeLa cells | 31061420 | 1.7 | 5.0 | 60.0 | CPRILMRCKQDSDCLAGCVCGPNGFCG | CPRILMRCKQDSDCLAGCVCGPNGFCG |
HeLa cells | 31061420 | 1.6 | 5.0 | 60.0 | CPRILMRCKQDSDCLAGCVCGPNGFCG | CPRILMRCKQDSDCLAGCVCGPNGFCG |
BCECs cells | 32674358 | -1.3 | 100.0 | 180.0 | YGRKKRRQRRRNIETDVIETDV | YGRKKRRQRRRNIETDVIETDV |
HEK293 cells | 28921993 | 0.9 | 2.0 | 240.0 | QQRKRKIWSILAPLGTTLVKLVAGIG | QQRKRKIWSILAPLGTTLVKLVAGIG |
HEK293 cells | 28921993 | 1.0 | 2.0 | 240.0 | PLILLRLLRGQF | PLILLRLLRGQF |
HEK293 cells | 28921993 | 0.0 | 2.0 | 240.0 | AAVLLPVLLAAP | AAVLLPVLLAAP |
HEK293 cells | 28921993 | 1.3 | 2.0 | 240.0 | KLALKALKALKAALKLA | KLALKALKALKAALKLA |
HEK293 cells | 28921993 | 0.7 | 2.0 | 240.0 | QQRKRKIWSKLAPDGTTLVKLVAGIG | QQRKRKIWSKLAPDGTTLVKLVAGIG |
HEK293 cells | 28921993 | 0.3 | 2.0 | 240.0 | PLIKLRLDRGQF | PLIKLRLDRGQF |
HEK293 cells | 28921993 | 0.0 | 2.0 | 240.0 | AAKLLPDLLAAP | AAKLLPDLLAAP |
HEK293 cells | 28921993 | 1.26 | 2.0 | 240.0 | KLALKALKKLKADLKLA | KLALKALKKLKADLKLA |
HeLa cells | 28921993 | 1.3 | 2.0 | 240.0 | QQRKRKIWSILAPLGTTLVKLVAGIG | QQRKRKIWSILAPLGTTLVKLVAGIG |
HeLa cells | 28921993 | 1.0 | 2.0 | 240.0 | PLILLRLLRGQF | PLILLRLLRGQF |
HeLa cells | 28921993 | 0.0 | 2.0 | 240.0 | AAVLLPVLLAAP | AAVLLPVLLAAP |
HeLa cells | 28921993 | 1.4 | 2.0 | 240.0 | KLALKALKALKAALKLA | KLALKALKALKAALKLA |
HeLa cells | 28921993 | 0.48 | 2.0 | 240.0 | QQRKRKIWSKLAPDGTTLVKLVAGIG | QQRKRKIWSKLAPDGTTLVKLVAGIG |
HeLa cells | 28921993 | 0.3 | 2.0 | 240.0 | PLIKLRLDRGQF | PLIKLRLDRGQF |
HeLa cells | 28921993 | 0.0 | 2.0 | 240.0 | AAKLLPDLLAAP | AAKLLPDLLAAP |
HeLa cells | 28921993 | 1.18 | 2.0 | 240.0 | KLALKALKKLKADLKLA | KLALKALKKLKADLKLA |
A549 cells | 29396568 | 1.4 | 16.0 | 1.66666666666666 | FKKLKKLFSKLWNWK | FKKLKKLFSKLWNWK |
A549 cells | 29396568 | 1.54 | 16.0 | 1.66666666666666 | FKKLKKLFSKLWNWKCRGDKGPDC | FKKLKKLFSKLWNWKCRGDKGPDC |
A549 cells | 33995950 | 2.0 | 25.0 | 90.0 | RRRRRRRRRR | RRRRRRRRRR |
A549 cells | 33995950 | 1.88 | 25.0 | 90.0 | KKKKKKKKKK | KKKKKKKKKK |
HeLa cells | 35395514 | 2.0 | 6.0 | 60.0 | IWLTALKFLGKHAAKHEAKQQLSKLGK | IWLTALKFLGKHAAKHEAKQQLSKLGK |
HeLa cells | 35395514 | 2.3 | 6.0 | 60.0 | IWLTALKFLGKHAAKHEAKQQLSKLGRRGK | IWLTALKFLGKHAAKHEAKQQLSKLGRRGK |
HeLa cells | 35395514 | 2.95 | 6.0 | 60.0 | IWLTALKFLGKHAAKHEAKQQLSKLGRRRRGK | IWLTALKFLGKHAAKHEAKQQLSKLGRRRRGK |
HeLa cells | 35395514 | 2.34 | 6.0 | 60.0 | RRGIWLTALKFLGKHAAKHEAKQQLSKLGK | RRGIWLTALKFLGKHAAKHEAKQQLSKLGK |
HeLa cells | 35395514 | 2.9 | 6.0 | 60.0 | RRRRGIWLTALKFLGKHAAKHEAKQQLSKLGK | RRRRGIWLTALKFLGKHAAKHEAKQQLSKLGK |
MDA-MB-231 cells | 35456715 | 1.0 | 0.05 | 1440.0 | HRHRHRHR | HRHRHRHR |
MDA-MB-231 cells | 35456715 | 1.7 | 0.05 | 1440.0 | RHRHRHRHR | RHRHRHRHR |
MDA-MB-231 cells | 35456715 | 2.0 | 0.05 | 1440.0 | RRHRHRHRHR | RRHRHRHRHR |
MDA-MB-231 cells | 35456715 | 2.4 | 0.05 | 1440.0 | RRRHRHRHRHR | RRRHRHRHRHR |
MDA-MB-231 cells | 35456715 | 2.6 | 0.05 | 1440.0 | RRRRHRHRHRHR | RRRRHRHRHRHR |
MDA-MB-231 cells | 35456715 | 2.7 | 0.05 | 1440.0 | RRRRRHRHRHRHR | RRRRRHRHRHRHR |
Jurkat | 11087855 | 2.81 | 12.5 | 15.0 | RKKRRQRRR | RKKRRQRRR |
Jurkat | 11087855 | 1.49 | 12.5 | 10.0 | RKKRRQRR | RKKRRQRR |
Jurkat | 11087855 | 1.0 | 12.5 | 10.0 | RKKRRQR | RKKRRQR |
Jurkat | 11087855 | 1.35 | 12.5 | 10.0 | KKRRQRRR | KKRRQRRR |
Jurkat | 11087855 | 1.3 | 12.5 | 10.0 | KRRQRRR | KRRQRRR |
Jurkat | 11087855 | 3.39 | 12.5 | 15.0 | RRRQRRKKR | RRRQRRKKR |
Jurkat | 11087855 | 1.21 | 12.5 | 10.0 | AKKRRQRRR | AKKRRQRRR |
Jurkat | 11087855 | 1.51 | 12.5 | 10.0 | RAKRRQRRR | RAKRRQRRR |
Jurkat | 11087855 | 1.57 | 12.5 | 10.0 | RKARRQRRR | RKARRQRRR |
Jurkat | 11087855 | 1.3 | 12.5 | 10.0 | RKKARQRRR | RKKARQRRR |
Jurkat | 11087855 | 1.48 | 12.5 | 10.0 | RKKRAQRRR | RKKRAQRRR |
Jurkat | 11087855 | 2.12 | 12.5 | 10.0 | RKKRRARRR | RKKRRARRR |
Jurkat | 11087855 | 1.51 | 12.5 | 10.0 | RKKRRQARR | RKKRRQARR |
Jurkat | 11087855 | 1.54 | 12.5 | 10.0 | RKKRRQRAR | RKKRRQRAR |
Jurkat | 11087855 | 1.1 | 12.5 | 10.0 | RKKRRQRRA | RKKRRQRRA |
Jurkat | 11087855 | 2.0 | 12.5 | 15.0 | RRRRR | RRRRR |
Jurkat | 11087855 | 2.7 | 12.5 | 15.0 | RRRRRR | RRRRRR |
Jurkat | 11087855 | 3.09 | 12.5 | 15.0 | RRRRRRR | RRRRRRR |
Jurkat | 11087855 | 3.23 | 12.5 | 15.0 | RRRRRRRR | RRRRRRRR |
Jurkat | 11087855 | 3.42 | 12.5 | 15.0 | RRRRRRRRR | RRRRRRRRR |
NIH-3T3 | 21319732 | 3.5 | 2.5 | 1080.0 | KMDCRWRWKCCKK | KMDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.52 | 2.5 | 1080.0 | MDCRWRWKCCKK | MDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.28 | 2.5 | 1080.0 | DCRWRWKCCKK | DCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.61 | 2.5 | 1080.0 | CRWRWKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.18 | 2.5 | 1080.0 | RWRWKCCKK | RWRWKCCKK |
NIH-3T3 | 21319732 | 3.18 | 2.5 | 1080.0 | KMDCRWRWKCKK | KMDCRWRWKCKK |
NIH-3T3 | 21319732 | 3.08 | 2.5 | 1080.0 | KMDCRWRWKKK | KMDCRWRWKKK |
NIH-3T3 | 21319732 | 2.0 | 2.5 | 1080.0 | KMDRWRWKKK | KMDRWRWKKK |
NIH-3T3 | 21319732 | 3.02 | 2.5 | 1080.0 | KDCRWRWKCCKK | KDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.2 | 2.5 | 1080.0 | KCRWRWKCCKK | KCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.09 | 2.5 | 1080.0 | KRWRWKCCKK | KRWRWKCCKK |
NIH-3T3 | 21319732 | 3.34 | 2.5 | 1080.0 | CRWRWKCSKK | CRWRWKCSKK |
NIH-3T3 | 21319732 | 3.27 | 2.5 | 1080.0 | SRWRWKCCKK | SRWRWKCCKK |
NIH-3T3 | 21319732 | 2.76 | 2.5 | 1080.0 | SRWRWKCSKK | SRWRWKCSKK |
NIH-3T3 | 21319732 | 2.68 | 2.5 | 1080.0 | SRWRWKSCKK | SRWRWKSCKK |
NIH-3T3 | 21319732 | 2.62 | 2.5 | 1080.0 | CRWRWKSSKK | CRWRWKSSKK |
NIH-3T3 | 21319732 | 2.29 | 2.5 | 1080.0 | SRWRWKSSKK | SRWRWKSSKK |
NIH-3T3 | 21319732 | 3.42 | 2.5 | 1080.0 | CRFRWKCCKK | CRFRWKCCKK |
NIH-3T3 | 21319732 | 3.39 | 2.5 | 1080.0 | CRWRFKCCKK | CRWRFKCCKK |
NIH-3T3 | 21319732 | 3.41 | 2.5 | 1080.0 | CRFRFKCCKK | CRFRFKCCKK |
NIH-3T3 | 21319732 | 3.23 | 2.5 | 1080.0 | KCCKWRWRCK | KCCKWRWRCK |
NIH-3T3 | 21319732 | 3.38 | 2.5 | 1080.0 | CRWRWKCGCKK | CRWRWKCGCKK |
NIH-3T3 | 21319732 | 3.49 | 2.5 | 1080.0 | KCGCRWRWKCGCKK | KCGCRWRWKCGCKK |
NIH-3T3 | 21319732 | 3.28 | 2.5 | 1080.0 | CRWRWKCG | CRWRWKCG |
NIH-3T3 | 21319732 | 3.37 | 2.5 | 1080.0 | KMDCRWRWKCSKK | KMDCRWRWKCSKK |
NIH-3T3 | 21319732 | 3.07 | 2.5 | 1080.0 | KMDCRWRWKSCKK | KMDCRWRWKSCKK |
NIH-3T3 | 21319732 | 2.99 | 2.5 | 1080.0 | KMDSRWRWKCCKK | KMDSRWRWKCCKK |
NIH-3T3 | 21319732 | 2.79 | 2.5 | 1080.0 | KMDCRWRWKSSKK | KMDCRWRWKSSKK |
NIH-3T3 | 21319732 | 2.7 | 2.5 | 1080.0 | KMDSRWRWKSSKK | KMDSRWRWKSSKK |
NIH-3T3 | 21319732 | 2.93 | 2.5 | 1080.0 | KMDSRWRWKSCKK | KMDSRWRWKSCKK |
NIH-3T3 | 21319732 | 3.09 | 2.5 | 1080.0 | KMDSRWRWKCSKK | KMDSRWRWKCSKK |
NIH-3T3 | 21319732 | 3.1 | 2.5 | 1080.0 | KMDCRWRPKCCKK | KMDCRWRPKCCKK |
NIH-3T3 | 21319732 | 2.54 | 2.5 | 1080.0 | KMDCRPRPKCCKK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 1.44 | 2.5 | 1080.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
HeLa | 21359136 | 3.11 | 1600.0 | 180.0 | VPTLK | VPTLK |
CHO | 19956900 | 2.9 | 50.0 | 60.0 | KLWMRWYSPTTRRYG | KLWMRWYSPTTRRYG |
CHO | 19956900 | 2.81 | 50.0 | 60.0 | RLWMRWYSPTTRRYG | RLWMRWYSPTTRRYG |
CHO | 19956900 | 2.9 | 50.0 | 60.0 | KLWMRWYSATTRRYG | KLWMRWYSATTRRYG |
CHO | 19956900 | 2.93 | 50.0 | 60.0 | KLWMRWYSPWTRRYG | KLWMRWYSPWTRRYG |
CHO | 19956900 | 2.81 | 50.0 | 60.0 | RLWMRWYSPWTRRYG | RLWMRWYSPWTRRYG |
CHO | 19956900 | 2.72 | 50.0 | 60.0 | RLWMRWYSPWTRRWG | RLWMRWYSPWTRRWG |
CHO | 19956900 | 2.34 | 50.0 | 60.0 | ALWMRWYSPTTRRYG | ALWMRWYSPTTRRYG |
CHO | 19956900 | 2.9 | 50.0 | 60.0 | RAWMRWYSPTTRRYG | RAWMRWYSPTTRRYG |
CHO | 19956900 | 2.88 | 50.0 | 60.0 | RLAMRWYSPTTRRYG | RLAMRWYSPTTRRYG |
CHO | 19956900 | 2.88 | 50.0 | 60.0 | RLWARWYSPTTRRYG | RLWARWYSPTTRRYG |
CHO | 19956900 | 1.95 | 50.0 | 60.0 | RLWMAWYSPTTRRYG | RLWMAWYSPTTRRYG |
CHO | 19956900 | 1.7 | 50.0 | 60.0 | RLWMRAYSPTTRRYG | RLWMRAYSPTTRRYG |
CHO | 19956900 | 2.9 | 50.0 | 60.0 | RLWMRWASPTTRRYG | RLWMRWASPTTRRYG |
CHO | 19956900 | 2.9 | 50.0 | 60.0 | RLWMRWYAPTTRRYG | RLWMRWYAPTTRRYG |
CHO | 19956900 | 2.94 | 50.0 | 60.0 | RLWMRWYSPATRRYG | RLWMRWYSPATRRYG |
CHO | 19956900 | 2.91 | 50.0 | 60.0 | RLWMRWYSPTARRYG | RLWMRWYSPTARRYG |
CHO | 19956900 | 2.57 | 50.0 | 60.0 | RLWMRWYSPTTARYG | RLWMRWYSPTTARYG |
CHO | 19956900 | 2.18 | 50.0 | 60.0 | RLWMRWYSPTTRAYG | RLWMRWYSPTTRAYG |
CHO | 19956900 | 2.92 | 50.0 | 60.0 | RLWMRWYSPTTRRAG | RLWMRWYSPTTRRAG |
CHO | 19956900 | 2.93 | 50.0 | 60.0 | RLWMRWYSPTTRRYA | RLWMRWYSPTTRRYA |
CHO | 19956900 | 2.64 | 50.0 | 60.0 | RLLMRLYSPTTRRYG | RLLMRLYSPTTRRYG |
CHO | 19956900 | 2.92 | 50.0 | 60.0 | RLFMRFYSPTTRRYG | RLFMRFYSPTTRRYG |
CHO | 19956900 | 2.93 | 50.0 | 60.0 | RLIMRIYSPTTRRYG | RLIMRIYSPTTRRYG |
CHO | 19956900 | 2.77 | 50.0 | 60.0 | RLVMRVYSPTTRRYG | RLVMRVYSPTTRRYG |
CHO | 19956900 | 2.95 | 50.0 | 60.0 | RLYMRYYSPTTRRYG | RLYMRYYSPTTRRYG |
RAW 264.7 | 12450378 | 1.95 | 5.0 | 30.0 | RRIRPRP | RRIRPRP |
RAW 264.7 | 12450378 | 2.3 | 5.0 | 30.0 | RRIRPRPPRLPRPRP | RRIRPRPPRLPRPRP |
RAW 264.7 | 12450378 | 1.54 | 5.0 | 30.0 | RRIRPRPPRLPRPRPRPLPFPRPG | RRIRPRPPRLPRPRPRPLPFPRPG |
RAW 264.7 | 12450378 | 2.11 | 5.0 | 30.0 | RRIRPRPPRLPRPRPRP | RRIRPRPPRLPRPRPRP |
RAW 264.7 | 12450378 | 1.78 | 5.0 | 30.0 | PRPPRLPRPRPRPLPFPRPG | PRPPRLPRPRPRPLPFPRPG |
RAW 264.7 | 12450378 | 1.95 | 5.0 | 30.0 | PPRLPRPRPRPLPFPRPG | PPRLPRPRPRPLPFPRPG |
RAW 264.7 | 12450378 | 2.0 | 5.0 | 30.0 | RLPRPRPRPLPFPRPG | RLPRPRPRPLPFPRPG |
RAW 264.7 | 12450378 | 1.9 | 5.0 | 30.0 | PRPRPLPFPRPG | PRPRPLPFPRPG |
RAW 264.7 | 12450378 | 2.74 | 5.0 | 30.0 | PRPLPFPRPG | PRPLPFPRPG |
U373MG cells | 20659686 | 2.0 | 5.0 | 60.0 | GTKMIFVGIKKKEERADLIAYLKKA | GTKMIFVGIKKKEERADLIAYLKKA |
U373MG cells | 20659686 | 0.6 | 5.0 | 60.0 | KKKEERADLIAYLKKA | KKKEERADLIAYLKKA |
U373MG cells | 20659686 | 0.9 | 5.0 | 60.0 | KMIFVGIKKKEERA | KMIFVGIKKKEERA |
U373MG cells | 20659686 | 0.65 | 5.0 | 60.0 | KMIFVGIKKK | KMIFVGIKKK |
U373MG cells | 20659686 | 0.85 | 5.0 | 60.0 | EKGKKIFIMK | EKGKKIFIMK |
U373MG cells | 20659686 | 1.61 | 5.0 | 60.0 | KGKKIFIMK | KGKKIFIMK |
HeLa | 19858187 | 1.6 | 10.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 19858187 | 1.53 | 10.0 | 30.0 | KCFQWQRNMRKVRGPPVSC | KCFQWQRNMRKVRGPPVSC |
HeLa | 19858187 | 0.88 | 10.0 | 30.0 | KCFQWQRNMRKVRGPPVSSIKR | KCFQWQRNMRKVRGPPVSSIKR |
HeLa | 19858187 | 0.8 | 10.0 | 30.0 | KCFQWQRNMRKVR | KCFQWQRNMRKVR |
HeLa | 19858187 | 0.64 | 10.0 | 30.0 | FQWQRNMRKVRGPPVS | FQWQRNMRKVRGPPVS |
HeLa | 19858187 | 0.88 | 10.0 | 30.0 | QWQRNMRKVRGPPVSCIKR | QWQRNMRKVRGPPVSCIKR |
HeLa | 19858187 | 0.57 | 10.0 | 30.0 | QWQRNMRKVR | QWQRNMRKVR |
HeLa | 21365733 | 1.05 | 50.0 | 180.0 | VELPPPVELPPPVELPPP | VELPPPVELPPPVELPPP |
A549 | 21365733 | 0.7 | 50.0 | 180.0 | VELPPPVELPPPVELPPP | VELPPPVELPPPVELPPP |
DU-145 | 21029412 | 2.78 | 300.0 | 240.0 | EEEAAGRKRKKRT | EEEAAGRKRKKRT |
DU-145 | 21029412 | 2.15 | 300.0 | 240.0 | EEE | EEE |
DU-145 | 21029412 | 2.08 | 300.0 | 240.0 | EEEAA | EEEAA |
DU-145 | 21029412 | 2.45 | 300.0 | 240.0 | EEEAAKKK | EEEAAKKK |
DU-145 | 21029412 | 2.76 | 300.0 | 240.0 | GRKRKKRT | GRKRKKRT |
DU-145 | 21029412 | 2.0 | 300.0 | 60.0 | FFFAAGRKRKKRT | FFFAAGRKRKKRT |
DU-145 | 21029412 | 1.74 | 300.0 | 60.0 | NNNAAGRKRKKRT | NNNAAGRKRKKRT |
DU-145 | 21029412 | 2.06 | 300.0 | 60.0 | YYYAAGRKRKKRT | YYYAAGRKRKKRT |
MCF-7 | 12204694 | 0.6 | 50.0 | 240.0 | VQRKRQKLMP | VQRKRQKLMP |
MCF-7 | 12204694 | 0.7 | 50.0 | 240.0 | SKKKKTKV | SKKKKTKV |
MCF-7 | 12204694 | 1.15 | 50.0 | 240.0 | GRKRKKRT | GRKRKKRT |
MCF-7 | 12204694 | 0.85 | 50.0 | 240.0 | GKKKKRKREKL | GKKKKRKREKL |
MCF-7 | 12204694 | 0.48 | 50.0 | 240.0 | PKKKRKV | PKKKRKV |
MCF-7 | 12204694 | 0.6 | 50.0 | 240.0 | ERKKRRRE | ERKKRRRE |
MCF-7 | 12204694 | 0.45 | 50.0 | 240.0 | FKKFRKF | FKKFRKF |
K562 cells | 12783857 | 0.85 | 6.0 | 65.0 | RGGRLSYSRRRFSTSTGR | RGGRLSYSRRRFSTSTGR |
K562 cells | 12783857 | 1.2 | 6.0 | 65.0 | RRLSYSRRRF | RRLSYSRRRF |
K562 cells | 12783857 | 1.8 | 3.0 | 65.0 | RGGRLAYLRRRWAVLGR | RGGRLAYLRRRWAVLGR |
HeLa or TM12 cells | 12417587 | 1.2 | 15.0 | 30.0 | GIGKFLHSAKKWGKAFVGQIMNC | GIGKFLHSAKKWGKAFVGQIMNC |
HeLa or TM12 cells | 12417587 | 0.18 | 15.0 | 30.0 | TRSSRAGLQWPVGRVHRLLRKGGC | TRSSRAGLQWPVGRVHRLLRKGGC |
HeLa | 15054781 | 0.0 | 50.0 | 180.0 | VRLPPP | VRLPPP |
HeLa | 15054781 | 2.0 | 50.0 | 180.0 | VRLPPPVRLPPP | VRLPPPVRLPPP |
HeLa | 15054781 | 2.76 | 50.0 | 180.0 | VRLPPPVRLPPPVRLPPP | VRLPPPVRLPPPVRLPPP |
HeLa | 15054781 | 0.0 | 50.0 | 180.0 | VHLPPP | VHLPPP |
HeLa | 15054781 | 1.0 | 50.0 | 180.0 | VHLPPPVHLPPP | VHLPPPVHLPPP |
HeLa | 15054781 | 2.2 | 50.0 | 180.0 | VHLPPPVHLPPPVHLPPP | VHLPPPVHLPPPVHLPPP |
HeLa | 15054781 | 0.0 | 50.0 | 180.0 | VKLPPP | VKLPPP |
HeLa | 15054781 | 2.3 | 50.0 | 180.0 | VKLPPPVKLPPP | VKLPPPVKLPPP |
HeLa | 15054781 | 2.36 | 50.0 | 180.0 | VKLPPPVKLPPPVKLPPP | VKLPPPVKLPPPVKLPPP |
ECV-304 | 15346201 | 1.87 | 4.0 | 60.0 | KRVSRNKSEKKRR | KRVSRNKSEKKRR |
CHO K1 | 15937518 | 1.33 | 5.0 | 30.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
HeLa | 15937518 | 0.5 | 5.0 | 30.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
A549 cells | 15937518 | 0.36 | 5.0 | 30.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
CHO K1 | 15937518 | 1.33 | 5.0 | 30.0 | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
HeLa | 15937518 | 0.91 | 5.0 | 30.0 | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
A549 cells | 15937518 | 0.62 | 5.0 | 30.0 | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI | RQIKIWFQNRRMKWKKTYADFIASGRTGRRNAI |
CHO K1 | 15937518 | 0.55 | 5.0 | 30.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
HeLa | 15937518 | 0.26 | 5.0 | 30.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
A549 cells | 15937518 | 0.23 | 5.0 | 30.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
CHO K1 | 15937518 | 0.73 | 5.0 | 30.0 | GRKKRRQRRRPPQTYADFIASGRTGRRNAI | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
HeLa | 15937518 | 0.4 | 5.0 | 30.0 | GRKKRRQRRRPPQTYADFIASGRTGRRNAI | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
A549 cells | 15937518 | 0.26 | 5.0 | 30.0 | GRKKRRQRRRPPQTYADFIASGRTGRRNAI | GRKKRRQRRRPPQTYADFIASGRTGRRNAI |
CHO K1 | 15937518 | 0.3 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
HeLa | 15937518 | 0.2 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
A549 cells | 15937518 | 0.0 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
CHO K1 | 15937518 | 1.26 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
HeLa | 15937518 | 1.19 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
A549 cells | 15937518 | 0.95 | 5.0 | 30.0 | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI | AGYLLGKINLKALAALAKKILTYADFIASGRTGRRNAI |
CHO K1 | 15937518 | 1.49 | 5.0 | 30.0 | RRRRRRRRRRR | RRRRRRRRRRR |
HeLa | 15937518 | 1.64 | 5.0 | 30.0 | RRRRRRRRRRR | RRRRRRRRRRR |
A549 cells | 15937518 | 1.08 | 5.0 | 30.0 | RRRRRRRRRRR | RRRRRRRRRRR |
CHO K1 | 15937518 | 0.88 | 5.0 | 30.0 | RRRRRRRRRRRTYADFIASGRTGRRNAI | RRRRRRRRRRRTYADFIASGRTGRRNAI |
HeLa | 15937518 | 0.78 | 5.0 | 30.0 | RRRRRRRRRRRTYADFIASGRTGRRNAI | RRRRRRRRRRRTYADFIASGRTGRRNAI |
A549 cells | 15937518 | 0.56 | 5.0 | 30.0 | RRRRRRRRRRRTYADFIASGRTGRRNAI | RRRRRRRRRRRTYADFIASGRTGRRNAI |
A549 | 21875799 | 1.18 | 2.0 | 360.0 | KLALKLALKALKAALKLAGC | KLALKLALKALKAALKLAGC |
SK-OV-3 | 23301519 | 1.49 | 5.0 | 60.0 | RWRWRWRW | RWRWRWRW |
SK-OV-3 | 23301519 | 1.91 | 5.0 | 60.0 | WRWKKKKA | WRWKKKKA |
Human keratinocyte (HaCaT) cell | 23515421 | 1.73 | 500.0 | 240.0 | KETWWETWWTEWSQPKKKRKVC | KETWWETWWTEWSQPKKKRKVC |
human cervical cancer HeLa | 23515421 | 2.2 | 500.0 | 240.0 | KETWWETWWTEWSQPKKKRKVC | KETWWETWWTEWSQPKKKRKVC |
Human prostate adenocarcinoma cells (PC-3) | 23521800 | 2.17 | 5.0 | 180.0 | YTFGLKTSFNVQ | YTFGLKTSFNVQ |
Human prostate carcinoma cells (LNCaP) | 23521800 | 1.57 | 5.0 | 180.0 | YTFGLKTSFNVQ | YTFGLKTSFNVQ |
human embryonic lung fibroblasts (MRC-9) | 23521800 | 2.02 | 5.0 | 180.0 | YTFGLKTSFNVQ | YTFGLKTSFNVQ |
human spleen fibroblasts (Hs 697.Sp) | 23521800 | 1.41 | 5.0 | 180.0 | YTFGLKTSFNVQ | YTFGLKTSFNVQ |
HEK293T cells | 23521800 | 1.26 | 5.0 | 180.0 | YTFGLKTSFNVQ | YTFGLKTSFNVQ |
Human prostate adenocarcinoma cells (PC-3) | 23521800 | 3.13 | 5.0 | 180.0 | YTFGLKTSFNVQYTFGLKTSFNVQ | YTFGLKTSFNVQYTFGLKTSFNVQ |
Human prostate carcinoma cells (LNCaP) | 23521800 | 2.65 | 5.0 | 180.0 | YTFGLKTSFNVQYTFGLKTSFNVQ | YTFGLKTSFNVQYTFGLKTSFNVQ |
human embryonic lung fibroblasts (MRC-9) | 23521800 | 2.57 | 5.0 | 180.0 | YTFGLKTSFNVQYTFGLKTSFNVQ | YTFGLKTSFNVQYTFGLKTSFNVQ |
human spleen fibroblasts (Hs 697.Sp) | 23521800 | 2.0 | 5.0 | 180.0 | YTFGLKTSFNVQYTFGLKTSFNVQ | YTFGLKTSFNVQYTFGLKTSFNVQ |
HEK293T cells | 23521800 | 1.7 | 5.0 | 180.0 | YTFGLKTSFNVQYTFGLKTSFNVQ | YTFGLKTSFNVQYTFGLKTSFNVQ |
CHO-K1 cells | 25193363 | 2.41 | 0.1 | 180.0 | RRRRRRRR | RRRRRRRR |
CHO-K1 cells | 25193363 | 2.2 | 0.1 | 180.0 | HHHHHHHHRRRRRRRR | HHHHHHHHRRRRRRRR |
CHO-K1 cells | 25193363 | 2.29 | 0.1 | 180.0 | HHHHHHHHRRRRRRRRRRRRRRR | HHHHHHHHRRRRRRRRRRRRRRR |
CHO-K1 cells | 25193363 | 2.27 | 0.1 | 180.0 | HHHHHHHHHHHHRRRRRRRRRRRRRRR | HHHHHHHHHHHHRRRRRRRRRRRRRRR |
CHO-K1 cells | 25193363 | 2.34 | 0.1 | 180.0 | HHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR | HHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
CHO-K1 cells | 25193363 | 2.32 | 0.1 | 180.0 | HHHHHHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR | HHHHHHHHHHHHHHHHHHHHRRRRRRRRRRRRRRR |
HeLa | 25188671 | -0.74 | 0.1 | 120.0 | RLLRLLRLL | RLLRLLRLL |
HeLa | 24270856 | 2.0 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Jurkat E6.1 leukemia cells | 24270856 | 2.0 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Ovcar-3 cells | 24270856 | 2.0 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Caco-2 cells | 24270856 | 2.0 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.72 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.86 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.74 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.86 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.88 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.85 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.86 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.85 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.76 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 2.38 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Jurkat E6.1 leukemia cells | 24270856 | 1.98 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Ovcar-3 cells | 24270856 | 1.95 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Caco-2 cells | 24270856 | 2.12 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 2.14 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Jurkat E6.1 leukemia cells | 24270856 | 2.3 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Ovcar-3 cells | 24270856 | 2.22 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Caco-2 cells | 24270856 | 2.66 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.76 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Jurkat E6.1 leukemia cells | 24270856 | 1.94 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Ovcar-3 cells | 24270856 | 1.74 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Caco-2 cells | 24270856 | 1.93 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24270856 | 1.7 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Jurkat E6.1 leukemia cells | 24270856 | 1.88 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Ovcar-3 cells | 24270856 | 1.78 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
Caco-2 cells | 24270856 | 1.94 | 5.0 | 30.0 | KCFQWQRNMRKVRGPPVSCIKR | KCFQWQRNMRKVRGPPVSCIKR |
LNCaP | 24704199 | 1.89 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
SK-OV-3 | 24704199 | 1.22 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
MCF-7 as Hpn-expressing cells | 24704199 | 1.5 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
DU-145 | 24704199 | 1.0 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
PC-3 | 24704199 | 1.37 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
HaCaT as Hpn-non-expressing cells | 24704199 | 0.62 | 1.0 | 120.0 | IPLVVPLRRRRRRRRC | IPLVVPLRRRRRRRRC |
LNCaP | 24704199 | 1.09 | 3.0 | 120.0 | RRRRRRRRC | RRRRRRRRC |
LNCaP | 24704199 | 0.95 | 3.0 | 120.0 | IPLVVPLC | IPLVVPLC |
HeLa | 24768403 | 2.0 | 100.0 | 60.0 | YARVRRRGPRR | YARVRRRGPRR |
HeLa | 24896852 | 2.98 | 10.0 | 120.0 | Ac-RRRRRRRRR-miniPEG_linker-DELI | GRRRRRRRRRADELI |
HeLa | 24896852 | 2.46 | 10.0 | 120.0 | Ac-RKKRRQRRR-miniPEG_linker-DELI | GRKKRRQRRRADELI |
HeLa | 24896852 | 2.6 | 10.0 | 120.0 | Ac-RQIKIWFQNRRMKWKK-miniPEG_linker-DELI | GRQIKIWFQNRRMKWKKADELI |
HepG2 | 24811205 | 3.27 | 10.0 | 180.0 | LCLR | LCLR |
HepG2 | 24811205 | 2.4 | 10.0 | 180.0 | LLR | LLR |
HepG2 | 24811205 | 2.88 | 10.0 | 180.0 | LLLR | LLLR |
HepG2 | 24811205 | 2.76 | 10.0 | 180.0 | LLLLR | LLLLR |
HepG2 | 24811205 | 2.48 | 10.0 | 180.0 | LLLRR | LLLRR |
HepG2 | 24811205 | 3.08 | 10.0 | 180.0 | IIIR | IIIR |
HepG2 | 24811205 | 3.06 | 10.0 | 180.0 | VVVR | VVVR |
HepG2 | 24811205 | 2.98 | 10.0 | 180.0 | LCLK | LCLK |
HepG2 | 24811205 | 3.18 | 10.0 | 180.0 | LCLH | LCLH |
HepG2 | 24811205 | 3.22 | 10.0 | 180.0 | LCLE | LCLE |
HepG2 | 24811205 | 3.06 | 10.0 | 180.0 | LCLN | LCLN |
HepG2 | 24811205 | 3.19 | 10.0 | 180.0 | LCLQ | LCLQ |
HeLa | 25108152 | 2.17 | 2.0 | 60.0 | RRRRRRRR | RRRRRRRR |
KG1a cells | 25108152 | 2.18 | 2.0 | 60.0 | RRRRRRRR | RRRRRRRR |
HeLa | 25108152 | 2.02 | 2.0 | 60.0 | RRRRRRRR | RRRRRRRR |
KG1a cells | 25108152 | 2.0 | 2.0 | 60.0 | RRRRRRRR | RRRRRRRR |
HeLa | 25108152 | 2.34 | 2.0 | 60.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
KG1a cells | 25108152 | 2.07 | 2.0 | 60.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
HeLa | 25108152 | 2.02 | 2.0 | 60.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
KG1a cells | 25108152 | 2.0 | 2.0 | 60.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
HeLa | 25108152 | 2.95 | 2.0 | 60.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
KG1a cells | 25108152 | 2.67 | 2.0 | 60.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
HeLa | 25108152 | 2.02 | 2.0 | 60.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
KG1a cells | 25108152 | 2.0 | 2.0 | 60.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
Pluripotent mouse mesenchymal progenitor cell line (C3H10T1/2) | 24648725 | 2.0 | 0.1 | 20.0 | VSRRRRRRGGRRRR | VSRRRRRRGGRRRR |
Undifferentiated malignant glioma rat (F98) cell line | 24276021 | 4.95 | 10.0 | 120.0 | YGRKKRRQRRRC | YGRKKRRQRRRC |
Undifferentiated malignant glioma rat (F98) cell line | 24276021 | 5.11 | 10.0 | 120.0 | RQIKIWFQNRRMKWKKC | RQIKIWFQNRRMKWKKC |
Undifferentiated malignant glioma rat (F98) cell line | 24276021 | 5.15 | 10.0 | 120.0 | RRRRRRRRRC | RRRRRRRRRC |
MCF-7 | 24480922 | 3.16 | 50.0 | 60.0 | KKLFKKILKKL | KKLFKKILKKL |
mouse embryonic fibroblast 3T3 | 24480922 | 3.26 | 50.0 | 60.0 | KKLFKKILKKL | KKLFKKILKKL |
MCF-7 | 24480922 | 3.63 | 25.0 | 180.0 | KKLFKKILKKL | KKLFKKILKKL |
HeLa | 24611762 | 0.3 | 10.0 | 60.0 | RRRRR | RRRRR |
HeLa | 24611762 | 1.0 | 10.0 | 60.0 | RRRRRRRR | RRRRRRRR |
HeLa | 24611762 | 1.0 | 10.0 | 60.0 | YGRKKRRQRRR | YGRKKRRQRRR |
HeLa | 24611762 | 0.6 | 10.0 | 60.0 | YGRGGRRGRRR | YGRGGRRGRRR |
HeLa | 24697151 | 0.0 | 5.0 | 60.0 | ACSGSGSGCGSGSGSCG | ACSGSGSGCGSGSGSCG |
HeLa | 24697151 | 0.1 | 5.0 | 60.0 | ACSGRGSGCGSGRGSCG | ACSGRGSGCGSGRGSCG |
HeLa | 24697151 | 0.57 | 5.0 | 60.0 | ACRGSGRGCGRGSGRCG | ACRGSGRGCGRGSGRCG |
HeLa | 24697151 | 1.0 | 5.0 | 60.0 | ACSGRGRGCGRGRGSCG | ACSGRGRGCGRGRGSCG |
HeLa | 24697151 | 1.3 | 5.0 | 60.0 | ACGRGRGRCRGRGRGCG | ACGRGRGRCRGRGRGCG |
HeLa | 24697151 | 1.65 | 5.0 | 60.0 | ACRRSRRGCGRRSRRCG | ACRRSRRGCGRRSRRCG |
HeLa | 25056130 | 1.83 | 0.1 | 720.0 | LKKLLKLLKKLLKLAG | LKKLLKLLKKLLKLAG |
HeLa | 25056130 | 1.85 | 0.1 | 720.0 | LKKLCKLLKKLCKLAG | LKKLCKLLKKLCKLAG |
HEp-2 | 25154664 | 1.55 | 0.001 | 2880.0 | VTPHHVLVDEYTGEWVDSQFK | VTPHHVLVDEYTGEWVDSQFK |
HeLa | 25154664 | 1.64 | 0.001 | 2880.0 | VTPHHVLVDEYTGEWVDSQFK | VTPHHVLVDEYTGEWVDSQFK |
Vero | 25154664 | 1.51 | 0.001 | 2880.0 | VTPHHVLVDEYTGEWVDSQFK | VTPHHVLVDEYTGEWVDSQFK |
Cos-7 cells | 25154664 | 1.42 | 0.001 | 2880.0 | VTPHHVLVDEYTGEWVDSQFK | VTPHHVLVDEYTGEWVDSQFK |
SK-OV-3 cells | 25157458 | 3.56 | 5.0 | 60.0 | RRRRWWWW | RRRRWWWW |
A549 | 24928321 | 3.45 | 13.0 | 1440.0 | YGRKKRRQRRR | YGRKKRRQRRR |
A549 | 24928321 | 3.59 | 13.0 | 1440.0 | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
CHO-K1 | 24928321 | 4.2 | 13.0 | 1440.0 | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR | YGRKKRRQRRRYGRKKRRQRRRYGRKKRRQRRR |
HeLa | 24985034 | 0.0 | 8.0 | 60.0 | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
HeLa | 24985034 | -0.02 | 8.0 | 60.0 | GGVCPKILKKCRRDSDCPGACICRGNGWCGSGSD | GGVCPKILKKCRRDSDCPGACICRGNGWCGSGSD |
HeLa | 24985034 | 0.03 | 8.0 | 60.0 | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSD | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSD |
HeLa | 24985034 | -0.28 | 8.0 | 60.0 | GGVCPKILRRCRRDSDCPGACICRGNGWCGSGSD | GGVCPKILRRCRRDSDCPGACICRGNGWCGSGSD |
HeLa | 24985034 | 0.22 | 8.0 | 60.0 | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSR | GGVCPKILRRCRRDSDCPGACICRGNGYCGSGSR |
HeLa | 24985034 | 0.24 | 8.0 | 60.0 | GGVCPRILRRCRRDSDCPGACICRGNGYCGSGSK | GGVCPRILRRCRRDSDCPGACICRGNGYCGSGSK |
HeLa | 24985034 | 0.29 | 8.0 | 60.0 | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD | GGVCPKILKKCRRDSDCPGACICRGNGYCGSGSD |
HeLa | 24985034 | 0.0 | 16.0 | 60.0 | GRCTKSIPPICFPD | GRCTKSIPPICFPD |
HeLa | 24985034 | 0.02 | 16.0 | 60.0 | GACTKSIPPICFPD | GACTKSIPPICFPD |
HeLa | 24985034 | -0.07 | 16.0 | 60.0 | GRCTKSIPPICFPA | GRCTKSIPPICFPA |
HeLa | 24985034 | 0.05 | 16.0 | 60.0 | GRCTKSIPPICWPD | GRCTKSIPPICWPD |
HeLa | 24985034 | 0.0 | 16.0 | 60.0 | GRCTKSIPPICWPK | GRCTKSIPPICWPK |
HeLa | 24985034 | 0.1 | 16.0 | 60.0 | GRCTRSIPPKCWPD | GRCTRSIPPKCWPD |
HeLa | 24985034 | -0.3 | 8.0 | 60.0 | YGRKKRRQRRRPPQG | YGRKKRRQRRRPPQG |
Rat basophilic leukemia RBL-2H3 cells | 25016968 | 3.78 | 1.0 | 30.0 | KLALKLALKALKAALKLA | KLALKLALKALKAALKLA |
Rat basophilic leukemia RBL-2H3 cells | 25016968 | 3.52 | 1.0 | 30.0 | RQIKIWFQNRRMKWKK | RQIKIWFQNRRMKWKK |
Rat basophilic leukemia RBL-2H3 cells | 25016968 | 3.88 | 1.0 | 30.0 | RRRRRRRRR | RRRRRRRRR |
K-562 | 25387797 | 1.41 | 5.0 | 1080.0 | KSTGKANKITITNDKGRLSK | KSTGKANKITITNDKGRLSK |
primary culture of human corneal epithelial cells | 25467959 | 4.53 | 5.0 | 60.0 | RKKRRQRRRRKKRRQRRR | RKKRRQRRRRKKRRQRRR |
primary culture of human corneal epithelial cells | 25467959 | 4.04 | 5.0 | 60.0 | AKKRRQRRRAKKRRQRRR | AKKRRQRRRAKKRRQRRR |
HT29 | 25511292 | 2.6 | 4.0 | 120.0 | GWTLNSAGYLLGKINLKALAALAKKIL | GWTLNSAGYLLGKINLKALAALAKKIL |
HCT116 | 25511292 | 2.34 | 4.0 | 120.0 | GWTLNSAGYLLGKINLKALAALAKKIL | GWTLNSAGYLLGKINLKALAALAKKIL |
HT29 | 25511292 | 1.9 | 4.0 | 120.0 | GWTLNSAGYLLGKINLKALAALAKKIL | GWTLNSAGYLLGKINLKALAALAKKIL |
HCT116 | 25511292 | 1.95 | 4.0 | 120.0 | GWTLNSAGYLLGKINLKALAALAKKIL | GWTLNSAGYLLGKINLKALAALAKKIL |
HT29 | 25511292 | 1.7 | 4.0 | 120.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
HCT116 | 25511292 | 2.18 | 4.0 | 120.0 | AGYLLGKINLKALAALAKKIL | AGYLLGKINLKALAALAKKIL |
Plant cells | 25514997 | 2.06 | 20.0 | 60.0 | KWCFRVCYRGICYRRCRGK | KWCFRVCYRGICYRRCRGK |
HeLa cells | 25514997 | 2.18 | 30.0 | 60.0 | KWCFRVCYRGICYRRCRGK | KWCFRVCYRGICYRRCRGK |
Plant cells | 25514997 | 2.06 | 20.0 | 60.0 | KWSFRVSYRGISYRRSRGK | KWSFRVSYRGISYRRSRGK |
HeLa cells | 25514997 | 2.16 | 30.0 | 60.0 | KWSFRVSYRGISYRRSRGK | KWSFRVSYRGISYRRSRGK |
Plant cells | 25514997 | 2.18 | 20.0 | 60.0 | KWFRVYRGIYRRRGK | KWFRVYRGIYRRRGK |
HeLa cells | 25514997 | 2.69 | 30.0 | 60.0 | KWFRVYRGIYRRRGK | KWFRVYRGIYRRRGK |
Plant cells | 25514997 | 1.53 | 20.0 | 60.0 | KWCFAVCYAGICYAACAGK | KWCFAVCYAGICYAACAGK |
HeLa cells | 25514997 | 1.54 | 30.0 | 60.0 | KWCFAVCYAGICYAACAGK | KWCFAVCYAGICYAACAGK |
Jurkat E6 cells | 25524829 | 2.97 | 10.0 | 10.0 | RRGRRG | RRGRRG |
Jurkat E6 cells | 25524829 | 3.44 | 10.0 | 10.0 | RRRRRR | RRRRRR |
Jurkat E6 cells | 25524829 | 0.0 | 10.0 | 10.0 | RRRRRR | RRRRRR |
MCF-7 cells | 25547808 | 1.39 | 1.0 | 240.0 | HHHRRRRRRRR | HHHRRRRRRRR |
MCF-7 cells | 25547808 | 2.23 | 1.0 | 240.0 | HHHRRRRRRRR | HHHRRRRRRRR |
Bone marrow dendritic cells | 24901376 | 1.03 | 40.0 | 120.0 | RRRRRRRR | RRRRRRRR |
HeLa | 24930129 | 3.11 | 1.0 | 60.0 | CKYGRKKRRQRRR | CKYGRKKRRQRRR |
MEF cells | 24583082 | 1.93 | 100.0 | 240.0 | KRKRWHW | KRKRWHW |
Cultured Human Dental Pulp Stem Cells (hDPSCs) | 21990606 | 2.0 | 0.5 | 30.0 | VSRRRRRRGGRRRR | VSRRRRRRGGRRRR |
ARPE-19 | 22100438 | 0.0 | 2.1 | 30.0 | CGRKKRRQRRRPPQ | CGRKKRRQRRRPPQ |
CHO wt | 22100438 | 0.0 | 2.1 | 30.0 | CGRKKRRQRRRPPQ | CGRKKRRQRRRPPQ |
CHO pgsB-618 cells | 22100438 | 0.0 | 2.1 | 30.0 | CGRKKRRQRRRPPQ | CGRKKRRQRRRPPQ |
ARPE-19 | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRWWRQRRRPPQ | CGRKKRWWRQRRRPPQ |
CHO wt | 22100438 | -0.04 | 2.1 | 30.0 | CGRKKRWWRQRRRPPQ | CGRKKRWWRQRRRPPQ |
CHO pgsB-618 cells | 22100438 | 0.06 | 2.1 | 30.0 | CGRKKRWWRQRRRPPQ | CGRKKRWWRQRRRPPQ |
ARPE-19 | 22100438 | -0.05 | 2.1 | 30.0 | CGRKKRRQRRWWRPPQ | CGRKKRRQRRWWRPPQ |
CHO wt | 22100438 | 0.0 | 2.1 | 30.0 | CGRKKRRQRRWWRPPQ | CGRKKRRQRRWWRPPQ |
CHO pgsB-618 cells | 22100438 | 0.02 | 2.1 | 30.0 | CGRKKRRQRRWWRPPQ | CGRKKRRQRRWWRPPQ |
ARPE-19 | 22100438 | -0.02 | 2.1 | 30.0 | CGRKKRRQRWWRRPPQ | CGRKKRRQRWWRRPPQ |
CHO wt | 22100438 | 0.06 | 2.1 | 30.0 | CGRKKRRQRWWRRPPQ | CGRKKRRQRWWRRPPQ |
CHO pgsB-618 cells | 22100438 | 0.03 | 2.1 | 30.0 | CGRKKRRQRWWRRPPQ | CGRKKRRQRWWRRPPQ |
ARPE-19 | 22100438 | -0.09 | 2.1 | 30.0 | CGRKKRWWRQRWWRWWRPPQ | CGRKKRWWRQRWWRWWRPPQ |
CHO wt | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRWWRQRWWRWWRPPQ | CGRKKRWWRQRWWRWWRPPQ |
CHO pgsB-618 cells | 22100438 | -0.01 | 2.1 | 30.0 | CGRKKRWWRQRWWRWWRPPQ | CGRKKRWWRQRWWRWWRPPQ |
ARPE-19 | 22100438 | 0.01 | 2.1 | 30.0 | CGRKKRAARQRRRPPQ | CGRKKRAARQRRRPPQ |
CHO wt | 22100438 | -0.04 | 2.1 | 30.0 | CGRKKRAARQRRRPPQ | CGRKKRAARQRRRPPQ |
CHO pgsB-618 cells | 22100438 | -0.04 | 2.1 | 30.0 | CGRKKRAARQRRRPPQ | CGRKKRAARQRRRPPQ |
ARPE-19 | 22100438 | -0.04 | 2.1 | 30.0 | CGRKKRRQRRAARPPQ | CGRKKRRQRRAARPPQ |
CHO wt | 22100438 | -0.05 | 2.1 | 30.0 | CGRKKRRQRRAARPPQ | CGRKKRRQRRAARPPQ |
CHO pgsB-618 cells | 22100438 | -0.06 | 2.1 | 30.0 | CGRKKRRQRRAARPPQ | CGRKKRRQRRAARPPQ |
ARPE-19 | 22100438 | -0.06 | 2.1 | 30.0 | CGRKKRRQRAARRPPQ | CGRKKRRQRAARRPPQ |
CHO wt | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRRQRAARRPPQ | CGRKKRRQRAARRPPQ |
CHO pgsB-618 cells | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRRQRAARRPPQ | CGRKKRRQRAARRPPQ |
ARPE-19 | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRAARQRAARAARPPQ | CGRKKRAARQRAARAARPPQ |
CHO wt | 22100438 | -0.12 | 2.1 | 30.0 | CGRKKRAARQRAARAARPPQ | CGRKKRAARQRAARAARPPQ |
CHO pgsB-618 cells | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRAARQRAARAARPPQ | CGRKKRAARQRAARAARPPQ |
ARPE-19 | 22100438 | -0.02 | 2.1 | 30.0 | CGRKKRLLRQRRRPPQ | CGRKKRLLRQRRRPPQ |
CHO wt | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRLLRQRRRPPQ | CGRKKRLLRQRRRPPQ |
CHO pgsB-618 cells | 22100438 | -0.11 | 2.1 | 30.0 | CGRKKRLLRQRRRPPQ | CGRKKRLLRQRRRPPQ |
ARPE-19 | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRRQRRLLRPPQ | CGRKKRRQRRLLRPPQ |
CHO wt | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRRQRRLLRPPQ | CGRKKRRQRRLLRPPQ |
CHO pgsB-618 cells | 22100438 | -0.14 | 2.1 | 30.0 | CGRKKRRQRRLLRPPQ | CGRKKRRQRRLLRPPQ |
ARPE-19 | 22100438 | -0.05 | 2.1 | 30.0 | CGRKKRRQRLLRRPPQ | CGRKKRRQRLLRRPPQ |
CHO wt | 22100438 | -0.06 | 2.1 | 30.0 | CGRKKRRQRLLRRPPQ | CGRKKRRQRLLRRPPQ |
CHO pgsB-618 cells | 22100438 | -0.12 | 2.1 | 30.0 | CGRKKRRQRLLRRPPQ | CGRKKRRQRLLRRPPQ |
ARPE-19 | 22100438 | 0.07 | 2.1 | 30.0 | CGRKKRLLRQRLLRLLRPPQ | CGRKKRLLRQRLLRLLRPPQ |
CHO wt | 22100438 | 0.13 | 2.1 | 30.0 | CGRKKRLLRQRLLRLLRPPQ | CGRKKRLLRQRLLRLLRPPQ |
CHO pgsB-618 cells | 22100438 | -0.02 | 2.1 | 30.0 | CGRKKRLLRQRLLRLLRPPQ | CGRKKRLLRQRLLRLLRPPQ |
U373 MG cells | 22148546 | 1.2 | 5.0 | 60.0 | INLKALAALAKKIL | INLKALAALAKKIL |
U373 MG cells | 22148546 | 0.99 | 5.0 | 60.0 | LIKKALAALAKLNI | LIKKALAALAKLNI |
U251-MG | 22465335 | 1.74 | 1.0 | 30.0 | RRR | RRR |
HeLa | 22486588 | 1.79 | 1.0 | 15.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
HeLa | 22486588 | 1.27 | 1.0 | 15.0 | LILIGRRRRRRRRGC | LILIGRRRRRRRRGC |
HeLa | 22486588 | 1.34 | 1.0 | 15.0 | FFGRRRRRRRGC | FFGRRRRRRRGC |
HeLa | 22486588 | 2.0 | 1.0 | 15.0 | FFFFGRRRRRRRRGC | FFFFGRRRRRRRRGC |
The HeLa cells | 22688249 | 1.8 | 10.0 | 60.0 | GLWWKAWWKAWWKSLWWRKRKRKA | GLWWKAWWKAWWKSLWWRKRKRKA |
CHO-K1 cells | 22712882 | 2.88 | 10.0 | 60.0 | RRRRWWWWRRRR | RRRRWWWWRRRR |
CHO-K1 cells | 22712882 | 3.15 | 10.0 | 60.0 | RWRRWRRWRRWR | RWRRWRRWRRWR |
NHDF | 22805558 | 0.28 | 10.0 | 180.0 | YGRKKRPQRRR | YGRKKRPQRRR |
Many Human neoplastic cells including HeLa | 22805558 | 0.6 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
Lovo | 22805558 | 1.59 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
A549 | 22805558 | 0.48 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
MCF-7 | 22805558 | 0.0 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
HepG2 | 22805558 | 0.7 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
U2OS | 22805558 | 0.78 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
K562 | 22805558 | 0.3 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
NHDF | 22805558 | 0.0 | 10.0 | 180.0 | DSLKSYWYLQKFSWR | DSLKSYWYLQKFSWR |
Many Human neoplastic cells including HeLa | 22805558 | 0.48 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
Lovo | 22805558 | 0.3 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
A549 | 22805558 | 0.0 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
MCF-7 | 22805558 | 0.0 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
HepG2 | 22805558 | 1.6 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
U2OS | 22805558 | 0.48 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
K562 | 22805558 | 1.85 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
NHDF | 22805558 | 0.0 | 10.0 | 180.0 | KRPTMRFRYTWNPMK | KRPTMRFRYTWNPMK |
MCF-7 cells | 22828784 | 1.75 | 8.0 | 60.0 | RRRRRRRR | RRRRRRRR |
Caco-2 cell culture | 23863452 | -0.69 | 0.5 | 480.0 | VSRRRRRRGGRRRR | VSRRRRRRGGRRRR |
HeLa cells | 25459448 | 2.05 | 10.0 | 60.0 | KKKKKKNKKLQQRGD | KKKKKKNKKLQQRGD |
HeLa cells | 25459448 | 1.32 | 10.0 | 60.0 | RGDGPRRRPRKRRGR | RGDGPRRRPRKRRGR |
HeLa cells | 25459448 | 2.22 | 10.0 | 60.0 | RRRQKRIVVRRRLIR | RRRQKRIVVRRRLIR |
HeLa cells | 25459448 | 2.0 | 10.0 | 60.0 | RRVWRRYRRQRWCRR | RRVWRRYRRQRWCRR |
HeLa cells | 25459448 | 1.88 | 10.0 | 60.0 | RRARRPRRLRPAPGR | RRARRPRRLRPAPGR |
HeLa cells | 25459448 | 2.32 | 10.0 | 60.0 | LLRARWRRRRSRRFR | LLRARWRRRRSRRFR |
HeLa cells | 25459448 | 1.92 | 10.0 | 60.0 | RGPRRQPRRHRRPRR | RGPRRQPRRHRRPRR |
HeLa cells | 25459448 | 2.98 | 10.0 | 60.0 | RRWRRWNRFNRRRCR | RRWRRWNRFNRRRCR |
HeLa cells | 25459448 | 2.0 | 10.0 | 60.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
HeLa | 34504427 | 1.51 | 10.0 | 120.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
HeLa | 34504427 | 1.58 | 10.0 | 120.0 | VLERAKRRAV | VLERAKRRAV |
HeLa | 34504427 | 1.73 | 10.0 | 120.0 | PDDIKPRRIRKPRY | PDDIKPRRIRKPRY |
HeLa | 34504427 | 0.3 | 10.0 | 120.0 | NTKRRLEGAKKA | NTKRRLEGAKKA |
HeLa | 34504427 | 0.95 | 10.0 | 120.0 | AAKFIKKRRTKSS | AAKFIKKRRTKSS |
HeLa | 34504427 | 0.6 | 10.0 | 120.0 | TQKEKKAARARSK | TQKEKKAARARSK |
HeLa | 34504427 | 1.0 | 10.0 | 120.0 | RKRRESASSSSSVKKAKKP | RKRRESASSSSSVKKAKKP |
HeLa | 34504427 | 1.45 | 10.0 | 120.0 | KRKGRLRSKGKK | KRKGRLRSKGKK |
HeLa | 34504427 | 0.9 | 10.0 | 120.0 | AEADKPRRLGRLK | AEADKPRRLGRLK |
HeLa | 34504427 | 1.58 | 10.0 | 120.0 | GECTYAGRKRRRPLQK | GECTYAGRKRRRPLQK |
HeLa | 34504427 | 1.2 | 10.0 | 120.0 | TPPTSAKKRKL | TPPTSAKKRKL |
HeLa | 34504427 | 0.6 | 10.0 | 120.0 | VAAKKRKKDML | VAAKKRKKDML |
PC3 | 34504427 | 1.81 | 10.0 | 120.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
PC3 | 34504427 | 1.78 | 10.0 | 120.0 | VLERAKRRAV | VLERAKRRAV |
PC3 | 34504427 | 1.87 | 10.0 | 120.0 | PDDIKPRRIRKPRY | PDDIKPRRIRKPRY |
PC3 | 34504427 | 0.78 | 10.0 | 120.0 | NTKRRLEGAKKA | NTKRRLEGAKKA |
PC3 | 34504427 | 1.26 | 10.0 | 120.0 | AAKFIKKRRTKSS | AAKFIKKRRTKSS |
PC3 | 34504427 | 0.78 | 10.0 | 120.0 | TQKEKKAARARSK | TQKEKKAARARSK |
PC3 | 34504427 | 1.34 | 10.0 | 120.0 | RKRRESASSSSSVKKAKKP | RKRRESASSSSSVKKAKKP |
PC3 | 34504427 | 1.66 | 10.0 | 120.0 | KRKGRLRSKGKK | KRKGRLRSKGKK |
PC3 | 34504427 | 1.26 | 10.0 | 120.0 | AEADKPRRLGRLK | AEADKPRRLGRLK |
PC3 | 34504427 | 1.73 | 10.0 | 120.0 | GECTYAGRKRRRPLQK | GECTYAGRKRRRPLQK |
PC3 | 34504427 | 1.32 | 10.0 | 120.0 | TPPTSAKKRKL | TPPTSAKKRKL |
PC3 | 34504427 | 1.0 | 10.0 | 120.0 | VAAKKRKKDML | VAAKKRKKDML |
U87 | 34504427 | 1.51 | 10.0 | 120.0 | GRKKRRQRRRPPQ | GRKKRRQRRRPPQ |
U87 | 34504427 | 1.6 | 10.0 | 120.0 | VLERAKRRAV | VLERAKRRAV |
U87 | 34504427 | 1.69 | 10.0 | 120.0 | PDDIKPRRIRKPRY | PDDIKPRRIRKPRY |
U87 | 34504427 | 0.48 | 10.0 | 120.0 | NTKRRLEGAKKA | NTKRRLEGAKKA |
U87 | 34504427 | 1.38 | 10.0 | 120.0 | AAKFIKKRRTKSS | AAKFIKKRRTKSS |
U87 | 34504427 | 1.04 | 10.0 | 120.0 | TQKEKKAARARSK | TQKEKKAARARSK |
U87 | 34504427 | 1.51 | 10.0 | 120.0 | RKRRESASSSSSVKKAKKP | RKRRESASSSSSVKKAKKP |
U87 | 34504427 | 1.45 | 10.0 | 120.0 | KRKGRLRSKGKK | KRKGRLRSKGKK |
U87 | 34504427 | 1.0 | 10.0 | 120.0 | AEADKPRRLGRLK | AEADKPRRLGRLK |
U87 | 34504427 | 1.56 | 10.0 | 120.0 | GECTYAGRKRRRPLQK | GECTYAGRKRRRPLQK |
U87 | 34504427 | 1.26 | 10.0 | 120.0 | TPPTSAKKRKL | TPPTSAKKRKL |
U87 | 34504427 | 0.48 | 10.0 | 120.0 | VAAKKRKKDML | VAAKKRKKDML |
Saos-2 cells | 30410976 | -3.4 | 1.0 | 30.0 | MGPSQPTYPGDDAPVRDLIRFYRDLRRYLNVVTRHRY | MGPSQPTYPGDDAPVRDLIRFYRDLRRYLNVVTRHRY |
Saos-2 cells | 30410976 | -3.14 | 1.0 | 30.0 | MRRRRRRR | MRRRRRRR |
Saos-2 cells | 30410976 | -3.12 | 1.0 | 30.0 | MLEPGEKPYKCPECGKSFSASAALVAHQRTHTGKKTS | MLEPGEKPYKCPECGKSFSASAALVAHQRTHTGKKTS |
Saos-2 cells | 30410976 | -2.85 | 1.0 | 30.0 | MRQIKIWFQNRRMKWKK | MRQIKIWFQNRRMKWKK |
Saos-2 cells | 30410976 | -2.67 | 1.0 | 30.0 | MYSCNVCGKAFVLSRHLNRHLRVHRRAT | MYSCNVCGKAFVLSRHLNRHLRVHRRAT |
HEK293 | 30135446 | 1.34 | 40.0 | 60.0 | GRKKRRQRRRPPQRKC | GRKKRRQRRRPPQRKC |
HEK293 | 30135446 | 1.56 | 40.0 | 60.0 | RKQKSLQTKLAENPPVPRKKRQSRPRWKQWLQK | RKQKSLQTKLAENPPVPRKKRQSRPRWKQWLQK |
HEK293 | 30135446 | 1.86 | 40.0 | 60.0 | PLKPKKPKTQEKKKKQPPKPKKPKTQEKKKKQPPKPKR | PLKPKKPKTQEKKKKQPPKPKKPKTQEKKKKQPPKPKR |
eGFP HeLa 654 | 29721534 | 4.26 | 5.0 | 1320.0 | KQPRIKRKK | KQPRIKRKK |
eGFP HeLa 654 | 29721534 | 4.24 | 5.0 | 1320.0 | LKKRRKLPKKKPIRNEQ | LKKRRKLPKKKPIRNEQ |
eGFP HeLa 654 | 29721534 | 4.37 | 5.0 | 1320.0 | KKYRGRKRHPR | KKYRGRKRHPR |
eGFP HeLa 654 | 29721534 | 4.33 | 5.0 | 1320.0 | APKRKKLKKRF | APKRKKLKKRF |
eGFP HeLa 654 | 29721534 | 4.27 | 5.0 | 1320.0 | GRKAARAPGRRKQ | GRKAARAPGRRKQ |
eGFP HeLa 654 | 29721534 | 3.7 | 5.0 | 1320.0 | HDLPKGG | HDLPKGG |
eGFP HeLa 654 | 29721534 | 3.97 | 5.0 | 1320.0 | AGSHRRL | AGSHRRL |
MDA-MB-231 | 27189051 | 5.21 | 2.5 | 30.0 | RRWRRWNRFNRRRCR | RRWRRWNRFNRRRCR |
A549 | 26942714 | 1.97 | 10.0 | 60.0 | CHHHHHRRRRRRRRRHHHHHC | CHHHHHRRRRRRRRRHHHHHC |
A549 | 26942714 | 1.97 | 10.0 | 60.0 | CRRWQWRMKKLGC | CRRWQWRMKKLGC |
A549 | 26942714 | 1.99 | 10.0 | 60.0 | FKCRRWQWRMKK | FKCRRWQWRMKK |
A549 | 26942714 | 1.97 | 10.0 | 60.0 | KCRRWQWRMKK | KCRRWQWRMKK |
A549 | 26942714 | 1.89 | 10.0 | 60.0 | RRWQWRMKK | RRWQWRMKK |
A549 | 26942714 | 1.99 | 10.0 | 60.0 | RRWQWR | RRWQWR |
A549 | 26942714 | 1.98 | 10.0 | 60.0 | RRWQW | RRWQW |
A549 | 26942714 | 1.4 | 10.0 | 60.0 | RWQWR | RWQWR |
A549 | 26942714 | 0.95 | 10.0 | 60.0 | RWQW | RWQW |
MCF7 | 35216417 | 0.51 | 2.0 | 1440.0 | RGGRLSYSRRRFSTSTGR | RGGRLSYSRRRFSTSTGR |
MCF7 | 35216417 | -0.1 | 2.0 | 1440.0 | RGGRLSYSRRRFSTSTGR | RGGRLSYSRRRFSTSTGR |
NCI/ADR | 35216417 | 0.11 | 2.0 | 1440.0 | RGGRLSYSRRRFSTSTGR | RGGRLSYSRRRFSTSTGR |
NCI/ADR | 35216417 | 0.04 | 2.0 | 1440.0 | RGGRLSYSRRRFSTSTGR | RGGRLSYSRRRFSTSTGR |
P. falciparum-infected erythrocytes | 35074306 | 1.66 | 5.0 | 30.0 | YKQCHKKGGHCFPKEKICLPPSSDFGKMDCRWRWKCCKKGSG | YKQCHKKGGHCFPKEKICLPPSSDFGKMDCRWRWKCCKKGSG |
HeLa | 34994362 | 2.74 | 10.0 | 30.0 | RKLRRLLRRLKRL | RKLRRLLRRLKRL |
HeLa | 34994362 | 2.82 | 10.0 | 30.0 | KRKLRRLLRRLKRL | KRKLRRLLRRLKRL |
HeLa | 34994362 | 2.93 | 10.0 | 30.0 | RKLRRLLRRLKRL | RKLRRLLRRLKRL |
HeLa | 34994362 | 2.86 | 10.0 | 30.0 | KRKLRRLLRRLKRL | KRKLRRLLRRLKRL |
HeLa | 34994362 | 2.93 | 10.0 | 30.0 | RKLRRLLRRLKRL | RKLRRLLRRLKRL |
HeLa | 34994362 | 2.86 | 10.0 | 30.0 | KRKLRRLLRRLKRL | KRKLRRLLRRLKRL |
HeLa | 27836642 | 2.4 | 5.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
HeLa | 27836642 | 2.41 | 10.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
HeLa | 27836642 | 2.54 | 15.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
HeLa | 27836642 | 2.6 | 20.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
HeLa | 27836642 | 2.65 | 30.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
HeLa | 27836642 | 2.7 | 40.0 | 120.0 | CRWRWKCCKK | CRWRWKCCKK |
DC2.4 cells | 31339694 | 1.7 | 10.0 | 1440.0 | KVRVRVRVDPPTRVRERVKC | KVRVRVRVDPPTRVRERVKC |
CCRF-CEM | 34491768 | 2.08 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
CCRF-CEM | 34491768 | 2.0 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
CCRF-CEM | 34491768 | 2.3 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
CCRF-CEM | 34491768 | 2.48 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
CCRF-CEM | 34491768 | 2.7 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
SK-OV-3 | 34491768 | 2.0 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
SK-OV-3 | 34491768 | 2.08 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
SK-OV-3 | 34491768 | 2.08 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
SK-OV-3 | 34491768 | 2.11 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
SK-OV-3 | 34491768 | 2.11 | 10.0 | 180.0 | RWRWRWRWRWKRWRWRWRWRW | RWRWRWRWRWKRWRWRWRWRW |
HeLa cells | 34959356 | 0.0 | 1.0 | 120.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 3.0 | 1.0 | 120.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 3.4 | 1.0 | 120.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 4.04 | 1.0 | 120.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 3.4 | 1.0 | 120.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 2.0 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 2.48 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 2.54 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 3.04 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 34959356 | 2.3 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
A375 cells | 30240193 | 1.0 | 0.001 | 1440.0 | CAAKA | CAAKA |
A375-R cells | 30240193 | 1.23 | 0.001 | 1440.0 | CAAKA | CAAKA |
MSTO cells | 30240193 | 0.9 | 0.001 | 1440.0 | CAAKA | CAAKA |
MSTO-R cells | 30240193 | 1.4 | 0.001 | 1440.0 | CAAKA | CAAKA |
9L cells | 30240193 | 0.48 | 0.001 | 1440.0 | CAAKA | CAAKA |
9L-R cells | 30240193 | 0.48 | 0.001 | 1440.0 | CAAKA | CAAKA |
LN18 cells | 30240193 | 0.9 | 0.001 | 1440.0 | CAAKA | CAAKA |
U87 cells | 30240193 | 0.9 | 0.001 | 1440.0 | CAAKA | CAAKA |
HeLa cells | 28159722 | 4.7 | 20.0 | 60.0 | KWRRKLKKLRPKKKRKV | KWRRKLKKLRPKKKRKV |
HeLa cells | 28159722 | 3.9 | 20.0 | 60.0 | KWRRKLKKLR | KWRRKLKKLR |
HeLa cells | 28159722 | 0.0 | 20.0 | 60.0 | PKKKRKV | PKKKRKV |
HeLa cells | 28159722 | 0.0 | 20.0 | 60.0 | AWRRKLKALAPAKKAKV | AWRRKLKALAPAKKAKV |
HDF cells | 32374475 | 2.42 | 0.2 | 30.0 | GRKKRRQRRK | GRKKRRQRRK |
HDF cells | 32374475 | 2.32 | 2.0 | 30.0 | GRKKRRQRRK | GRKKRRQRRK |
HDF cells | 32374475 | 2.32 | 0.2 | 30.0 | RNQRKTVRCFRCRQAGHWISDCRLKSK | RNQRKTVRCFRCRQAGHWISDCRLKSK |
HDF cells | 32374475 | 3.26 | 2.0 | 30.0 | RNQRKTVRCFRCRQAGHWISDCRLKSK | RNQRKTVRCFRCRQAGHWISDCRLKSK |
hDPSC cells | 32374475 | 2.24 | 0.2 | 30.0 | GRKKRRQRRK | GRKKRRQRRK |
hDPSC cells | 32374475 | 2.36 | 2.0 | 30.0 | GRKKRRQRRK | GRKKRRQRRK |
hDPSC cells | 32374475 | 2.38 | 0.2 | 30.0 | RNQRKTVRCFRCRQAGHWISDCRLKSK | RNQRKTVRCFRCRQAGHWISDCRLKSK |
hDPSC cells | 32374475 | 3.7 | 2.0 | 30.0 | RNQRKTVRCFRCRQAGHWISDCRLKSK | RNQRKTVRCFRCRQAGHWISDCRLKSK |
PK15 cells | 30108178 | 2.84 | 6.0 | 30.0 | MTYPRRRFRRRRHRPRS | MTYPRRRFRRRRHRPRS |
HeLa cells | 30108178 | 2.76 | 6.0 | 30.0 | MTYPRRRFRRRRHRPRS | MTYPRRRFRRRRHRPRS |
3T3 cells | 30108178 | 2.88 | 6.0 | 30.0 | MTYPRRRFRRRRHRPRS | MTYPRRRFRRRRHRPRS |
HeLa cells | 31936737 | 0.9 | 1.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 0.85 | 10.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.51 | 25.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.45 | 50.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 0.85 | 1.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.08 | 10.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.7 | 25.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.72 | 50.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 0.7 | 1.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.34 | 10.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.76 | 25.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.88 | 50.0 | 60.0 | GRKKRRQRRR | GRKKRRQRRR |
HeLa cells | 31936737 | 1.04 | 1.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.26 | 10.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.08 | 25.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.08 | 50.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 0.9 | 1.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.23 | 10.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.11 | 25.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.11 | 50.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.0 | 1.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.43 | 10.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.41 | 25.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 31936737 | 1.4 | 50.0 | 60.0 | RRMKWKK | RRMKWKK |
HeLa cells | 34152716 | 0.0 | 4.0 | 60.0 | YGRKKRRQRRRPPQG | YGRKKRRQRRRPPQG |
HeLa cells | 34152716 | -0.7 | 4.0 | 60.0 | YGGGKGGQGGGPPQG | YGGGKGGQGGGPPQG |
HeLa cells | 34152716 | -0.52 | 4.0 | 60.0 | CPKILKKCRRDSDCPGACICRGNGYCGSGSDEETGEGGV | CPKILKKCRRDSDCPGACICRGNGYCGSGSDEETGEGGV |
HeLa cells | 34152716 | -0.4 | 4.0 | 60.0 | CPFWRRRRCKRDSDCPGACICRGNGYCGSGCDEETGECGV | CPFWRRRRCKRDSDCPGACICRGNGYCGSGCDEETGECGV |
MCF-7 cells | 32116040 | 1.4 | 5.0 | 60.0 | RRWWWWRR | RRWWWWRR |
MCF-7 cells | 32116040 | 1.86 | 10.0 | 60.0 | RRWWWWRR | RRWWWWRR |
MCF-7 cells | 32116040 | 1.85 | 15.0 | 60.0 | RRWWWWRR | RRWWWWRR |
MCF-7 cells | 32116040 | 1.97 | 25.0 | 60.0 | RRWWWWRR | RRWWWWRR |
MCF-7 cells | 32116040 | 0.3 | 5.0 | 60.0 | WWWRRRRWWW | WWWRRRRWWW |
MCF-7 cells | 32116040 | 0.3 | 10.0 | 60.0 | WWWRRRRWWW | WWWRRRRWWW |
MCF-7 cells | 32116040 | 0.9 | 15.0 | 60.0 | WWWRRRRWWW | WWWRRRRWWW |
MCF-7 cells | 32116040 | 1.08 | 25.0 | 60.0 | WWWRRRRWWW | WWWRRRRWWW |
bEnd.3 cell | 32561686 | 0.7 | 0.1 | 6.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.0 | 0.1 | 15.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.3 | 0.1 | 30.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.59 | 0.1 | 60.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.85 | 0.1 | 240.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 0.7 | 0.1 | 6.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.26 | 0.1 | 15.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.4 | 0.1 | 30.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.57 | 0.1 | 60.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.85 | 0.1 | 240.0 | GIGAVLKVLTTGLPALISWIKRKRQ | GIGAVLKVLTTGLPALISWIKRKRQ |
bEnd.3 cell | 32561686 | 1.0 | 0.1 | 6.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.23 | 0.1 | 15.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.26 | 0.1 | 30.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.59 | 0.1 | 60.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.86 | 0.1 | 240.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 0.9 | 0.1 | 6.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.26 | 0.1 | 15.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.34 | 0.1 | 30.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.6 | 0.1 | 60.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 1.86 | 0.1 | 240.0 | AAVALLPAVLLALLAP | AAVALLPAVLLALLAP |
bEnd.3 cell | 32561686 | 0.6 | 0.1 | 6.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 0.85 | 0.1 | 15.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.48 | 0.1 | 30.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.62 | 0.1 | 60.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.83 | 0.1 | 240.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 0.6 | 0.1 | 6.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 0.85 | 0.1 | 15.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.45 | 0.1 | 30.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.6 | 0.1 | 60.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
bEnd.3 cell | 32561686 | 1.86 | 0.1 | 240.0 | FFLIPKGRRRRRRRRGC | FFLIPKGRRRRRRRRGC |
CHO-K1 cells | 29247010 | 2.78 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 2.95 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 3.11 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 2.78 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 3.18 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 3.2 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 3.18 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
CHO-K1 cells | 29247010 | 3.0 | 50.0 | 30.0 | NVFKGNTISDKISFNFSDK | NVFKGNTISDKISFNFSDK |
HeLa cells | 27189051 | 4.4 | 5.0 | 60.0 | RRWRRWNRFNRRRCR | RRWRRWNRFNRRRCR |
MCF-7 cel | 28933182 | 1.93 | 10.0 | 120.0 | KWKWKWKW | KWKWKWKW |
MCF-7 cel | 28933182 | 1.95 | 25.0 | 120.0 | KWKWKWKW | KWKWKWKW |
MCF-7 cel | 28933182 | 1.85 | 50.0 | 120.0 | KWKWKWKW | KWKWKWKW |
MCF-7 cel | 28933182 | 1.78 | 10.0 | 120.0 | KWKWKWKWKW | KWKWKWKWKW |
MCF-7 cel | 28933182 | 1.95 | 25.0 | 120.0 | KWKWKWKWKW | KWKWKWKWKW |
MCF-7 cel | 28933182 | 1.88 | 50.0 | 120.0 | KWKWKWKWKW | KWKWKWKWKW |
MCF-7 cel | 28933182 | 1.9 | 10.0 | 120.0 | KKWWWWKK | KKWWWWKK |
MCF-7 cel | 28933182 | 1.95 | 25.0 | 120.0 | KKWWWWKK | KKWWWWKK |
MCF-7 cel | 28933182 | 1.93 | 50.0 | 120.0 | KKWWWWKK | KKWWWWKK |
MCF-7 cel | 28933182 | 1.9 | 10.0 | 120.0 | KKKWWWWKKK | KKKWWWWKKK |
MCF-7 cel | 28933182 | 1.95 | 25.0 | 120.0 | KKKWWWWKKK | KKKWWWWKKK |
MCF-7 cel | 28933182 | 1.95 | 50.0 | 120.0 | KKKWWWWKKK | KKKWWWWKKK |
MCF-7 cel | 28933182 | 1.54 | 10.0 | 120.0 | WWKKKKWW | WWKKKKWW |
MCF-7 cel | 28933182 | 1.3 | 25.0 | 120.0 | WWKKKKWW | WWKKKKWW |
MCF-7 cel | 28933182 | 1.48 | 50.0 | 120.0 | WWKKKKWW | WWKKKKWW |
MCF-7 cel | 28933182 | 1.9 | 10.0 | 120.0 | WWWKKKKWWW | WWWKKKKWWW |
MCF-7 cel | 28933182 | 1.95 | 25.0 | 120.0 | WWWKKKKWWW | WWWKKKKWWW |
MCF-7 cel | 28933182 | 1.93 | 50.0 | 120.0 | WWWKKKKWWW | WWWKKKKWWW |
A549 cells | 28694765 | 1.51 | 10.0 | 90.0 | RWRWRW | RWRWRW |
A549 cells | 28694765 | 1.8 | 25.0 | 90.0 | RWRWRW | RWRWRW |
A549 cells | 28694765 | 1.95 | 50.0 | 90.0 | RWRWRW | RWRWRW |
A549 cells | 28694765 | 1.76 | 10.0 | 90.0 | RWRWRWRW | RWRWRWRW |
A549 cells | 28694765 | 1.9 | 25.0 | 90.0 | RWRWRWRW | RWRWRWRW |
A549 cells | 28694765 | 1.9 | 50.0 | 90.0 | RWRWRWRW | RWRWRWRW |
A549 cells | 28694765 | 1.78 | 10.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A549 cells | 28694765 | 1.85 | 25.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A549 cells | 28694765 | 1.9 | 50.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A549 cells | 28694765 | 1.67 | 10.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
A549 cells | 28694765 | 1.77 | 25.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
A549 cells | 28694765 | 1.94 | 50.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
HCT116 cells | 33141296 | 1.0 | 0.1 | 0.0 | LKRLRRRYKFRHRRRQRYRRR | LKRLRRRYKFRHRRRQRYRRR |
HCT116 cells | 33141296 | 1.88 | 1.0 | 0.0 | LKRLRRRYKFRHRRRQRYRRR | LKRLRRRYKFRHRRRQRYRRR |
HCT116 cells | 33141296 | 2.0 | 10.0 | 0.0 | LKRLRRRYKFRHRRRQRYRRR | LKRLRRRYKFRHRRRQRYRRR |
HCT116 cells | 33141296 | 1.94 | 10.0 | 0.0 | LKRLRRRYKFRHRRRQRYRRR | LKRLRRRYKFRHRRRQRYRRR |
Caski cells | 30230543 | 2.54 | 2.5 | 60.0 | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Caski cells | 30230543 | 3.04 | 5.0 | 60.0 | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Caski cells | 30230543 | 3.13 | 7.5 | 60.0 | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
Caski cells | 30230543 | 3.15 | 10.0 | 60.0 | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR | VSRRRRRRGGRRRRGGGSYARVRRRGPRRGYARVRRRGPRR |
U87 cells | 29686590 | 4.15 | 10.0 | 60.0 | CREKAPLGLAGRKKRRQRRRC | CREKAPLGLAGRKKRRQRRRC |
U87 cells | 29686590 | 3.41 | 10.0 | 60.0 | CREKAPLGLAGRKKRRQRRRC | CREKAPLGLAGRKKRRQRRRC |
HeLa cells | 30367921 | -1.3 | 10.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
HeLa cells | 30367921 | 0.0 | 1.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
HeLa cells | 30367921 | -0.19 | 10.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -1.0 | 1.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -1.3 | 10.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
HeLa cells | 30367921 | 0.0 | 1.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
HeLa cells | 30367921 | -0.1 | 10.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -1.0 | 1.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -1.3 | 10.0 | 30.0 | KQRFIR | KQRFIR |
HeLa cells | 30367921 | 0.0 | 1.0 | 30.0 | KQRFIR | KQRFIR |
HeLa cells | 30367921 | -0.12 | 10.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -1.1 | 1.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -0.4 | 10.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -0.82 | 1.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | -0.7 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
HeLa cells | 30367921 | 0.0 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -2.0 | 10.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
MCF-7 cells | 30367921 | -2.0 | 1.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
MCF-7 cells | 30367921 | -0.46 | 10.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.1 | 1.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.7 | 10.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
MCF-7 cells | 30367921 | -2.0 | 1.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
MCF-7 cells | 30367921 | -0.1 | 10.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.3 | 1.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.4 | 10.0 | 30.0 | KQRFIR | KQRFIR |
MCF-7 cells | 30367921 | 0.0 | 1.0 | 30.0 | KQRFIR | KQRFIR |
MCF-7 cells | 30367921 | -0.1 | 10.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.3 | 1.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -0.82 | 10.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.1 | 1.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | -1.0 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MCF-7 cells | 30367921 | 0.0 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -2.0 | 10.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
TDA cells | 30367921 | 0.0 | 1.0 | 30.0 | LSRTRAAAPNSRIFTR | LSRTRAAAPNSRIFTR |
TDA cells | 30367921 | -0.7 | 10.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -1.0 | 1.0 | 30.0 | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK | LSRTRAAAPNSRIFTRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -2.0 | 10.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
TDA cells | 30367921 | 0.0 | 1.0 | 30.0 | LRSSVVRSRATLR | LRSSVVRSRATLR |
TDA cells | 30367921 | -0.7 | 10.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -1.0 | 1.0 | 30.0 | LRSSVVRSRATLRGLRKRLRKFRNKIKEK | LRSSVVRSRATLRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -2.0 | 10.0 | 30.0 | KQRFIR | KQRFIR |
TDA cells | 30367921 | 0.0 | 1.0 | 30.0 | KQRFIR | KQRFIR |
TDA cells | 30367921 | -0.52 | 10.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -1.1 | 1.0 | 30.0 | KQRFIRGLRKRLRKFRNKIKEK | KQRFIRGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -0.6 | 10.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -0.7 | 1.0 | 30.0 | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK | SEEIITPVYCTGVSAQVQKGLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -0.82 | 10.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
TDA cells | 30367921 | -1.3 | 1.0 | 30.0 | GLRKRLRKFRNKIKEK | GLRKRLRKFRNKIKEK |
MDA-MB-435S cells | 31714739 | 3.78 | 2.0 | 60.0 | KWCFRVCYRGICYRRCR | KWCFRVCYRGICYRRCR |
MDA-MB-435S cells | 31714739 | 3.0 | 2.0 | 60.0 | KWCFRVCYRGICYRRCRG | KWCFRVCYRGICYRRCRG |
MDA-MB-435S cells | 31714739 | 3.7 | 2.0 | 60.0 | KWCFRVCSRGSCYRRCRG | KWCFRVCSRGSCYRRCRG |
MDA-MB-435S cells | 31714739 | 2.7 | 2.0 | 60.0 | KWCSRVCYRGICSRRCRG | KWCSRVCYRGICSRRCRG |
MM96L cells | 31714739 | 3.74 | 2.0 | 60.0 | KWCFRVCYRGICYRRCR | KWCFRVCYRGICYRRCR |
MM96L cells | 31714739 | 3.4 | 2.0 | 60.0 | KWCFRVCYRGICYRRCRG | KWCFRVCYRGICYRRCRG |
MM96L cells | 31714739 | 3.65 | 2.0 | 60.0 | KWCFRVCSRGSCYRRCRG | KWCFRVCSRGSCYRRCRG |
MM96L cells | 31714739 | 3.3 | 2.0 | 60.0 | KWCSRVCYRGICSRRCRG | KWCSRVCYRGICSRRCRG |
HeLa cells | 31714739 | 3.48 | 2.0 | 60.0 | KWCFRVCYRGICYRRCR | KWCFRVCYRGICYRRCR |
HeLa cells | 31714739 | 3.0 | 2.0 | 60.0 | KWCFRVCYRGICYRRCRG | KWCFRVCYRGICYRRCRG |
HeLa cells | 31714739 | 3.3 | 2.0 | 60.0 | KWCFRVCSRGSCYRRCRG | KWCFRVCSRGSCYRRCRG |
HeLa cells | 31714739 | 2.7 | 2.0 | 60.0 | KWCSRVCYRGICSRRCRG | KWCSRVCYRGICSRRCRG |
HaCaT cells | 31714739 | 3.4 | 2.0 | 60.0 | KWCFRVCYRGICYRRCR | KWCFRVCYRGICYRRCR |
HaCaT cells | 31714739 | 3.18 | 2.0 | 60.0 | KWCFRVCYRGICYRRCRG | KWCFRVCYRGICYRRCRG |
HaCaT cells | 31714739 | 3.3 | 2.0 | 60.0 | KWCFRVCSRGSCYRRCRG | KWCFRVCSRGSCYRRCRG |
HaCaT cells | 31714739 | 3.0 | 2.0 | 60.0 | KWCSRVCYRGICSRRCRG | KWCSRVCYRGICSRRCRG |
MCF7 cells | 33533253 | 0.7 | 2.0 | 60.0 | LTFKEYWDQLTSAA | LTFKEYWDQLTSAA |
HeLa cells | 33533253 | 0.48 | 2.0 | 60.0 | LTFKEYWDQLTSAA | LTFKEYWDQLTSAA |
MCF7 cells | 33533253 | 0.0 | 2.0 | 120.0 | LTFKEYWDQLTSAA | LTFKEYWDQLTSAA |
HeLa cells | 33533253 | -0.7 | 2.0 | 120.0 | LTFKEYWDQLTSAA | LTFKEYWDQLTSAA |
HeLa cells | 29977402 | 4.18 | 10.0 | 30.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
HeLa cells | 29977402 | 3.85 | 10.0 | 120.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
HeLa cells | 29977402 | 3.0 | 10.0 | 30.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
HeLa cells | 29977402 | 4.11 | 10.0 | 30.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
HeLa cells | 29977402 | 4.0 | 10.0 | 120.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
HeLa cells | 29977402 | 3.46 | 10.0 | 30.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
MCF7 cells | 29977402 | 4.23 | 10.0 | 30.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
MCF7 cells | 29977402 | 4.11 | 10.0 | 120.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
MCF7 cells | 29977402 | 4.2 | 10.0 | 30.0 | VQRKRQKLMPGLRKRLRKFRNK | VQRKRQKLMPGLRKRLRKFRNK |
MCF7 cells | 29977402 | 4.32 | 10.0 | 30.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
MCF7 cells | 29977402 | 3.85 | 10.0 | 120.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
MCF7 cells | 29977402 | 3.88 | 10.0 | 30.0 | YKQCHKKGGKKGSGGLRKRLRKFRNK | YKQCHKKGGKKGSGGLRKRLRKFRNK |
HEK293 cells | 33866927 | 2.18 | 10.0 | 30.0 | LKPSFSPRNY | LKPSFSPRNY |
HEK293 cells | 33866927 | 1.9 | 10.0 | 30.0 | KALSEVQGWKQRMAAKELAR | KALSEVQGWKQRMAAKELAR |
HEK293 cells | 33866927 | 2.18 | 10.0 | 30.0 | KQRMAAKELAR | KQRMAAKELAR |
3T3-L1 cells | 33866927 | 3.4 | 10.0 | 30.0 | LKPSFSPRNY | LKPSFSPRNY |
3T3-L1 cells | 33866927 | 3.3 | 10.0 | 30.0 | KALSEVQGWKQRMAAKELAR | KALSEVQGWKQRMAAKELAR |
3T3-L1 cells | 33866927 | 3.3 | 10.0 | 30.0 | KQRMAAKELAR | KQRMAAKELAR |
A549 cells | 27074859 | 1.81 | 10.0 | 90.0 | RRRRRRRRR | RRRRRRRRR |
A549 cells | 27074859 | 1.85 | 10.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
A549 cells | 27074859 | 1.86 | 10.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A549 cells | 27074859 | 1.86 | 25.0 | 90.0 | RRRRRRRRR | RRRRRRRRR |
A549 cells | 27074859 | 1.9 | 25.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
A549 cells | 27074859 | 1.9 | 25.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A549 cells | 27074859 | 1.94 | 50.0 | 90.0 | RRRRRRRRR | RRRRRRRRR |
A549 cells | 27074859 | 1.98 | 50.0 | 90.0 | RRRRRWWWRRRR | RRRRRWWWRRRR |
A549 cells | 27074859 | 1.93 | 50.0 | 90.0 | RWRWRWRWRWRW | RWRWRWRWRWRW |
A375 cells | 31672541 | 1.4 | 5.0 | 120.0 | GGLIKTKRKRKKQRVKIAYEEIFVKNM | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
A375 cells | 31672541 | 0.9 | 5.0 | 120.0 | GGLIKTKRKRKKQRVKIAYEEIFVKNM | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
HeLa cells | 31672541 | 1.54 | 5.0 | 120.0 | GGLIKTKRKRKKQRVKIAYEEIFVKNM | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
HeLa cells | 31672541 | 1.26 | 5.0 | 120.0 | GGLIKTKRKRKKQRVKIAYEEIFVKNM | GGLIKTKRKRKKQRVKIAYEEIFVKNM |
HeLa cells | 28096156 | 1.26 | 1.0 | 120.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HeLa cells | 28096156 | 1.26 | 1.0 | 240.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HeLa cells | 28096156 | 1.28 | 1.0 | 360.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HeLa cells | 28096156 | 1.08 | 1.0 | 1440.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HeLa cells | 28096156 | 1.11 | 1.0 | 120.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HeLa cells | 28096156 | 1.15 | 1.0 | 240.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HeLa cells | 28096156 | 1.08 | 1.0 | 360.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HeLa cells | 28096156 | 0.9 | 1.0 | 1440.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HBMEC cells | 28096156 | 1.4 | 1.0 | 120.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HBMEC cells | 28096156 | 1.48 | 1.0 | 240.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HBMEC cells | 28096156 | 1.36 | 1.0 | 360.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HBMEC cells | 28096156 | 1.48 | 1.0 | 1440.0 | KSKTEYYNAWAVWERNAP | KSKTEYYNAWAVWERNAP |
HBMEC cells | 28096156 | 1.6 | 1.0 | 120.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HBMEC cells | 28096156 | 1.65 | 1.0 | 240.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HBMEC cells | 28096156 | 1.54 | 1.0 | 360.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HBMEC cells | 28096156 | 1.6 | 1.0 | 1440.0 | GNGEQREMAVSRLRDCLDRQA | GNGEQREMAVSRLRDCLDRQA |
HeLa cells | 33355559 | 2.0 | 2.0 | 120.0 | YGRKKRRQRRR | YGRKKRRQRRR |
HeLa cells | 33355559 | 1.9 | 2.0 | 120.0 | YGRKERRQKRR | YGRKERRQKRR |
human endothelial cells | 26748549 | 1.26 | 10.0 | 240.0 | RRRRRRRRR | RRRRRRRRR |
human endothelial cells | 26748549 | 1.54 | 25.0 | 240.0 | RRRRRRRRR | RRRRRRRRR |
human endothelial cells | 26748549 | 1.7 | 50.0 | 240.0 | RRRRRRRRR | RRRRRRRRR |
MCF-7 cells | 25853477 | 1.3 | 7.0 | 180.0 | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
MCF-7 cells | 25853477 | 1.6 | 7.0 | 180.0 | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
MCF-7/Adr cells | 25853477 | 1.38 | 7.0 | 180.0 | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
MCF-7/Adr cells | 25853477 | 1.54 | 7.0 | 180.0 | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG | AEQNPIYWARYADWLFTTPLLLLDLALLVDADEGTCG |
ECV304 cells | 27070736 | 3.48 | 2.5 | 60.0 | KPKRKRRKKKGHGWSR | KPKRKRRKKKGHGWSR |
ECV304 cells | 27070736 | 3.7 | 5.0 | 60.0 | KPKRKRRKKKGHGWSR | KPKRKRRKKKGHGWSR |
ECV304 cells | 27070736 | 3.72 | 7.5 | 60.0 | KPKRKRRKKKGHGWSR | KPKRKRRKKKGHGWSR |
ECV304 cells | 27070736 | 3.76 | 10.0 | 60.0 | KPKRKRRKKKGHGWSR | KPKRKRRKKKGHGWSR |
RAW264.7 cells | 30095906 | 1.86 | 5.0 | 120.0 | GFAWNVCVYRNGVRVCHRRAN | GFAWNVCVYRNGVRVCHRRAN |
HeLa cells | 28459137 | 1.6 | 6.0 | 60.0 | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
HeLa cells | 28459137 | 1.58 | 6.0 | 60.0 | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
HeLa cells | 28459137 | 1.69 | 6.0 | 60.0 | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR | MCMPCFTTDHQMARRCDDCCGGRGRGKCYGPQCLCR |
HeLa cells | 28459137 | 1.88 | 6.0 | 60.0 | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR | MCMPCFTTDHQMARRCDDCCGGRGRGKCWGPQCLCR |
HeLa cells | 29026300 | 1.8 | 10.0 | 30.0 | RRRRQWWQW | RRRRQWWQW |
HeLa cells | 29026300 | 1.87 | 100.0 | 30.0 | RRRRQWWQW | RRRRQWWQW |
BCECs cells | 32674358 | -1.7 | 100.0 | 180.0 | KLSSIESDV | KLSSIESDV |
BCECs cells | 32674358 | -1.05 | 100.0 | 180.0 | YGRKKRRQRRRKLSSIESDV | YGRKKRRQRRRKLSSIESDV |
U87 cells | 30243823 | 3.18 | 1.0 | 240.0 | KLKLALALALAVQRKRQKLMPC | KLKLALALALAVQRKRQKLMPC |
U87 cells | 30243823 | 2.7 | 0.1 | 240.0 | KLKLALALALAVQRKRQKLMPC | KLKLALALALAVQRKRQKLMPC |
U87 cells | 30243823 | 1.85 | 0.01 | 240.0 | KLKLALALALAVQRKRQKLMPC | KLKLALALALAVQRKRQKLMPC |
A2780 cells | 26784985 | 1.62 | 5.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
A2780 cells | 26784985 | 1.89 | 10.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
A2780 cells | 26784985 | 2.0 | 15.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
A2780 cells | 26784985 | 2.06 | 20.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
A2780 cells | 26784985 | 2.08 | 25.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
A2780 cells | 26784985 | 2.11 | 30.0 | 60.0 | CRRRRRRRRVKRKKKP | CRRRRRRRRVKRKKKP |
MDA-MB-231 cells | 35839086 | 2.7 | 10.0 | 240.0 | KRKIFCL | KRKIFCL |
MDA-MB-231 cells | 35839086 | 2.6 | 10.0 | 240.0 | KRKIFCL | KRKIFCL |
MDA-MB-231 cells | 35839086 | 2.9 | 10.0 | 240.0 | KRKIFCL | KRKIFCL |
MDA-MB-231 cells | 35839086 | 3.3 | 10.0 | 240.0 | KRKIFCL | KRKIFCL |
NIH-3T3 fibroblast cells | 35752142 | 3.85 | 2.5 | 1080.0 | CRWRWKCCKK | CRWRWKCCKK |
Jurkat | 11087855 | 3.26 | 12.5 | 15.0 | Ahx-rkkrrqrrr | KRKKRRQRRR |
Jurkat | 11087855 | 3.56 | 12.5 | 15.0 | Ahx-rrrqrrkkr | KRRRQRRKKR |
Jurkat | 11087855 | 2.18 | 12.5 | 15.0 | Ahx-rrrrr | KRRRRR |
Jurkat | 11087855 | 2.98 | 12.5 | 15.0 | Ahx-rrrrrr | KRRRRRR |
Jurkat | 11087855 | 3.49 | 12.5 | 15.0 | Ahx-rrrrrrr | KRRRRRRR |
Jurkat | 11087855 | 3.64 | 12.5 | 15.0 | Ahx-rrrrrrrr | KRRRRRRRR |
Jurkat | 11087855 | 3.71 | 12.5 | 15.0 | Ahx-rrrrrrrrr | KRRRRRRRRR |
NIH-3T3 | 21319732 | 3.29 | 2.5 | 1080.0 | MDCRWRWK-Abu-CKK | MDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.24 | 2.5 | 1080.0 | DCRWRWK-Abu-CKK | DCRWRWKCCKK |
NIH-3T3 | 21319732 | 2.97 | 2.5 | 1080.0 | DCRWRWKC-Abu-KK | DCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.31 | 2.5 | 1080.0 | CRWRWK-Abu-CKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.13 | 2.5 | 1080.0 | CRWRWKC-Abu-KK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.08 | 2.5 | 1080.0 | RWRWK-Abu-CKK | RWRWKCCKK |
NIH-3T3 | 21319732 | 3.1 | 2.5 | 1080.0 | MDCRWRWK-Abu-Abu-KK | MDCRWRWKCCKK |
NIH-3T3 | 21319732 | 2.94 | 2.5 | 1080.0 | DCRWRWK-Abu-Abu-KK | DCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.14 | 2.5 | 1080.0 | CRWRWK-Abu-Abu-KK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 2.61 | 2.5 | 1080.0 | RWRWK-Abu-Abu-KK | RWRWKCCKK |
NIH-3T3 | 21319732 | 3.32 | 2.5 | 1080.0 | crwrwkcckk | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.16 | 2.5 | 1080.0 | kcckwrwrck | KCCKWRWRCK |
NIH-3T3 | 21319732 | 3.18 | 2.5 | 1080.0 | CrWRWKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.09 | 2.5 | 1080.0 | CRwRWKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.12 | 2.5 | 1080.0 | CRWrWKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.15 | 2.5 | 1080.0 | CRWRwKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.17 | 2.5 | 1080.0 | CrwrwKCCKK | CRWRWKCCKK |
NIH-3T3 | 21319732 | 3.29 | 2.5 | 1080.0 | KMD-Abu-RWRWKCCKK | KMDCRWRWKCCKK |
NIH-3T3 | 21319732 | 2.87 | 2.5 | 1080.0 | KMD-Abu-RWRWK-Abu-CKK | KMDCRWRWKCCKK |
NIH-3T3 | 21319732 | 2.21 | 2.5 | 1080.0 | KMD-Abu-RWRWK-Abu-Abu-KK | KMDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.45 | 2.5 | 1080.0 | KMD-Abu-RWRWKC-Abu-KK | KMDCRWRWKCCKK |
NIH-3T3 | 21319732 | 3.19 | 2.5 | 1080.0 | MDCRWRWKC-Abu-KK | MDCRWRWKCCKK |
NIH-3T3 | 21319732 | 2.4 | 2.5 | 1080.0 | KMD-Abu-RPRPKCCKK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 2.35 | 2.5 | 1080.0 | KMD-Abu-RPRPK-Abu-CKK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 2.41 | 2.5 | 1080.0 | KMD-Abu-RPRPKC-Abu-KK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 2.47 | 2.5 | 1080.0 | KMDCRPRPK-Abu-CKK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 2.55 | 2.5 | 1080.0 | KMDCRPRPKC-Abu-KK | KMDCRPRPKCCKK |
NIH-3T3 | 21319732 | 1.74 | 2.5 | 1080.0 | rkkrrqrrr | RKKRRQRRR |
NIH-3T3 | 21319732 | 1.67 | 2.5 | 1080.0 | rrrqrrkkr | RRRQRRKKR |
NIH-3T3 | 21319732 | 1.68 | 2.5 | 1080.0 | rrrrrrrr | RRRRRRRR |
K562 cells | 12783857 | 0.88 | 6.0 | 65.0 | rggrlsysrrrfststgr | RGGRLSYSRRRFSTSTGR |
K562 cells | 12783857 | 1.24 | 6.0 | 65.0 | rrlsysrrrf | RRLSYSRRRF |
A549 | 21875799 | 2.2 | 2.0 | 360.0 | Ac-KL-Aib-LKL-Aib-LK-Aib-LKA-Aib-LKL-Aib-GC-NH2 | GKLALKLALKALKAALKLAGC |
HeLa | 25188671 | -0.64 | 0.1 | 120.0 | gRLLRLLRL-Ac5c-NH2 | GRLLRLLRLP |
HeLa | 25188671 | -0.64 | 0.1 | 120.0 | gRLLRL-Ac5c-RL-Ac5c-NH2 | GRLLRLPRLP |
HeLa | 25188671 | -0.07 | 0.1 | 120.0 | gRL-Ac5c-RL-Ac5c-RL-Ac5c-NH2 | GRLPRLPRLP |
HeLa | 24270856 | 1.93 | 5.0 | 30.0 | K-Hcy-FQWQRNMRKVRGPPVS-Hcy-IKR-NH2 | KCFQWQRNMRKVRGPPVSCIKR |
HeLa | 24661993 | 3.18 | 3.0 | 120.0 | betaA-RR-Aib-RR-Aib-RR-Aib | ARRARRARRA |
HeLa | 24661993 | 3.29 | 3.0 | 120.0 | betaA-rr-Aib-rr-Aib-rr-Aib | ARRARRARRA |
HeLa | 24661993 | 2.93 | 3.0 | 120.0 | betaA-Rr-Aib-Rr-Aib-Rr-Aib | ARRARRARRA |
HeLa | 24896852 | 3.55 | 10.0 | 120.0 | F-LNap-RRRRQ-miniPEG_linker-DELI-NH2 | FARRRRQADELI |
HepG2 | 24811205 | 3.5 | 10.0 | 180.0 | lclr | LCLR |
HepG2 | 24811205 | 3.22 | 10.0 | 180.0 | lcl | LCL |
HepG2 | 24811205 | 2.88 | 10.0 | 180.0 | icir | ICIR |
HepG2 | 24811205 | 2.7 | 10.0 | 180.0 | vcvr | VCVR |
HepG2 | 24811205 | 3.06 | 10.0 | 180.0 | vlclr | VLCLR |
Murine H2k mdx myoblasts | 24366877 | 4.11 | 1.0 | 240.0 | Ac-R-Ahx-RR-betaA-RR-Ahx-RYQFLIR-Ahx-R-betaA-R-Ahx-R-betaA | GRKRRARRKRYQFLIRKRARKRA |
C2C12 cells | 24366877 | 3.9 | 1.0 | 240.0 | Ac-R-Ahx-RR-betaA-RR-Ahx-RYQFLIR-Ahx-R-betaA-R-Ahx-R-betaA | GRKRRARRKRYQFLIRKRARKRA |
MCF-7 cells | 24480922 | 3.25 | 25.0 | 180.0 | CREKAKKLFKKILKKL-NH2 | CREKAKKLFKKILKKL |
mouse embryonic fibroblast 3T3 | 24480922 | 3.11 | 25.0 | 180.0 | CREKAKKLFKKILKKL-NH2 | CREKAKKLFKKILKKL |
MCF-7 cells | 24480922 | 3.6 | 25.0 | 180.0 | CREKAKKLFKKILKKL-NH2 | CREKAKKLFKKILKKL |
HeLa | 24985034 | 0.07 | 16.0 | 60.0 | grctksippicfpd | GRCTKSIPPICFPD |
HeLa | 24985034 | 0.05 | 16.0 | 60.0 | GR-Abu-TKSIPPI-Abu-FPD | GRCTKSIPPICFPD |
HeLa | 24985034 | -0.09 | 16.0 | 60.0 | GR-Abu-TKSIPPI-Abu-FPD | GRCTKSIPPICFPD |
CHO-K1 | 25096299 | 1.81 | 10.0 | 240.0 | R-aeLP-RR-aeLP-RR-aeLP-RR-aeLP-R-NH2 | RAELPRRAELPRRAELPRRAELPR |
CHO-K1 | 25096299 | 1.85 | 10.0 | 240.0 | R-aeDP-RR-aeDP-RR-aeDP-RR-aeDP-R-NH2 | RAEDPRRAEDPRRAEDPRRAEDPR |
CHO-K1 | 25096299 | 1.93 | 10.0 | 240.0 | R-apLP-RR-apLP-RR-apLP-RR-apLP-R-NH2 | RAPLPRRAPLPRRAPLPRRAPLPR |
CHO-K1 | 25096299 | 1.88 | 10.0 | 240.0 | R-apDP-RR-apDP-RR-apDP-RR-apDP-R-NH2 | RAPDPRRAPDPRRAPDPRRAPDPR |
CHO-K1 | 25096299 | 1.49 | 10.0 | 240.0 | R-Ahx-RR-Ahx-RR-Ahx-RR-Ahx-R-NH2 | RKRRKRRKRRKR |
ARPE-19 | 22100438 | -0.06 | 2.1 | 30.0 | CGRKKRRQRR-Ahx-RPPQ | CGRKKRRQRRKRPPQ |
CHO wt | 22100438 | -0.08 | 2.1 | 30.0 | CGRKKRRQRR-Ahx-RPPQ | CGRKKRRQRRKRPPQ |
CHO pgsB-618 cells | 22100438 | -0.12 | 2.1 | 30.0 | CGRKKRRQRR-Ahx-RPPQ | CGRKKRRQRRKRPPQ |
ARPE-19 | 22100438 | -0.01 | 2.1 | 30.0 | CGRKKR-Ahx-RQRRRPPQ | CGRKKRKRQRRRPPQ |
CHO wt | 22100438 | -0.06 | 2.1 | 30.0 | CGRKKR-Ahx-RQRRRPPQ | CGRKKRKRQRRRPPQ |
CHO pgsB-618 cells | 22100438 | -0.12 | 2.1 | 30.0 | CGRKKR-Ahx-RQRRRPPQ | CGRKKRKRQRRRPPQ |
ARPE-19 | 22100438 | 0.03 | 2.1 | 30.0 | CGRKKRRQR-Ahx-RRPPQ | CGRKKRRQRKRRPPQ |
CHO wt | 22100438 | -0.05 | 2.1 | 30.0 | CGRKKRRQR-Ahx-RRPPQ | CGRKKRRQRKRRPPQ |
CHO pgsB-618 cells | 22100438 | -0.07 | 2.1 | 30.0 | CGRKKRRQR-Ahx-RRPPQ | CGRKKRRQRKRRPPQ |
ARPE-19 | 22100438 | -0.05 | 2.1 | 30.0 | CGRKKR-Ahx-RQR-Ahx-R-Ahx-RPPQ | CGRKKRKRQRKRKRPPQ |
CHO wt | 22100438 | -0.13 | 2.1 | 30.0 | CGRKKR-Ahx-RQR-Ahx-R-Ahx-RPPQ | CGRKKRKRQRKRKRPPQ |
CHO pgsB-618 cells | 22100438 | -0.11 | 2.1 | 30.0 | CGRKKR-Ahx-RQR-Ahx-R-Ahx-RPPQ | CGRKKRKRQRKRKRPPQ |
U373 MG cells | 22148546 | 2.0 | 5.0 | 60.0 | inlkalaalakkil | INLKALAALAKKIL |
U373 MG cells | 22148546 | 0.9 | 5.0 | 60.0 | likkalaalaklni | LIKKALAALAKLNI |
U373 MG cells | 22148546 | 1.91 | 5.0 | 60.0 | INLKKLAKL-Aib-KKIL | INLKKLAKLAKKIL |
U373 MG cells | 22148546 | 1.8 | 5.0 | 60.0 | inlkklakl-Aib-kkil | INLKKLAKLAKKIL |
U373 MG cells | 22148546 | 1.17 | 5.0 | 60.0 | LIKK-Aib-LKALKKLNI | LIKKALKALKKLNI |
U373 MG cells | 22148546 | 1.37 | 5.0 | 60.0 | likk-Aib-lkalkklni | LIKKALKALKKLNI |
CHO-K1 | 22509923 | 2.56 | 5.0 | 60.0 | r-ahx-rr-ahx-rr-ahx-rr-ahx-r-Cbz | RAHRRAHRRAHRRAHRA |
CHO-K1 | 22509923 | 2.48 | 5.0 | 60.0 | rrrrrrrr-Cbz | RRRRRRRRA |
A549 cells | 25468041 | 1.18 | 10.0 | 120.0 | Ac-Aib-NII-Aib-PLL-Aib-PIC-NH2 | GANIIAPLLAPIC |
A549 cells | 25468041 | 0.0 | 10.0 | 120.0 | Ac-Aib-NII-Aib-PLL-A-PIC-NH2 | GANIIAPLLAPIC |
A549 cells | 25468041 | 0.7 | 10.0 | 120.0 | Ac-A-NII-Aib-PLL-Aib-PIC-NH2 | GANIIAPLLAPIC |
A549 cells | 25468041 | 0.4 | 10.0 | 120.0 | Ac-Aib-NII-A-PLL-Aib-PIC-NH2 | GANIIAPLLAPIC |
A549 cells | 25468041 | 2.51 | 10.0 | 120.0 | Ac-Aib-NII-Aib-Aib-LL-Aib-Aib-IC-NH2 | GANIIAALLAAIC |
A549 cells | 25468041 | 1.3 | 10.0 | 120.0 | Ac-Aib-NII-Aib-PLL-Aib-Aib-IC-NH2 | GANIIAPLLAAIC |
A549 cells | 25468041 | 1.26 | 10.0 | 120.0 | Ac-Aib-NII-Aib-Aib-LL-Aib-PIC-NH2 | GANIIAALLAPIC |
Cal 27 | 31450798 | -0.26 | 10.0 | 120.0 | 4Iph-TSPLNIHNGQKL | ATSPLNIHNGQKL |
Cal 27 | 31450798 | 0.0 | 10.0 | 120.0 | Fmoc-TSPLNIHNGQKL | WTSPLNIHNGQKL |
Cal 27 | 31450798 | -0.52 | 10.0 | 120.0 | NQHSKNTLLIGP | NQHSKNTLLIGP |
Cal 27 | 31450798 | 0.65 | 10.0 | 120.0 | 4Iph_yl-Fmoc-LPNSNHIKQGL | AWLPNSNHIKQGL |
Cal 27 | 31450798 | 0.23 | 10.0 | 120.0 | Fmoc-TLPNSNHIKQGL | WTLPNSNHIKQGL |
Saos-2 cells | 30410976 | -3.76 | 1.0 | 30.0 | f-LNap-RrRrQ-PEG2 | FARRRRQA |
Saos-2 cells | 30410976 | -3.4 | 1.0 | 30.0 | Ff-LNap-RrRrQ-PEG2 | FFARRRRQA |
HepG2 | 35024246 | 3.56 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
HepG2 | 35024246 | 3.2 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
HepG2 | 35024246 | 3.32 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
HepG2 | 35024246 | 3.41 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
HepG2 | 35024246 | 3.59 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
RAW 264.7 | 35024246 | 3.08 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
RAW 264.7 | 35024246 | 2.88 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
RAW 264.7 | 35024246 | 2.94 | 100.0 | 240.0 | CKRRMKWKK | CKRRMKWKK |
HeLa | 30718681 | 2.26 | 1.0 | 120.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
HeLa | 30718681 | 2.26 | 1.0 | 360.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
HeLa | 30718681 | 1.48 | 1.0 | 1440.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
HeLa | 30718681 | 1.48 | 1.0 | 120.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
HeLa | 30718681 | 1.54 | 1.0 | 360.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
HeLa | 30718681 | 1.4 | 1.0 | 1440.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
HeLa | 30718681 | 1.85 | 1.0 | 120.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
HeLa | 30718681 | 2.13 | 1.0 | 360.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
HeLa | 30718681 | 2.08 | 1.0 | 1440.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
HeLa | 30718681 | 1.48 | 1.0 | 120.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
HeLa | 30718681 | 1.65 | 1.0 | 360.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
HeLa | 30718681 | 1.78 | 1.0 | 1440.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
HeLa | 30718681 | 1.7 | 1.0 | 120.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
HeLa | 30718681 | 1.85 | 1.0 | 360.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
HeLa | 30718681 | 1.78 | 1.0 | 1440.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.26 | 1.0 | 120.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
CHO-K1 | 30718681 | 1.08 | 1.0 | 360.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
CHO-K1 | 30718681 | 0.0 | 1.0 | 1440.0 | RRRRRRRRR-NH2 | RRRRRRRRR |
CHO-K1 | 30718681 | 0.7 | 1.0 | 120.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 0.7 | 1.0 | 360.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 0.0 | 1.0 | 1440.0 | RRLRRLRRL-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 1.18 | 1.0 | 120.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 1.34 | 1.0 | 360.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 1.04 | 1.0 | 1440.0 | RR-MeLeu-RR-MeLeu-RR-MeLeu-NH2 | RRLRRLRRL |
CHO-K1 | 30718681 | 0.7 | 1.0 | 120.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.04 | 1.0 | 360.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.0 | 1.0 | 1440.0 | RR-Ac5cdOM-RR-Ac5cdOM-RR-Ac5cdOM-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.3 | 1.0 | 120.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.6 | 1.0 | 360.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
CHO-K1 | 30718681 | 1.0 | 1.0 | 1440.0 | RR-Ac5c-RR-Ac5c-RR-Ac5c-NH2 | RRPRRPRRP |
BMDC | 32686113 | 1.0 | 0.5 | 240.0 | FKFEFKFESGSGSGRKKRRQRRRPQ | FKFEFKFESGSGSGRKKRRQRRRPQ |
BMDC | 32686113 | 1.4 | 1.0 | 240.0 | FKFEFKFESGSGSGRKKRRQRRRPQ | FKFEFKFESGSGSGRKKRRQRRRPQ |
BMDC | 32686113 | 1.54 | 2.0 | 240.0 | FKFEFKFESGSGSGRKKRRQRRRPQ | FKFEFKFESGSGSGRKKRRQRRRPQ |
HeLa | 29275934 | 1.7 | 5.0 | 30.0 | RKKRRQRRREIWIAQELRRIGDEFNAYYARLLCCLLRAYYANFEDGIRRLEQAIWIERRRQRRKKR | RKKRRQRRREIWIAQELRRIGDEFNAYYARLLCCLLRAYYANFEDGIRRLEQAIWIERRRQRRKKR |
HeLa | 29275934 | 1.95 | 10.0 | 30.0 | RKKRRQRRREIWIAQELRRIGDEFNAYYARLLC | RKKRRQRRREIWIAQELRRIGDEFNAYYARLLC |
HSC-T6 | 34338123 | 2.9 | 5.0 | 60.0 | KKKKKRFSFKKSFKLSGFSFKKNKK | KKKKKRFSFKKSFKLSGFSFKKNKK |
A549 | 34338123 | 2.88 | 5.0 | 60.0 | KKKKKRFSFKKSFKLSGFSFKKNKK | KKKKKRFSFKKSFKLSGFSFKKNKK |
BV2 | 34338123 | 2.88 | 5.0 | 60.0 | KKKKKRFSFKKSFKLSGFSFKKNKK | KKKKKRFSFKKSFKLSGFSFKKNKK |
MCF7.00 | 34338123 | 2.95 | 5.0 | 60.0 | KKKKKRFSFKKSFKLSGFSFKKNKK | KKKKKRFSFKKSFKLSGFSFKKNKK |
HeLa | 34463179 | 3.23 | 5.0 | 60.0 | RKRRQTSMTDFYHSKRRLIFS | RKRRQTSMTDFYHSKRRLIFS |
MCF7.00 | 34463179 | 3.15 | 5.0 | 60.0 | RKRRQTSMTDFYHSKRRLIFS | RKRRQTSMTDFYHSKRRLIFS |
HepG2 | 34463179 | 3.15 | 5.0 | 60.0 | RKRRQTSMTDFYHSKRRLIFS | RKRRQTSMTDFYHSKRRLIFS |
A549 | 34463179 | 3.0 | 5.0 | 60.0 | RKRRQTSMTDFYHSKRRLIFS | RKRRQTSMTDFYHSKRRLIFS |
HSC-T6 | 34463179 | 2.9 | 5.0 | 60.0 | RKRRQTSMTDFYHSKRRLIFS | RKRRQTSMTDFYHSKRRLIFS |
A375 cells | 30240193 | 1.18 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
A375-R cells | 30240193 | 1.6 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
MSTO cells | 30240193 | 1.11 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
MSTO-R cells | 30240193 | 1.0 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
9L cells | 30240193 | 1.3 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
9L-R cells | 30240193 | 1.3 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
LN18 cells | 30240193 | 1.26 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
U87 cells | 30240193 | 1.56 | 0.001 | 1440.0 | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD | CDAATATRGRSAASRPTERPRAPARSASRPRRPVD |
A375 cells | 30240193 | 0.7 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
A375-R cells | 30240193 | 0.78 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
MSTO cells | 30240193 | 0.6 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
MSTO-R cells | 30240193 | 1.34 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
9L cells | 30240193 | 0.3 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
9L-R cells | 30240193 | 0.9 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
LN18 cells | 30240193 | 1.26 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
U87 cells | 30240193 | 1.0 | 0.001 | 1440.0 | CYGRKKRRQRRR | CYGRKKRRQRRR |
A375 cells | 30240193 | 1.18 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
A375-R cells | 30240193 | 1.3 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
MSTO cells | 30240193 | 1.32 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
MSTO-R cells | 30240193 | 1.3 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
9L cells | 30240193 | 0.48 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
9L-R cells | 30240193 | 0.9 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
LN18 cells | 30240193 | 1.18 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
U87 cells | 30240193 | 1.0 | 0.001 | 1440.0 | CGALFLGWLGAAGSTMGA | CGALFLGWLGAAGSTMGA |
A375 cells | 30240193 | 1.48 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
A375-R cells | 30240193 | 1.88 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
MSTO cells | 30240193 | 1.7 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
9L cells | 30240193 | 1.41 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
9L-R cells | 30240193 | 1.48 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
LN18 cells | 30240193 | 1.65 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
U87 cells | 30240193 | 1.7 | 0.001 | 1440.0 | CPMLKE | CPMLKE |
A375 cells | 30240193 | 1.6 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
A375-R cells | 30240193 | 1.95 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
MSTO cells | 30240193 | 1.6 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
9L cells | 30240193 | 1.74 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
9L-R cells | 30240193 | 2.0 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
LN18 cells | 30240193 | 1.3 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
U87 cells | 30240193 | 1.6 | 0.001 | 1440.0 | CLGTYTQDFNKFHTFPQTAIGVGAP | CLGTYTQDFNKFHTFPQTAIGVGAP |
A375 cells | 30240193 | 0.7 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
A375-R cells | 30240193 | 0.78 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
MSTO cells | 30240193 | 1.0 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
9L cells | 30240193 | 0.3 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
9L-R cells | 30240193 | 0.6 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
LN18 cells | 30240193 | 0.48 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
U87 cells | 30240193 | 1.26 | 0.001 | 1440.0 | CVTVLALGALAGVGVG | CVTVLALGALAGVGVG |
A375 cells | 30240193 | 0.78 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
A375-R cells | 30240193 | 1.0 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
MSTO cells | 30240193 | 1.18 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
MSTO-R cells | 30240193 | 1.26 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
9L cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
9L-R cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
LN18 cells | 30240193 | 0.7 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |
U87 cells | 30240193 | 1.36 | 0.001 | 1440.0 | CAAVALLPAVLLAHLLAP | CAAVALLPAVLLAHLLAP |